Search Count: 9
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Factor Xia In Complex With A Clorophenyl-Tetrazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2012-04-11 Classification: Hydrolase/Hydrolase inhibitor Ligands: CIT, O58 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-04-11
Ligands: CIT, O58
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Benzothiazinone Inhibitor In Complex With Fxia
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.58 Å Release Date: 2012-04-11 Classification: Hydrolase/Hydrolase Inhibitor Ligands: CIT, TRS, O61 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-04-11
Ligands: CIT, TRS, O61
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6-Phenyl-1H-Imidazo[4,5-C]Pyridine-4-Carbonitrile As Cathepsin S Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2011-04-06 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: EF3, DMS, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-04-06
Ligands: EF3, DMS, SO4
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Cathepsin S In Complex With A Covalent Inhibitor With An Aldehyde Warhead
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.49 Å Release Date: 2010-12-22 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: O64, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-12-22
Ligands: O64, DMS
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Cathepsin K In Complex With A Covalent Inhibitor With A Ketoamide Warhead
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2010-12-22 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: O96, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-12-22
Ligands: O96, SO4
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4-(3-Trifluoromethylphenyl)-Pyrimidine-2-Carbonitrile As Cathepsin S Inhibitors: N3, Not N1 Is Critically Important
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2010-07-14 Classification: HYDROLASE Ligands: PEG, DMS, 935, 93N, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-07-14
Ligands: PEG, DMS, 935, 93N, SO4, GOL
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X-Ray Structure Of Cathepsin K Covalently Bound To A Triazine Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2010-03-02 Classification: HYDROLASE Ligands: ORG, TFA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-03-02
Ligands: ORG, TFA
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Cathepsin K In Complex With A Non-Selective 2-Cyano-Pyrimidine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.49 Å Release Date: 2010-03-02 Classification: HYDROLASE Ligands: SO4, KWZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-03-02
Ligands: SO4, KWZ
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Cathepsin K In Complex With A Selective 2-Cyano-Pyrimidine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.51 Å Release Date: 2010-03-02 Classification: HYDROLASE Ligands: KX1, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-03-02
Ligands: KX1, SO4
