Search Count: 13
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Discovery Of An Orally Bioavailable Reversible Covalent Sars-Cov-2 Mpro Inhibitor With Pan-Coronavirus Activity
Organism: Severe acute respiratory syndrome coronavirus 2, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.37 Å Release Date: 2025-08-20 Classification: HYDROLASE/INHIBOTOR Ligands: A1L7M |
Organism: Severe acute respiratory syndrome coronavirus 2, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2025-08-20
Ligands: A1L7M
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Discovery Of An Orally Bioavailable Reversible Covalent Sars-Cov-2 Mpro Inhibitor With Pan-Coronavirus Activity
Organism: Severe acute respiratory syndrome coronavirus 2, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2025-08-20 Classification: HYDROLASE/INHIBITOR |
Organism: Severe acute respiratory syndrome coronavirus 2, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2025-08-20
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Discovery Of An Orally Bioavailable Reversible Covalent Sars-Cov-2 Mpro Inhibitor With Pan-Coronavirus Activity
Organism: Severe acute respiratory syndrome coronavirus 2, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2025-08-20 Classification: HYDROLASE/INHIBITOR |
Organism: Severe acute respiratory syndrome coronavirus 2, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2025-08-20
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Discovery Of An Orally Bioavailable Reversible Covalent Sars-Cov-2 Mpro Inhibitor With Pan-Coronavirus Activity
Organism: Severe acute respiratory syndrome coronavirus 2, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.47 Å Release Date: 2025-08-20 Classification: HYDROLASE/INHIBITOR Ligands: A1L7M |
Organism: Severe acute respiratory syndrome coronavirus 2, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2025-08-20
Ligands: A1L7M
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Discovery Of An Orally Bioavailable Reversible Covalent Sars-Cov-2 Mpro Inhibitor With Pan-Coronavirus Activity
Organism: Severe acute respiratory syndrome coronavirus 2, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2025-08-20 Classification: HYDROLASE/INHIBITOR Ligands: A1L7M |
Organism: Severe acute respiratory syndrome coronavirus 2, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2025-08-20
Ligands: A1L7M
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Structure Of Rat Beta-Arrestin 1 By Fiducial-Assisted Cryo-Em
Organism: Homo sapiens, Rattus norvegicus
Method: ELECTRON MICROSCOPY Release Date: 2025-01-22 Classification: SIGNALING PROTEIN/Immune System |
Organism: Homo sapiens, Rattus norvegicus
Method: ELECTRON MICROSCOPY
Release Date: 2025-01-22
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Structure Of Rat Beta-Arrestin 1 Bound To Allosteric Inhibitor
Organism: Homo sapiens, Rattus norvegicus
Method: ELECTRON MICROSCOPY Release Date: 2025-01-22 Classification: SIGNALING PROTEIN/Immune System Ligands: ODN |
Organism: Homo sapiens, Rattus norvegicus
Method: ELECTRON MICROSCOPY
Release Date: 2025-01-22
Ligands: ODN
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Solution Nmr Structure Of Vibrio Cholerae Ferrous Iron Transport Protein C (Feoc)
Organism: Vibrio cholerae o1
Method: SOLUTION NMR Release Date: 2022-07-13 Classification: CYTOSOLIC PROTEIN |
Organism: Vibrio cholerae o1
Method: SOLUTION NMR
Release Date: 2022-07-13
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Fragment-Based Lead Discovery Of Indazole-Based Compounds As Axl Kinase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.15 Å Release Date: 2021-10-13 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: E56 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-13
Ligands: E56
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Crystal Structure Of Smyd3 In Complex With Covalent Inhibitor 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2019-08-14 Classification: TRANSFERASE/INHIBITOR Ligands: A8U, ZN, SAM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-14
Ligands: A8U, ZN, SAM
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Crystal Structure Of Smyd3 In Complex With Covalent Inhibitor 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2018-10-17 Classification: TRANSFERASE/INHIBITOR Ligands: ZN, 8W0, SAM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-17
Ligands: ZN, 8W0, SAM
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Structure Of Ppargamma Ligand Binding Domain-Pioglitazone Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2017-12-20 Classification: TRANSCRIPTION Ligands: 8N6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-20
Ligands: 8N6
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Structure Of Ppargamma Ligand Binding Domain - Lobeglitazone Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2017-12-20 Classification: TRANSCRIPTION Ligands: 8LX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-20
Ligands: 8LX
