Search Count: 77
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Gas41 Yeats Domain In Complex With Dlg-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2026-02-25 Classification: PROTEIN BINDING Ligands: PEG, SO4, A1B9P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-02-25
Ligands: PEG, SO4, A1B9P
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Menin Mutant G331R In Complex With Mll Peptide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.54 Å Release Date: 2025-05-21 Classification: PROTEIN BINDING Ligands: SO4, 1PE, PG0, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-21
Ligands: SO4, 1PE, PG0, EDO
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Menin Mutant M327I In Complex With Mll Peptide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.46 Å Release Date: 2025-05-14 Classification: PROTEIN BINDING Ligands: SO4, 1PE, PG0, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-14
Ligands: SO4, 1PE, PG0, PEG
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Menin Mutant T349M In Complex With Mll Peptide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.57 Å Release Date: 2025-05-14 Classification: PROTEIN BINDING Ligands: PEG, SO4, 1PE, PG0, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-14
Ligands: PEG, SO4, 1PE, PG0, EDO
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Menin Mutant G331D In Complex With Mll Peptide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.47 Å Release Date: 2025-05-14 Classification: PROTEIN BINDING Ligands: SO4, 1PE, PG0, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-14
Ligands: SO4, 1PE, PG0, EDO
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Menin Mutant - G331R
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2025-05-14 Classification: PROTEIN BINDING Ligands: PG4, SO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-14
Ligands: PG4, SO4, EDO
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Menin Mutant - M327I
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.58 Å Release Date: 2025-05-14 Classification: PROTEIN BINDING Ligands: PG4, PEG, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-14
Ligands: PG4, PEG, SO4
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Menin Mutant - T349M
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.31 Å Release Date: 2025-05-14 Classification: PROTEIN BINDING Ligands: EDO, PG4, PEG, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-14
Ligands: EDO, PG4, PEG, SO4
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Menin Mutant - G331D
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2025-05-14 Classification: PROTEIN BINDING Ligands: PEG, SO4, PG4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-14
Ligands: PEG, SO4, PG4, EDO
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Menin Mutant - T349M In Complex With Ziftomenib (Ko-539)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2024-11-20 Classification: PROTEIN BINDING Ligands: K5O, PEG, PG4, EDO, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-20
Ligands: K5O, PEG, PG4, EDO, DMS
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Menin In Complex With Ziftomenib (Ko-539)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.57 Å Release Date: 2024-11-20 Classification: PROTEIN BINDING Ligands: K5O, PEG, SO4, DMS, PG4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-20
Ligands: K5O, PEG, SO4, DMS, PG4, EDO
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Gas41 Yeats Domain In Complex With 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2021-07-21 Classification: PROTEIN BINDING Ligands: V91, EDO, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-21
Ligands: V91, EDO, DMS
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First-In-Class Small Molecule Inhibitors Of Polycomb Repressive Complex 1 (Prc1) Ring Domain
Organism: Homo sapiens
Method: SOLUTION NMR Release Date: 2021-06-16 Classification: GENE REGULATION Ligands: ZN, U9E |
Organism: Homo sapiens
Method: SOLUTION NMR
Release Date: 2021-06-16
Ligands: ZN, U9E
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Ring1B-Bmi1 Fusion In Closed Conformation
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2021-04-14 Classification: LIGASE Ligands: ZN, EPE, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-14
Ligands: ZN, EPE, GOL
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Inhibitor Compound-Induced Confrontational Change In Ring1B-Bmi1 Domain Structure
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.09 Å Release Date: 2021-04-14 Classification: LIGASE Ligands: ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-14
Ligands: ZN
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Ash1L Set Domain In Complex With As-85
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2021-04-07 Classification: PROTEIN BINDING, TRANSFERASE/INHIBITOR Ligands: EPE, SAM, ZN, UG7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-07
Ligands: EPE, SAM, ZN, UG7
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Ash1L Set Domain Q2265A Mutant In Complex With As-5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2021-04-07 Classification: PROTEIN BINDING, TRANSFERASE/INHIBITOR Ligands: UK7, ZN, SAM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-07
Ligands: UK7, ZN, SAM
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Nsd1 Set Domain In Complex With Sam
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2020-09-02 Classification: TRANSFERASE Ligands: SAM, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-09-02
Ligands: SAM, ZN
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Nsd1 Set Domain In Complex With Bt3 And Sam
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2020-09-02 Classification: TRANSFERASE Ligands: SAM, DQL, DW9, ZN, CA, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-09-02
Ligands: SAM, DQL, DW9, ZN, CA, GOL
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Menin In Complex With Peptide Inhibitor 25
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2020-09-02 Classification: PROTEIN BINDING/INHIBITOR Ligands: DMS, SO4, PG4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-09-02
Ligands: DMS, SO4, PG4
