Search Count: 25
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Crystal Structure Of Kras-G12D (Gdp-Bound) In Complex With Bbo-11818
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2025-12-03 Classification: ONCOPROTEIN/INHIBITOR Ligands: GDP, MG, A1CG4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-12-03
Ligands: GDP, MG, A1CG4
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Crystal Structure Of Kras-G12D (Gmppnp-Bound) In Complex With Bbo-11818
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.35 Å Release Date: 2025-12-03 Classification: ONCOPROTEIN/INHIBITOR Ligands: GNP, MG, A1CG4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-12-03
Ligands: GNP, MG, A1CG4
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Crystal Structure Of Hras-G12D/Q95H (Gmppnp-Bound) In Complex With Bbo-11818
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2025-12-03 Classification: ONCOPROTEIN Ligands: GNP, MG, A1CG4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-12-03
Ligands: GNP, MG, A1CG4
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Crystal Structure Of P110Alpha-Rbd Covalently Bound To A Breaker Compound Bbo-10203 Via Cys242
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2025-06-25 Classification: ONCOPROTEIN Ligands: A1AIR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-06-25
Ligands: A1AIR
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Crystal Structure Of Active Kras-G12C (Gmppnp-Bound) In Complex With Bbo-8520
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2024-12-18 Classification: ONCOPROTEIN/INHIBITOR Ligands: GNP, MG, Y8N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: GNP, MG, Y8N
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Crystal Structure Of Kras-G12C (Gdp-Bound) In Complex With Bbo-8520
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2024-12-18 Classification: ONCOPROTEIN/INHIBITOR Ligands: GDP, MG, Y8N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: GDP, MG, Y8N
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Crystal Structure Of Human Hras G12C Covalently Bound To Amg 510
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2024-07-31 Classification: ONCOPROTEIN Ligands: GDP, MOV, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-07-31
Ligands: GDP, MOV, MG
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Solution Structures Of Full-Length K-Ras Bound To Gdp
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Organism: Homo sapiens
Method: SOLUTION NMR
Release Date: 2022-06-15
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Crystal Structure Of Wild-Type Kras4B(1-169) In Complex With Gmppnp And Mg Ion
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2021-02-10 Classification: ONCOPROTEIN Ligands: GNP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-02-10
Ligands: GNP, MG
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E. Coli Phosphoenolpyruvate Carboxykinase G209S Mutant Bound To Methanesulfonate
Organism: Escherichia coli (strain k12)
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2018-08-29 Classification: LYASE Ligands: ATP, MG, MN, 03S |
Organism: Escherichia coli (strain k12)
Method: X-RAY DIFFRACTION
Release Date: 2018-08-29
Ligands: ATP, MG, MN, 03S
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E. Coli Phosphoenolpyruvate Carboxykinase G209S K212C Mutant Bound To Thiosulfate
Organism: Escherichia coli (strain k12)
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2018-08-29 Classification: LYASE Ligands: ATP, MG, MN, XE, BTB, THJ |
Organism: Escherichia coli (strain k12)
Method: X-RAY DIFFRACTION
Release Date: 2018-08-29
Ligands: ATP, MG, MN, XE, BTB, THJ
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E. Coli Phosphoenolpyruvate Carboxykinase K212I F216V Mutant Bound To Methanesulfonate
Organism: Escherichia coli (strain k12)
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2018-08-29 Classification: LYASE Ligands: SO4, 03S |
Organism: Escherichia coli (strain k12)
Method: X-RAY DIFFRACTION
Release Date: 2018-08-29
Ligands: SO4, 03S
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E. Coli Phosphoenolpyruvate Carboxykinase G209N Mutant Bound To Thiosulfate
Organism: Escherichia coli (strain k12)
Method: X-RAY DIFFRACTION Resolution:1.44 Å Release Date: 2018-08-29 Classification: LYASE Ligands: ATP, MN, MG, TRS, THJ |
Organism: Escherichia coli (strain k12)
Method: X-RAY DIFFRACTION
Release Date: 2018-08-29
Ligands: ATP, MN, MG, TRS, THJ
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E. Coli Phosphoenolpyruvate Carboxykinase Y207F Mutant Bound To Thiosulfate And Oxaloacetate
Organism: Escherichia coli k-12
Method: X-RAY DIFFRACTION Resolution:1.46 Å Release Date: 2018-08-29 Classification: LYASE Ligands: OAA, THJ |
Organism: Escherichia coli k-12
Method: X-RAY DIFFRACTION
Release Date: 2018-08-29
Ligands: OAA, THJ
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E. Coli Phosphoenolpyruvate Carboxykinase Bound To Thiosulfate
Organism: Escherichia coli k-12
Method: X-RAY DIFFRACTION Resolution:1.33 Å Release Date: 2018-08-29 Classification: LYASE Ligands: THJ |
Organism: Escherichia coli k-12
Method: X-RAY DIFFRACTION
Release Date: 2018-08-29
Ligands: THJ
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Pyrrolopyrimidine Inhibitors Of Dna Gyrase B And Topoisomerase Iv, Part I: Structure Guided Discovery And Optimization Of Dual Targeting Agents With Potent, Broad-Spectrum Enzymatic Activity.
Organism: Enterococcus faecalis
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2013-02-13 Classification: Isomerase/Isomerase inhibitor Ligands: 0WT, GOL |
Organism: Enterococcus faecalis
Method: X-RAY DIFFRACTION
Release Date: 2013-02-13
Ligands: 0WT, GOL
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Pyrrolopyrimidine Inhibitors Of Dna Gyrase B And Topoisomerase Iv, Part I: Structure Guided Discovery And Optimization Of Dual Targeting Agents With Potent, Broad-Spectrum Enzymatic
Organism: Enterococcus faecalis
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2013-02-13 Classification: Isomerase/Isomerase inhibitor Ligands: SUY, GOL |
Organism: Enterococcus faecalis
Method: X-RAY DIFFRACTION
Release Date: 2013-02-13
Ligands: SUY, GOL
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Pyrrolopyrimidine Inhibitors Of Dna Gyrase B And Topoisomerase Iv, Part I: Structure Guided Discovery And Optimization Of Dual Targeting Agents With Potent, Broad-Spectrum Enzymatic Activity
Organism: Enterococcus faecalis
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2013-02-13 Classification: Isomerase/Isomerase inhibitor Ligands: CJC, GOL |
Organism: Enterococcus faecalis
Method: X-RAY DIFFRACTION
Release Date: 2013-02-13
Ligands: CJC, GOL
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Pyrrolopyrimidine Inhibitors Of Dna Gyrase B And Topoisomerase Iv, Part I: Structure Guided Discovery And Optimization Of Dual Targeting Agents With Potent, Broad-Spectrum Enzymatic Activity.
Organism: Enterococcus faecalis
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2013-02-13 Classification: Isomerase/Isomerase inhibitor Ligands: 1A0, TBU |
Organism: Enterococcus faecalis
Method: X-RAY DIFFRACTION
Release Date: 2013-02-13
Ligands: 1A0, TBU
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Pyrrolopyrimidine Inhibitors Of Dna Gyrase B And Topoisomerase Iv, Part I: Structure Guided Discovery And Optimization Of Dual Targeting Agents With Potent, Broad-Spectrum Enzymatic Activity.
Organism: Francisella tularensis subsp. holarctica
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2013-02-13 Classification: isomerase/isomerase inhibitor Ligands: 19Y |
Organism: Francisella tularensis subsp. holarctica
Method: X-RAY DIFFRACTION
Release Date: 2013-02-13
Ligands: 19Y
