Search Count: 33
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Structure Of Sars-Cov-2 Main Protease With Potent Peptide Aldehyde Inhibitor
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.35 Å Release Date: 2024-08-07 Classification: HYDROLASE/INHIBITOR Ligands: A1ADM, NA, EDO, PEG |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2024-08-07
Ligands: A1ADM, NA, EDO, PEG
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Sars-Cov-2 Main Protease With Covalent Inhibitor
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2024-04-03 Classification: VIRAL PROTEIN Ligands: BTB, A1AD0, DMS, EDO |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2024-04-03
Ligands: BTB, A1AD0, DMS, EDO
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Crystal Structure Of Wild Type Egfr In Complex With Tak-788
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.61 Å Release Date: 2022-12-07 Classification: HYDROLASE Ligands: R28 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-07
Ligands: R28
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Crystal Structure Of Egfr_D770_N771Insnpg/V948R In Complex With Tak-788
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2022-12-07 Classification: HYDROLASE/HYDROLASE Inhibitor Ligands: R28, EDO, CIT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-07
Ligands: R28, EDO, CIT
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Co-Complex Cyp46A1 With Compound 3F
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2022-07-27 Classification: OXIDOREDUCTASE Ligands: HEM, 0I1, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-07-27
Ligands: HEM, 0I1, EDO, GOL
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Co-Complex Cyp46A1 With 0420 (Compound 6)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2022-02-23 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: HEM, EDO, 04Y, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-02-23
Ligands: HEM, EDO, 04Y, GOL
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Co-Complex Cyp46A1 With 0431 (Compound 17)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2022-02-23 Classification: HYDROLASE Ligands: HEM, 05D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-02-23
Ligands: HEM, 05D
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Bacterial O-Glcnacase (Oga) With Compound
Organism: Escherichia coli k-12
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2021-01-13 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ACT, VUA, EDO |
Organism: Escherichia coli k-12
Method: X-RAY DIFFRACTION
Release Date: 2021-01-13
Ligands: ACT, VUA, EDO
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P38 In Complex With T-3220137
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2019-11-20 Classification: TRANSFERASE/INHIBITOR Ligands: MKP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-20
Ligands: MKP
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Structure Of Rorgt In Complex With A Novel Inverse Agonist 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.69 Å Release Date: 2018-01-03 Classification: SIGNALING PROTEIN Ligands: CFG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-01-03
Ligands: CFG
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Crystal Structure Of The Bcl6 Btb Domain In Complex With Compound 1A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.58 Å Release Date: 2017-08-16 Classification: Transcription/Inhibitor Ligands: 80R, EDO, K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-08-16
Ligands: 80R, EDO, K
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Crystal Structure Of The Bcl6 Btb Domain In Complex With Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2017-08-16 Classification: Transcription/Inhibitor Ligands: 80L |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-08-16
Ligands: 80L
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Crystal Structure Of The Bcl6 Btb Domain In Complex With Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2017-05-24 Classification: Transcription/Inhibitor Ligands: 7ZF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: 7ZF
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Crystal Structure Of The Bcl6 Btb Domain In Complex With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2017-05-24 Classification: Transcription/Inhibitor Ligands: 7ZL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: 7ZL, EDO
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Crystal Structure Of The Bcl6 Btb Domain In Complex With Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2017-05-24 Classification: Transcription/Inhibitor Ligands: YAM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: YAM
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Crystal Structure Of The Bcl6 Btb Domain In Complex With Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.06 Å Release Date: 2017-05-24 Classification: Transcription/Inhibitor Ligands: 7ZO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: 7ZO
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Crystal Structure Of The Bcl6 Btb Domain In Complex With Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2017-05-24 Classification: Transcription/Inhibitor Ligands: 7Z6, EDO, K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: 7Z6, EDO, K
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Human Givd Cytosolic Phospholipase A2 In Complex With Methyl Gamma-Linolenyl Fluorophosphonate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2016-06-08 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: 7FA, BA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-08
Ligands: 7FA, BA
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Human Givd Cytosolic Phospholipase A2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2016-06-08 Classification: HYDROLASE Ligands: SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-08
Ligands: SO4
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Human Givd Cytosolic Phospholipase A2 In Complex With Methyl Gamma-Linolenyl Fluorophosphonate Inhibitor And Terbium Chloride
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.25 Å Release Date: 2016-06-08 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: 7FA, TB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-08
Ligands: 7FA, TB
