Search Count: 40
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Crystal Structure Of Human Pla2G5 In Complex With A Smol Inhibitor (Compound 1)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2026-03-18 Classification: HYDROLASE Ligands: A1I5M, CA, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-03-18
Ligands: A1I5M, CA, CL
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Crystal Structure Of Human Map4K1 With An Inhibitor, Bay-405
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2024-06-26 Classification: TRANSFERASE Ligands: GOL, XON |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-26
Ligands: GOL, XON
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Crystal Structure Of Map4K1 With A Smol Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2024-06-26 Classification: TRANSFERASE Ligands: XOH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-26
Ligands: XOH
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Crystal Structure Of Map4K1 With A Smol Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2024-06-26 Classification: TRANSFERASE Ligands: XOR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-26
Ligands: XOR
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Crystal Structure Of Mst1 With A Map4K1 Smol Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2024-06-26 Classification: TRANSFERASE Ligands: XOZ, GOL, CXS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-26
Ligands: XOZ, GOL, CXS
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Crystal Structure Of Mst1 With A Map4K1 Smol Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2024-06-26 Classification: TRANSFERASE Ligands: ASP, XQL, GOL, CXS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-26
Ligands: ASP, XQL, GOL, CXS
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Crystal Structure Of Pparg And Ncor2 With An Inverse Agonist (Compound 7A)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2022-12-28 Classification: TRANSCRIPTION Ligands: Q2X, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-28
Ligands: Q2X, GOL
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Crystal Structure Of Pparg And Ncor2 With Sr10221, An Inverse Agonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2022-12-28 Classification: TRANSCRIPTION Ligands: A8R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-28
Ligands: A8R
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Crystal Structure Of Pparg And Ncor2 With An Inverse Agonist (Compound 7E)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2022-12-28 Classification: TRANSCRIPTION Ligands: Q33 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-28
Ligands: Q33
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Crystal Structure Of Mutant Pparg (C313A) And Ncor2 With An Inverse Agonist (Compound 7E)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2022-12-28 Classification: TRANSCRIPTION Ligands: Q33 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-28
Ligands: Q33
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Crystal Structure Of Pparg And Ncor2 With An Inverse Agonist (Compound 7D)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2022-12-28 Classification: TRANSCRIPTION Ligands: Q1R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-28
Ligands: Q1R
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Crystal Structure Of Mutant Pparg (C313A) And Ncor2 With An Inverse Agonist (Compound Si-1)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2022-12-28 Classification: TRANSCRIPTION Ligands: Q4O |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-28
Ligands: Q4O
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Crystal Structure Of Pparg And Ncor2 With An Inverse Agonist (Compound Si-2)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2022-12-28 Classification: TRANSCRIPTION Ligands: Q5X, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-28
Ligands: Q5X, SO4
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Crystal Structure Of Pparg And Ncor2 With An Inverse Agonist (Compound 15B)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2022-12-28 Classification: TRANSCRIPTION Ligands: Q8F |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-28
Ligands: Q8F
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Crystal Structure Of Pparg And Ncor2 With Bay-5516, An Inverse Agonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2022-12-28 Classification: TRANSCRIPTION Ligands: Q5O |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-28
Ligands: Q5O
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Crystal Structure Of Pparg And Ncor2 With Bay-9683, An Inverse Agonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2022-12-28 Classification: TRANSCRIPTION Ligands: Q4C |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-28
Ligands: Q4C
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Crystal Structure Of Pparg And Ncor2 With An Inverse Agonist (Compound 6A)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2022-11-09 Classification: TRANSCRIPTION Ligands: O2O |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: O2O
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Crystal Structure Of Pparg And Ncor2 With Bay-4931, An Inverse Agonist (Compound 6C)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2022-11-09 Classification: TRANSCRIPTION Ligands: O0U, GOL, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: O0U, GOL, CA
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X-Ray Structure Of Human Ldha With An Allosteric Inhibitor (Compound 3)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.91 Å Release Date: 2020-06-10 Classification: OXIDOREDUCTASE Ligands: L5N, NAI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-06-10
Ligands: L5N, NAI
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X-Ray Structure Of Human Ldh-A With An Allosteric Inhibitor (Compound 7)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2020-06-10 Classification: OXIDOREDUCTASE Ligands: L5K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-06-10
Ligands: L5K
