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Search Count: 13

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5W0F image
Crebbp Bromodomain In Complex With Cpd3 ((S)-1-(3-(6-(1-Methyl-1H-Pyrazol-4-Yl)-3,4-Dihydroquinolin-1(2H)-Yl)-1-(Tetrahydrofuran-3-Yl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridin-5-Yl)Ethan-1-One)

5W0I image
Crebbp Bromodomain In Complex With Cpd8 (1-(3-(7-(Difluoromethyl)-6-(1-Methyl-1H-Pyrazol-4-Yl)-3,4-Dihydroquinolin-1(2H)-Yl)-1-(Tetrahydrofuran-3-Yl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridin-5-Yl)Ethan-1-One)

5W0L image
Crebbp Bromodomain In Complex With Cpd10 (1-(3-(7-(Difluoromethyl)-6-(1-Methyl-1H-Pyrazol-4-Yl)-3,4-Dihydroquinolin-1(2H)-Yl)-1-(Tetrahydro-2H-Pyran-4-Yl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridin-5-Yl)Ethan-1-One)

5W0Q image
Crebbp Bromodomain In Complex With Cpd17 (N,2,7-Trimethyl-2,3-Dihydro-4H-Benzo[B][1,4]Oxazine-4-Carboxamide)

5KTU image
Crystal Structure Of The Bromodomain Of Human Crebbp Bound To Pyrazolopiperidine Scaffold
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.38 Å Release Date: 2016-11-02
Classification: TRANSFERASE
Ligands: 6XB, DMS

5KTW image
Crebbp Bromodomain In Complex With Cpd 44 (3-((5-Acetyl-1-(Cyclopropylmethyl)-4,5,6,7-Tetrahydro-1H-Pyrazolo[4,3-C]Pyridin-3-Yl)Amino)-N-Isopropylbenzamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.09 Å Release Date: 2016-11-02
Classification: TRANSFERASE
Ligands: 6XG, EDO

5KTX image
Crebbp Bromodomain In Complex With Cpd59 ((S)-1-(3-((2-Fluoro-4-(1-Methyl-1H-Pyrazol-4-Yl)Phenyl)Amino)-1-(Tetrahydrofuran-3-Yl)-6,7-Dihydro-1H-Pyrazolo[4,3-C]Pyridin-5(4H)-Yl)Ethanone)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.27 Å Release Date: 2016-11-02
Classification: TRANSFERASE
Ligands: 6XH, EDO, DMS

5KU3 image
Brd4 Bromodomain In Complex With Cpd59 ((S)-1-(3-((2-Fluoro-4-(1-Methyl-1H-Pyrazol-4-Yl)Phenyl)Amino)-1-(Tetrahydrofuran-3-Yl)-6,7-Dihydro-1H-Pyrazolo[4,3-C]Pyridin-5(4H)-Yl)Ethanone)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.14 Å Release Date: 2016-11-02
Classification: TRANSFERASE
Ligands: EDO, DMS, GOL, PEG, 6XH

3B0B image
Crystal Structure Of The Chicken Cenp-S/Cenp-X Complex

3B0C image
Crystal Structure Of The Chicken Cenp-T Histone Fold/Cenp-W Complex, Crystal Form I

3B0D image
Crystal Structure Of The Chicken Cenp-T Histone Fold/Cenp-W Complex, Crystal Form Ii

3VH5 image
Crystal Structure Of The Chicken Cenp-T Histone Fold/Cenp-W/Cenp-S/Cenp-X Heterotetrameric Complex, Crystal Form I

3VH6 image
Crystal Structure Of The Chicken Cenp-T Histone Fold/Cenp-W/Cenp-S/Cenp-X Heterotetrameric Complex, Crystal Form Ii
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