Search Count: 5
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First-In-Class Small Molecule Inhibitors Of Polycomb Repressive Complex 1 (Prc1) Ring Domain
Organism: Homo sapiens
Method: SOLUTION NMR Release Date: 2021-06-16 Classification: GENE REGULATION Ligands: ZN, U9E |
Organism: Homo sapiens
Method: SOLUTION NMR
Release Date: 2021-06-16
Ligands: ZN, U9E
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Ring1B-Bmi1 Fusion In Closed Conformation
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2021-04-14 Classification: LIGASE Ligands: ZN, EPE, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-14
Ligands: ZN, EPE, GOL
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Inhibitor Compound-Induced Confrontational Change In Ring1B-Bmi1 Domain Structure
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.09 Å Release Date: 2021-04-14 Classification: LIGASE Ligands: ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-14
Ligands: ZN
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Menin In Complex With Mi-503
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2015-04-15 Classification: protein binding/inhibitor Ligands: 3XW, DMS, PG4, SO4, EDO, EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-15
Ligands: 3XW, DMS, PG4, SO4, EDO, EPE
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Menin In Complex With Mi-136
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2015-04-15 Classification: protein binding/inhibitor Ligands: SO4, 3XY, PG4, DMS, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-15
Ligands: SO4, 3XY, PG4, DMS, EDO
