Search Count: 12
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A Potent And Selective Ror Gamma Inhibitor For The Treatment Of Autoimmune Diseases
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2026-04-29 Classification: DNA BINDING PROTEIN Ligands: A1MCM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-04-29
Ligands: A1MCM
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Crystal Structure Of The Mutant Human Ror Gamma Ligand Binding Domain With Jte-151
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2024-11-27 Classification: NUCLEAR PROTEIN/INHIBITOR Ligands: YAL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-27
Ligands: YAL
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Vascular Endothelial Protein Tyrosine Phosphatase In Complex With Cpd-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2024-02-28 Classification: HYDROLASE Ligands: EDO, U7C, EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-28
Ligands: EDO, U7C, EPE
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Vascular Endothelial Protein Tyrosine Phosphatase In Complex With Cpd-2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2024-02-28 Classification: HYDROLASE Ligands: U7L, EDO, EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-28
Ligands: U7L, EDO, EPE
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Crystal Structure Of Human Pyruvate Dehydrogenase Kinase 2 In Complex With Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.34 Å Release Date: 2021-08-04 Classification: TRANSFERASE/INHIBITOR Ligands: CL, ACT, DMS, W6P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-08-04
Ligands: CL, ACT, DMS, W6P
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Crystal Structure Of Human Pyruvate Dehydrogenase Kinase 2 In Complex With Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2021-08-04 Classification: TRANSFERASE Ligands: CL, ACT, DMS, 42A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-08-04
Ligands: CL, ACT, DMS, 42A
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Crystal Structure Of Human Pyruvate Dehydrogenase Kinase 4 In Complex With Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2021-08-04 Classification: TRANSFERASE Ligands: SO4, W6P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-08-04
Ligands: SO4, W6P
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Crystal Structure Of Human Pyruvate Dehydrogenase Kinase 4 In Complex With Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2021-08-04 Classification: TRANSFERASE Ligands: SO4, 42A, MG, ADP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-08-04
Ligands: SO4, 42A, MG, ADP
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Crystal Structure Of Human Pyruvate Dehydrogenase Kinase 4 In Complex With Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2021-08-04 Classification: TRANSFERASE Ligands: SO4, J0L, MG, ADP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-08-04
Ligands: SO4, J0L, MG, ADP
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Crystal Structure Of Human Pyruvate Dehydrogenase Kinase 2 In Complex With Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2021-08-04 Classification: TRANSFERASE Ligands: CL, ACT, DMS, J0F |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-08-04
Ligands: CL, ACT, DMS, J0F
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Discovery Of The Second Generation Ror Gamma Inhibitors Composed Of An Azole Scaffold.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2019-03-06 Classification: NUCLEAR PROTEIN/INHIBITOR Ligands: AYO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-06
Ligands: AYO
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Crystal Structure Of Yeast Cyclophilin A, Cpr1
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2003-11-18 Classification: ISOMERASE |
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION
Release Date: 2003-11-18
