Search Count: 20
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Structure Of Gpr61 Bound To Inverse Agonist Compound 15
Organism: Homo sapiens, Lama glama
Method: ELECTRON MICROSCOPY Resolution:3.08 Å Release Date: 2026-03-25 Classification: SIGNALING PROTEIN Ligands: A1CWB |
Organism: Homo sapiens, Lama glama
Method: ELECTRON MICROSCOPY
Release Date: 2026-03-25
Ligands: A1CWB
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Rat Branched Chain Ketoacid Dehydrogenase Kinase In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.16 Å Release Date: 2024-11-27 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ADP, MG, K, A1A40, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-27
Ligands: ADP, MG, K, A1A40, PO4
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Cryo-Em Structure Of Gpr61-G Protein Complex Stabilized By Scfv16
Organism: Homo sapiens, Escherichia coli
Method: ELECTRON MICROSCOPY Release Date: 2023-10-04 Classification: SIGNALING PROTEIN |
Organism: Homo sapiens, Escherichia coli
Method: ELECTRON MICROSCOPY
Release Date: 2023-10-04
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Cryo-Em Structure Of Gpr61-
Organism: Homo sapiens, Escherichia coli, Lama glama
Method: ELECTRON MICROSCOPY Release Date: 2023-10-04 Classification: SIGNALING PROTEIN Ligands: ZOB |
Organism: Homo sapiens, Escherichia coli, Lama glama
Method: ELECTRON MICROSCOPY
Release Date: 2023-10-04
Ligands: ZOB
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Human Branched Chain Ketoacid Dehydrogenase Kinase In Complex With Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.15 Å Release Date: 2023-07-05 Classification: SIGNALING PROTEIN,TRANSFERASE/INHIBITOR Ligands: ADP, MG, XGG, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-05
Ligands: ADP, MG, XGG, SO4
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Human Branched Chain Ketoacid Dehydrogenase Kinase In Complex With Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2023-07-05 Classification: SIGNALING PROTEIN,TRANSFERASE/INHIBITOR Ligands: ADP, MG, K, XER |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-05
Ligands: ADP, MG, K, XER
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Human Branched Chain Ketoacid Dehydrogenase Kinase In Complex With Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.79 Å Release Date: 2023-07-05 Classification: SIGNALING PROTEIN,TRANSFERASE/INHIBITOR Ligands: ADP, MG, K, XGT, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-05
Ligands: ADP, MG, K, XGT, SO4
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Branched Chain Ketoacid Dehydrogenase Kinase In Complex With Inhibitor
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2023-03-08 Classification: SIGNALING PROTEIN Ligands: ADP, MG, K, SO4, WIH |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2023-03-08
Ligands: ADP, MG, K, SO4, WIH
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Branched Chain Ketoacid Dehydrogenase Kinase In Complex With Inhibitor
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2023-03-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ADP, K, SO4, WIK |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2023-03-08
Ligands: ADP, K, SO4, WIK
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Branched Chain Ketoacid Dehydrogenase Kinase Complexes
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2023-03-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ADP, WJK, SO4 |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2023-03-08
Ligands: ADP, WJK, SO4
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Branched Chain Ketoacid Dehydrogenase Kinase Complexes
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2023-03-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ADP, U35, SO4 |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2023-03-08
Ligands: ADP, U35, SO4
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Pde2 Catalytic Domain Complexed With Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2017-06-28 Classification: Hydrolase/Hydrolase Inhibitor Ligands: 19F, ZN, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: 19F, ZN, MG
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Pde2 Catalytic Domain Complexed With Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2017-06-28 Classification: Hydrolase/Hydrolase Inhibitor Ligands: 7XS, ZN, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: 7XS, ZN, MG
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Pde2 Catalytic Domain Complexed With Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2017-06-28 Classification: Hydrolase/Hydrolase Inhibitor Ligands: 7XV, ZN, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: 7XV, ZN, MG
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Pde2 Catalytic Domain Complexed With Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.06 Å Release Date: 2017-06-28 Classification: Hydrolase/Hydrolase Inhibitor Ligands: ZN, MG, 7Y1, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: ZN, MG, 7Y1, CL
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Pde2 Catalytic Domain Complexed With Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.38 Å Release Date: 2017-06-28 Classification: Hydrolase/Hydrolase Inhibitor Ligands: 7Y4, ZN, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: 7Y4, ZN, MG
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Crystal Structure Of Mst3 With A Pyrrolopyrimidine Inhibitor (Pf-06447475)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2015-03-18 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: MN, 3FE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-03-18
Ligands: MN, 3FE
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Crystal Structure Of Mst3 With A Pyrrolopyrimidine Inhibitor (Pf-06454589).
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2015-03-18 Classification: transferase/transferase inhibitor Ligands: 3JA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-03-18
Ligands: 3JA
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Structure Of Mst3 With A Pyrrolopyrimidine Inhibitor (Pf-06645342)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2015-03-18 Classification: transferase/transferase inhibitor Ligands: 3JB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-03-18
Ligands: 3JB
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Crystal Structure Of Tyk2 In Complex With Compound 15, 6-((2,5-Dimethoxyphenyl)Thio)-3-(1-Methyl-1H-Pyrazol-4-Yl)-[1,2,4]Triazolo[4,3-B]Pyridazine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.16 Å Release Date: 2014-09-03 Classification: TRANSFERASE Ligands: 2YK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-09-03
Ligands: 2YK
