Search Count: 30
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Crystal Structure Of Menin In Complex With Inhibitor Compound 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2025-01-15 Classification: PROTEIN BINDING/INHIBITOR Ligands: A1AVE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-15
Ligands: A1AVE
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Crystal Structure Of Menin In Complex With Inhibitor Compound 26
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2025-01-15 Classification: PROTEIN BINDING/INHIBITOR Ligands: A1AVF, K, EPE, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-15
Ligands: A1AVF, K, EPE, SO4
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Crystal Structure Of Menin In Complex With Inhibitor Compound 20
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2025-01-15 Classification: PROTEIN BINDING/INHIBITOR Ligands: A1AVG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-15
Ligands: A1AVG
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Crystal Structure Of Mutant Cmet D1228N Kinase Domain In Complex With Inhibitor Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2024-08-21 Classification: SIGNALING PROTEIN Ligands: GOL, A1ATS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-08-21
Ligands: GOL, A1ATS
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Crystal Structure Of Braf Kinase Domain With Pf-07284890
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2024-08-14 Classification: SIGNALING PROTEIN Ligands: PEG, GOL, A1AN9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-08-14
Ligands: PEG, GOL, A1AN9
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Crystal Structure Of The Receptor Tyrosine Kinase Human Her2 (Erbb2) Yvma Mutant Kinase Domain In Complex With Inhibitor Compound 27
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2024-06-12 Classification: SIGNALING PROTEIN,TRANSFERASE/INHIBITOR Ligands: W9N, PEG, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-12
Ligands: W9N, PEG, CL
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Crystal Structure Of Non-Receptor Protein Tyrosine Phosphatase Shp2 In Complex With Pf-07284892
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.06 Å Release Date: 2024-05-29 Classification: HYDROLASE/INHIBITOR Ligands: A1AQ1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-05-29
Ligands: A1AQ1
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Highly Potent And Selective 3-N-Methylquinazoline-4(3H)-One Based Inhibitors Of B-Rafv600E Kinase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.40 Å Release Date: 2014-04-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 2VX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-09
Ligands: 2VX
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Human B-Raf Kinase Domain In Complex With An Imidazopyridine-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.60 Å Release Date: 2013-10-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: DFS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-10-02
Ligands: DFS
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B-Raf Kinase Domain In Complex With An Aminothienopyrimidine-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.30 Å Release Date: 2013-04-24 Classification: Transferase/Transferase Inhibitor Ligands: RI8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-24
Ligands: RI8
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B-Raf Kinase Domain In Complex With An Aminopyridimine-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.50 Å Release Date: 2013-04-24 Classification: Transferase/Transferase Inhibitor Ligands: RI9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-24
Ligands: RI9
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Human B-Raf Kinase Domain Bound To A Type Ii Pyrazolopyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.50 Å Release Date: 2012-11-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0WP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-11-14
Ligands: 0WP
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B-Raf V600E Kinase Domain Bound To A Type Ii Dihydroquinazoline Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2012-11-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: B1E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-11-14
Ligands: B1E
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Crystal Structure Of B-Raf Kinase Domain In Complex With A Dihydropyrido[2,3-D]Pyrimidinone-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.60 Å Release Date: 2012-05-09 Classification: Transferase/Transferase Inhibitor Ligands: T1Q |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-09
Ligands: T1Q
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Human B-Raf Kinase Domain In Complex With An Bromopyridine Benzamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.40 Å Release Date: 2011-10-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: TV4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-05
Ligands: TV4
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Human B-Raf Kinase Domain In Complex With A Methoxypyrazolopyridinyl Benzamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.30 Å Release Date: 2011-10-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: B0R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-05
Ligands: B0R
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Human B-Raf Kinase In Complex With An Amide Linked Pyrazolopyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2011-08-17 Classification: Transferase/Transferase Inhibitor Ligands: BR2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-17
Ligands: BR2
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Non-Oxime Pyrazole Based Inhibitors Of B-Raf Kinase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.60 Å Release Date: 2011-05-18 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SM7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-05-18
Ligands: SM7
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Human B-Raf Kinase In Complex With A Furopyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.70 Å Release Date: 2011-02-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: FOI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-02-02
Ligands: FOI
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Human B-Raf Kinase In Complex With A Non-Oxime Furopyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2011-02-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: FNI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-02-02
Ligands: FNI
