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9YDM image
Targeting Ptpn22 At Non-Orthosteric Binding Sites - A Fragment Approach
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.99 Å Release Date: 2026-01-28
Classification: IMMUNE SYSTEM
Ligands: EOH, GOL, SO4, A1CU3

9YG0 image
Targeting Ptpn22 At Non-Orthosteric Binding Sites - A Fragment Approach
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.76 Å Release Date: 2026-01-28
Classification: IMMUNE SYSTEM
Ligands: GOL, EOH, MG, A1CWM, SO4

9YG1 image
Targeting Ptpn22 At Non-Orthosteric Binding Sites - A Fragment Approach
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.97 Å Release Date: 2026-01-28
Classification: IMMUNE SYSTEM
Ligands: EOH, A1CWL, SO4, GOL, MG

9YG2 image
Targeting Ptpn22 At Non-Orthosteric Binding Sites - A Fragment Approach
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.26 Å Release Date: 2026-01-28
Classification: IMMUNE SYSTEM
Ligands: CL, EDO, GOL, A1CWK, MG

9YG3 image
Targeting Ptpn22 At Non-Orthosteric Binding Sites - A Fragment Approach
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.96 Å Release Date: 2026-01-28
Classification: IMMUNE SYSTEM
Ligands: EDO, NA, MG

9BI8 image
Crystal Structure Of Inhibitor Gne-6893 Bound To Hpk1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.25 Å Release Date: 2024-10-02
Classification: SIGNALING PROTEIN
Ligands: A1APL, DMS, NA

9BIK image
Crystal Structure Of Inhibitor 1 Bound To Hpk1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.25 Å Release Date: 2024-10-02
Classification: SIGNALING PROTEIN
Ligands: EDO, A1APO

9BJ1 image
Crystal Structure Of Inhibitor Gne-6893 Bound To Hpk1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.18 Å Release Date: 2024-10-02
Classification: SIGNALING PROTEIN
Ligands: MES, EDO, DMS, A1APR, NA, PEG, A1APQ

8UN3 image
Kras-G13D-Gdp In Complex With Cpd5 (1-((S)-10-(6-Amino-4-Methyl-3-(Trifluoromethyl)Pyridin-2-Yl)-11-Chloro-7-(((2S,4R)-4-Fluoro-1-Methylpyrrolidin-2-Yl)Methoxy)-3,4,13,13A-Tetrahydropyrazino[2',1':3,4][1,4]Oxazepino[5,6,7-De]Quinazolin-2(1H)-Yl)Prop-2-En-1-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.07 Å Release Date: 2023-12-20
Classification: HYDROLASE,ONCOPROTEIN/INHIBITOR
Ligands: XOI, GDP, CL, MG, EDO

8UN4 image
Kras-G13D-Gdp In Complex With Cpd36 ((E)-1-((3S)-4-(7-(6-Amino-4-Methyl-3-(Trifluoromethyl)Pyridin-2-Yl)-6-Chloro-8-Fluoro-2-(((S)-2-Methylenetetrahydro-1H-Pyrrolizin-7A(5H)-Yl)Methoxy)Quinazolin-4-Yl)-3-Methylpiperazin-1-Yl)-3-(4-((Dimethylamino)Methyl)-5-Methylpyridin-2-Yl)Prop-2-En-1-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.57 Å Release Date: 2023-12-20
Classification: HYDROLASE,ONCOPROTEIN/INHIBITOR
Ligands: MG, GDP, XV3

8UN5 image
Kras-G13D-Gdp In Complex With Cpd38 ((E)-1-((3S)-4-(7-(6-Amino-4-Methyl-3-(Trifluoromethyl)Pyridin-2-Yl)-6-Chloro-8-Fluoro-2-(((S)-2-Methylenetetrahydro-1H-Pyrrolizin-7A(5H)-Yl)Methoxy)Quinazolin-4-Yl)-3-Methylpiperazin-1-Yl)-3-(1,2,3,4-Tetrahydroisoquinolin-8-Yl)Prop-2-En-1-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.31 Å Release Date: 2023-12-20
Classification: HYDROLASE,ONCOPROTEIN/INHIBITOR
Ligands: GOL, GDP, MG, XQ6

7MDP image
Kras G12C In Complex With G-2897
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.96 Å Release Date: 2022-03-16
Classification: HYDROLASE/Immune System
Ligands: Z07, GDP, MG, ACT, CAD, P15, EDO, DMS

7RP2 image
Crystal Structure Of Kas G12C In Complex With 2H11 Clamp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.20 Å Release Date: 2022-03-16
Classification: Hydrolase/Immune System
Ligands: GDP, MG, CAC, EDO

7RP3 image
Crystal Structure Of Gne-1952 Alkylated Kras G12C In Complex With 2H11 Clamp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.00 Å Release Date: 2022-03-16
Classification: Hydrolase/Immune System
Ligands: MKZ, GDP, MG, GOL, EDO, SO4

7RP4 image
Crystal Structure Of Kras G12C In Complex With Gne-1952
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.15 Å Release Date: 2022-03-16
Classification: HYDROLASE
Ligands: MKZ, GDP, MG, GOL

7R9L image
Crystal Structure Of Hpk1 In Complex With Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.33 Å Release Date: 2022-01-05
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: 2YE

7R9N image
Crystal Structure Of Hpk1 In Complex With Gne1858
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.50 Å Release Date: 2022-01-05
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: F97, EDO, MES

7R9P image
Crystal Structure Of Hpk1 In Complex With Compound 14
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.27 Å Release Date: 2022-01-05
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: 2WI, SO4

7R9T image
Crystal Structure Of Hpk1 In Complex With Compound 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.00 Å Release Date: 2022-01-05
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: 2TR

6VBN image
Crystal Structure Of Htdo2 Bound To Inhibitor Gne1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:3.18 Å Release Date: 2020-05-06
Classification: OXIDOREDUCTASE/Inhibitor
Ligands: HEM, QVY
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