Search Count: 27
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Rat Branched Chain Ketoacid Dehydrogenase Kinase In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.16 Å Release Date: 2024-11-27 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ADP, MG, K, A1A40, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-27
Ligands: ADP, MG, K, A1A40, PO4
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Sars-Cov-2 Papain-Like Protease (Plpro) Bound To Pf-07957472
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2024-10-02 Classification: VIRAL PROTEIN Ligands: A1AZ1, TFA, ZN |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2024-10-02
Ligands: A1AZ1, TFA, ZN
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Structure Of Sars-Cov-2 Main Protease In Complex With A Covalent Inhibitor
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2024-05-15 Classification: VIRAL PROTEIN Ligands: YDL |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2024-05-15
Ligands: YDL
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Human Branched Chain Ketoacid Dehydrogenase Kinase In Complex With Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.15 Å Release Date: 2023-07-05 Classification: SIGNALING PROTEIN,TRANSFERASE/INHIBITOR Ligands: ADP, MG, XGG, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-05
Ligands: ADP, MG, XGG, SO4
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Human Branched Chain Ketoacid Dehydrogenase Kinase In Complex With Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2023-07-05 Classification: SIGNALING PROTEIN,TRANSFERASE/INHIBITOR Ligands: ADP, MG, K, XER |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-05
Ligands: ADP, MG, K, XER
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Human Branched Chain Ketoacid Dehydrogenase Kinase In Complex With Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.79 Å Release Date: 2023-07-05 Classification: SIGNALING PROTEIN,TRANSFERASE/INHIBITOR Ligands: ADP, MG, K, XGT, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-05
Ligands: ADP, MG, K, XGT, SO4
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Glp-1 Receptor Bound With Pfizer Small Molecule Agonist
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2022-06-08 Classification: MEMBRANE PROTEIN Ligands: 82L |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2022-06-08
Ligands: 82L
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Structure Of Sars-Cov-2 Main Protease In Complex With A Covalent Inhibitor
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2021-11-10 Classification: HYDROLASE/INHIBITOR Ligands: 4W8 |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2021-11-10
Ligands: 4W8
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Structure Of Sars-Cov-2 Main Protease In Complex With A Covalent Inhibitor
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2021-11-10 Classification: HYDROLASE/INHIBITOR Ligands: 4WI |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2021-11-10
Ligands: 4WI
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Structure Of Sars-Cov-2 Main Protease In Complex With A Covalent Inhibitor
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2021-11-10 Classification: HYDROLASE/INHIBITOR Ligands: 4YG |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2021-11-10
Ligands: 4YG
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Structure Of Sars-Cov-2 Main Protease In Complex With A Covalent Inhibitor
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2021-11-10 Classification: HYDROLASE/INHIBITOR Ligands: 4WI |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2021-11-10
Ligands: 4WI
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Structure Of Khk In Complex With Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2020-09-23 Classification: TRANSFERASE Ligands: RYS, SO4, CIT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-09-23
Ligands: RYS, SO4, CIT
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Structure Of Khk In Complex With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2020-09-23 Classification: TRANSFERASE Ligands: RZA, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-09-23
Ligands: RZA, SO4
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Structure Of Khk In Complex With Compound 4 (6-[(1~{S},5~{R})-6-(Hydroxymethyl)-3-Azabicyclo[3.1.0]Hexan-3-Yl]-2-[(2~{S},3~{R})-2-Methyl-3-Oxidanyl-Azetidin-1-Yl]-4-(Trifluoromethyl)Pyridine-3-Carbonitrile)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.38 Å Release Date: 2020-09-23 Classification: TRANSFERASE Ligands: S6J, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-09-23
Ligands: S6J, SO4
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Structure Of Khk In Complex With Compound 6 (2-[(1~{R},5~{S})-3-[5-Cyano-6-[(2~{S},3~{R})-2-Methyl-3-Oxidanyl-Azetidin-1-Yl]-4-(Trifluoromethyl)Pyridin-2-Yl]-3-Azabicyclo[3.1.0]Hexan-6-Yl]Ethanoic Acid)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.54 Å Release Date: 2020-09-23 Classification: TRANSFERASE Ligands: S6S, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-09-23
Ligands: S6S, SO4
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Structure Of Khk In Complex With Compound 8 (2-[(1~{S},5~{R})-3-[2-[(2~{S})-2-Methylazetidin-1-Yl]-6-(Trifluoromethyl)Pyrimidin-4-Yl]-3-Azabicyclo[3.1.0]Hexan-6-Yl]Ethanoic Acid)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2020-09-23 Classification: TRANSFERASE Ligands: S6D, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-09-23
Ligands: S6D, SO4
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Structure Of Ampk Bound To Activator
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:3.40 Å Release Date: 2018-08-08 Classification: TRANSFERASE Ligands: HTV, STU, CL, AMP, ADP, SO4 |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2018-08-08
Ligands: HTV, STU, CL, AMP, ADP, SO4
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Structure Of Ampk Bound To Activator
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:3.27 Å Release Date: 2018-08-08 Classification: TRANSFERASE Ligands: STU, HU7, CL, AMP, ADP, SO4 |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2018-08-08
Ligands: STU, HU7, CL, AMP, ADP, SO4
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Structure Of Ampk Bound To Activator
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:3.35 Å Release Date: 2018-08-08 Classification: TRANSFERASE Ligands: STU, HUG, CL, AMP, ADP, SO4 |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2018-08-08
Ligands: STU, HUG, CL, AMP, ADP, SO4
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Structure Of Ampk Bound To Activator
Organism: Rattus norvegicus, Mus musculus
Method: X-RAY DIFFRACTION Resolution:3.45 Å Release Date: 2017-05-17 Classification: TRANSFERASE/ACTIVATOR Ligands: STU, 85V, CL, SO4, AMP, ADP |
Organism: Rattus norvegicus, Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2017-05-17
Ligands: STU, 85V, CL, SO4, AMP, ADP
