Search Count: 22
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Structural Basis For Kinase Selectivity Of Three Clinical P38Alpha Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2012-07-04 Classification: TRANSFERASE Ligands: SB2, BOG, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-07-04
Ligands: SB2, BOG, EDO
 |
X-Ray Structure Of P38Alpha Bound To Tak-715
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2012-06-13 Classification: TRANSFERASE Ligands: T75, BOG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-06-13
Ligands: T75, BOG
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X-Ray Structure Of P38Alpha Bound To Scio-469
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2012-06-13 Classification: TRANSFERASE Ligands: 469, BOG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-06-13
Ligands: 469, BOG
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X-Ray Structure Of P38Alpha Bound To Vx-745
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2012-06-13 Classification: TRANSFERASE Ligands: 52P, BOG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-06-13
Ligands: 52P, BOG
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Pr X-Ray Structures In Agonist Conformations Reveal Two Different Mechanisms For Partial Agonism In 11Beta-Substituted Steroids
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2012-04-25 Classification: TRANSCRIPTION Ligands: OR8, SO4, A2K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-04-25
Ligands: OR8, SO4, A2K
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Factor Xia In Complex With A Clorophenyl-Tetrazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2012-04-11 Classification: Hydrolase/Hydrolase inhibitor Ligands: CIT, O58 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-04-11
Ligands: CIT, O58
 |
Benzothiazinone Inhibitor In Complex With Fxia
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.58 Å Release Date: 2012-04-11 Classification: Hydrolase/Hydrolase Inhibitor Ligands: CIT, TRS, O61 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-04-11
Ligands: CIT, TRS, O61
 |
Pr X-Ray Structures In Agonist Conformations Reveal Two Different Mechanisms For Partial Agonism In 11Beta-Substituted Steroids
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2012-04-04 Classification: TRANSCRIPTION Ligands: AS0, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-04-04
Ligands: AS0, SO4
 |
Novel Atp-Competitive Mk2 Inhibitors With Potent Biochemical And Cell-Based Activity Throughout The Series
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2011-12-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: I85 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-12-14
Ligands: I85
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Mk3 Kinase Bound To Compound 5B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2011-05-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 05B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-05-25
Ligands: 05B
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Mk2 Kinase Bound To Compound 5B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2011-05-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 05B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-05-25
Ligands: 05B
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Mk2 Kinase Bound To Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2011-05-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: MLI, P4O |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-05-25
Ligands: MLI, P4O
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Mk2 Kinase Bound To Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2011-05-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: CD2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-05-25
Ligands: CD2
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Ligand-Binding Domain Of Glua2 (Flip) Ionotropic Glutamate Receptor In Complex With An Allosteric Modulator
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2011-01-12 Classification: TRANSPORT PROTEIN Ligands: GLU, SO4, 557, GOL |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2011-01-12
Ligands: GLU, SO4, 557, GOL
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Ligand-Binding Domain Of Glua2 (Flip) Ionotropic Glutamate Receptor In Complex With An Allosteric Modulator
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2011-01-12 Classification: TRANSPORT PROTEIN Ligands: GLU, SO4, GOL, DMS, G69 |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2011-01-12
Ligands: GLU, SO4, GOL, DMS, G69
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Ligand-Binding Domain Of Glua2 (Flip) Ionotropic Glutamate Receptor In Complex With An Allosteric Modulator
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2011-01-12 Classification: TRANSPORT PROTEIN Ligands: GLU, SO4, GOL, DMS, EDO, 808 |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2011-01-12
Ligands: GLU, SO4, GOL, DMS, EDO, 808
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Ligand-Binding Domain Of Glua2 (Flip) Ionotropic Glutamate Receptor In Complex With An Allosteric Modulator
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2010-09-15 Classification: TRANSPORT PROTEIN Ligands: O28, GLU, SO4, DMS, GOL |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2010-09-15
Ligands: O28, GLU, SO4, DMS, GOL
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Ligand-Binding Domain Of Glua2 (Flip) Ionotropic Glutamate Receptor In Complex With An Allosteric Modulator
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2010-09-15 Classification: TRANSPORT PROTEIN Ligands: GLU, SO4, GOL, O29 |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2010-09-15
Ligands: GLU, SO4, GOL, O29
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Ligand-Binding Domain Of Glua2 (Flip) Ionotropic Glutamate Receptor In Complex With An Allosteric Modulator
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2010-09-15 Classification: TRANSPORT PROTEIN Ligands: O30, GLU, SO4, GOL |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2010-09-15
Ligands: O30, GLU, SO4, GOL
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Ligand-Binding Domain Of Glua2 (Flip) Ionotropic Glutamate Receptor In Complex With An Allosteric Modulator
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2010-09-15 Classification: TRANSPORT PROTEIN Ligands: GLU, SO4, O27, EDO |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2010-09-15
Ligands: GLU, SO4, O27, EDO