Search Count: 47
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Mapping The Shp2 Allosteric Pocket With Target-Biased Covalent Fragments
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2026-05-06 Classification: CYTOSOLIC PROTEIN Ligands: EDO, A1JWN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-05-06
Ligands: EDO, A1JWN
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Mtb Guab Dcbs In Complex With Inhibitor G1
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2024-11-27 Classification: OXIDOREDUCTASE Ligands: IMP, VOA, SO4 |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2024-11-27
Ligands: IMP, VOA, SO4
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Mtb Guab Dcbs In Complex With Inhibitor Compound 5
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2024-11-27 Classification: OXIDOREDUCTASE Ligands: IMP, A1A3K |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2024-11-27
Ligands: IMP, A1A3K
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Crystal Structure Of R9A Spin Labeled T4 Lysozyme Mutant K65R9A/R76R9A
Organism: Escherichia phage t4
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2024-06-05 Classification: ANTIMICROBIAL PROTEIN,HYDROLASE Ligands: GFX |
Organism: Escherichia phage t4
Method: X-RAY DIFFRACTION
Release Date: 2024-06-05
Ligands: GFX
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With The Ligand Zz001229A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.48 Å Release Date: 2024-02-07 Classification: GENE REGULATION Ligands: EDO, IX4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-07
Ligands: EDO, IX4
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The Crystal Structure Of Mtbtop1 In Complex With Both G- And T-Segments
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:2.78 Å Release Date: 2022-12-14 Classification: ISOMERASE/DNA Ligands: GOL, ACT, PO4 |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2022-12-14
Ligands: GOL, ACT, PO4
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Human Serum Transferrin With Five Osmium Binding Sites
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.06 Å Release Date: 2022-06-22 Classification: METAL TRANSPORT Ligands: 4TI, MLI, NTA, OS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-06-22
Ligands: 4TI, MLI, NTA, OS
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Osmium-Bound Human Serum Transferrin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2022-06-22 Classification: METAL TRANSPORT Ligands: FE, MLI, OS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-06-22
Ligands: FE, MLI, OS
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Gdc-9545 In Complex With Estrogen Receptor Alpha
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2021-06-02 Classification: TRANSCRIPTION Ligands: G9J, ZNM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-06-02
Ligands: G9J, ZNM
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Crystal Structure Of Mycobacterium Smegmatis Topoisomerase I With Ssdna Bound To Both N- And C-Terminal Domains
Organism: Mycobacterium smegmatis (strain atcc 700084 / mc(2)155), Mycolicibacterium smegmatis
Method: X-RAY DIFFRACTION Resolution:3.11 Å Release Date: 2020-03-25 Classification: ISOMERASE/DNA Ligands: SO4 |
Organism: Mycobacterium smegmatis (strain atcc 700084 / mc(2)155), Mycolicibacterium smegmatis
Method: X-RAY DIFFRACTION
Release Date: 2020-03-25
Ligands: SO4
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Crystal Structure Of 8-Hydroxychromene Compound 30 Bound To Estrogen Receptor Alpha
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2019-07-17 Classification: NUCLEAR PROTEIN Ligands: G9J, ODY, CL, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-17
Ligands: G9J, ODY, CL, DMS
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Crystal Structure Of Gdc-0927 Bound To Estrogen Receptor Alpha
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.84 Å Release Date: 2019-07-17 Classification: NUCLEAR PROTEIN Ligands: OGJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-17
Ligands: OGJ
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Crystal Structure Of Estrogen Receptor Alpha In Complex With Receptor Degrader 16Ab
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2019-02-20 Classification: NUCLEAR PROTEIN Ligands: G8Y, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-20
Ligands: G8Y, GOL
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Crystal Structure Of Estrogen Receptor Alpha In Complex With Receptor Degrader 16Aa
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2019-02-20 Classification: NUCLEAR PROTEIN Ligands: G9J, NI, G91, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-20
Ligands: G9J, NI, G91, GOL
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N-Terminal Bromodomain Of Brd4 In Complex With Plx5981
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2018-08-01 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: EDO, 6JC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-01
Ligands: EDO, 6JC
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N-Terminal Bromodomain Of Brd4 In Complex With Otx-015
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.27 Å Release Date: 2018-08-01 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: 6JE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-01
Ligands: 6JE
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N-Terminal Bromodomain Of Brd4 In Complex With Otx-015
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.19 Å Release Date: 2018-08-01 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: EDO, 6JF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-01
Ligands: EDO, 6JF
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Crystal Structure Of Mycobacterium Tuberculosis Topoisomerase I In Complex With Oligonucleotide Mts2-12 And Magnesium
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv), Mycobacterium tuberculosis h37rv
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2018-05-30 Classification: ISOMERASE/DNA Ligands: MG, PO4 |
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv), Mycobacterium tuberculosis h37rv
Method: X-RAY DIFFRACTION
Release Date: 2018-05-30
Ligands: MG, PO4
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2.42A Crystal Structure Of Mycobacterium Tuberculosis Topoisomerase I In Complex With An Oligonucleotide Mts2-11
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv), Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:2.42 Å Release Date: 2018-05-30 Classification: ISOMERASE/DNA Ligands: FMT, GOL, ACT |
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv), Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2018-05-30
Ligands: FMT, GOL, ACT
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Native Structure Of Ndm-1 Crystallized At Ph5.5
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION Resolution:0.95 Å Release Date: 2018-03-07 Classification: HYDROLASE Ligands: ZN, OH, EDO, SIN |
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION
Release Date: 2018-03-07
Ligands: ZN, OH, EDO, SIN
