Search Count: 100
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Crystal Structure Of Tead4 In Complex With Compound 9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2026-03-11 Classification: TRANSCRIPTION Ligands: U3O, A1ICN, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-03-11
Ligands: U3O, A1ICN, PO4
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Crystal Structure Of Tead4 In Complex With Vgll1-Peptide And Iag933
Organism: Homo sapiens, Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2026-03-11 Classification: TRANSCRIPTION Ligands: MYR, WCF |
Organism: Homo sapiens, Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2026-03-11
Ligands: MYR, WCF
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Crystal Structure Of Tead4 In Complex With Ytp-13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2023-04-12 Classification: TRANSCRIPTION Ligands: U3F, U3O, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-04-12
Ligands: U3F, U3O, PO4
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Crystal Structure Of Tead4 In Complex With Peptide 1
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2023-03-15 Classification: TRANSCRIPTION Ligands: GOL, MYR |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2023-03-15
Ligands: GOL, MYR
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Crystal Structure Of Tead3 In Complex With Cpd4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2022-08-17 Classification: TRANSCRIPTION Ligands: MYR, KMU, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-17
Ligands: MYR, KMU, PO4
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Crystal Structure Of Tead3 In Complex With Cpd2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2022-08-17 Classification: TRANSCRIPTION Ligands: MYR, DMS, KNE, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-17
Ligands: MYR, DMS, KNE, PO4
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X-Ray Structure Of Hdm2/Cmr19 At 1.45A: Discovery, X-Ray Structure And Cpp-Conjugation Enabled Uptake Of P53/Mdm2 Macrocyclic Peptide Inhibitors
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2021-09-22 Classification: LIGASE Ligands: SO4, CL |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2021-09-22
Ligands: SO4, CL
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Fkbp12 In Complex With The Bmp Potentiator Compound 9 At 1.55 A Resolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2021-03-10 Classification: ISOMERASE Ligands: 818, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-10
Ligands: 818, SO4
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Fkbp12 In Complex With The Bmp Potentiator Compound 8 At 1.12A Resolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.12 Å Release Date: 2021-03-10 Classification: ISOMERASE Ligands: OP8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-10
Ligands: OP8
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Fkbp12 In Complex With The Bmp Potentiator Compound 6 At 1.03A Resolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.03 Å Release Date: 2021-03-10 Classification: ISOMERASE Ligands: OP5, CD, CL, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-10
Ligands: OP5, CD, CL, NA
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Fkbp12 In Complex With The Bmp Potentiator Compound 10 At 1.00A Resolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.00 Å Release Date: 2021-03-10 Classification: ISOMERASE Ligands: OOZ, CD, CL, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-10
Ligands: OOZ, CD, CL, NA
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Rorcvar2 (Rorgt, 264-499) In Complex With Compound 1: Identification Of N-Aryl Imidazoles As Potent And Selective Rorgt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2019-11-27 Classification: TRANSCRIPTION Ligands: HJW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-27
Ligands: HJW
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Rorcvar2 (Rorgt, 264-499) In Complex With Compound 2 At 2.3A: Identification Of N-Aryl Imidazoles As Potent And Selective Rorgt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2019-11-27 Classification: TRANSCRIPTION Ligands: HKE, CHD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-27
Ligands: HKE, CHD
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Rorcvar2 (Rorgt, 264-499) In Complex With Compound 4 At 2.2A: Identification Of N-Aryl Imidazoles As Potent And Selective Rorgt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2019-11-27 Classification: TRANSCRIPTION Ligands: HKZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-27
Ligands: HKZ
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Rorcvar2 (Rorgt, 264-499) In Complex With Compound 9 At 2.3A: Identification Of N-Aryl Imidazoles As Potent And Selective Rorgt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2019-11-27 Classification: TRANSCRIPTION Ligands: HL8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-27
Ligands: HL8
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X-Ray Structure Of The P53-Mdm2 Inhibitor Nmi801 Bound To Hdm2 At 2.1A Resolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2019-11-20 Classification: LIGASE Ligands: H0W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-20
Ligands: H0W
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Tead4 (216-434) Complexed With Yap Peptide (60-100) And Myristoate (Covalently Bound) At 2.1A (P41212 Crystal Form)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2019-07-03 Classification: TRANSCRIPTION Ligands: GOL, MYR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-03
Ligands: GOL, MYR
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Tead4(216-434) Complexed With Optimized Peptide 9 And Myristoate (Covalently Bound) At 2.01A Resolution: Structure-Based Design Of Potent Linear Peptide Inhibitors Of The Yap-Tead Protein-Protein Interaction Derived From The Yap Omega-Loop Sequence
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.01 Å Release Date: 2019-07-03 Classification: TRANSCRIPTION Ligands: MYR, PO4 |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2019-07-03
Ligands: MYR, PO4
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Hdm2 (17-111, Wild Type) Complexed With Compound 12 At 1.8A; Structural States Of Hdm2 And Hdmx: X-Ray Elucidation Of Adaptations And Binding Interactions For Different Chemical Compound Classes
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2019-05-15 Classification: LIGASE Ligands: HRE, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-15
Ligands: HRE, SO4
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Hdm2 (17-111, Wild Type) Complexed With Compound 11 At 2.0A; Structural States Of Hdm2 And Hdmx: X-Ray Elucidation Of Adaptations And Binding Interactions For Different Chemical Compound Classes
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2019-05-15 Classification: LIGASE Ligands: HRH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-15
Ligands: HRH
