Search Count: 22
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Crystal Structure Of Casdatifan Bound To Hif2A-B*:Arnt-B* Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.56 Å Release Date: 2026-02-18 Classification: TRANSCRIPTION Ligands: A1I0H, FMT, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-02-18
Ligands: A1I0H, FMT, MG
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C-Terminal Bromodomain Of Human Brd2 With 7,8-Dimethoxy-3-Methyl-1,3-Dihydro-2H-Benzo[D]Azepin-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2022-11-30 Classification: TRANSCRIPTION Ligands: EDO, P4M, MES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-30
Ligands: EDO, P4M, MES
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C-Terminal Bromodomain Of Human Brd2 With (R)-7-((R)-1,2-Dihydroxyethyl)-1,3-Dimethyl-5-(1-Methyl-1H-Pyrazol-4-Yl)-1,3-Dihydro-2H-Benzo[D]Azepin-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2022-11-30 Classification: TRANSCRIPTION Ligands: EDO, 7PE, P4X |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-30
Ligands: EDO, 7PE, P4X
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C-Terminal Bromodomain Of Human Brd2 With 7,8-Dimethoxy-1,3-Dimethyl-1,3-Dihydro-2H-Benzo[D]Azepin-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2022-11-30 Classification: TRANSCRIPTION Ligands: EDO, PE4, P0U |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-30
Ligands: EDO, PE4, P0U
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C-Terminal Bromodomain Of Human Brd2 With 7,8-Dimethoxy-1,3-Dimethyl-1,3-Dihydro-2H-Benzo[D]Azepin-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2022-11-30 Classification: TRANSCRIPTION Ligands: EDO, PE4, P3R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-30
Ligands: EDO, PE4, P3R
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Crystal Structure Of Human Pi3K-Gamma In Complex With Compound 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.96 Å Release Date: 2021-11-03 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: V84 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-03
Ligands: V84
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Crystal Structure Of Human Pi3K-Gamma In Complex With Inhibitor Ipi-549
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.99 Å Release Date: 2020-09-16 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: V7Y, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-09-16
Ligands: V7Y, SO4
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Crystal Structure Of Human Pi3K-Gamma In Complex With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.88 Å Release Date: 2020-09-16 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: V81, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-09-16
Ligands: V81, SO4
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Human Ecto-5'-Nucleotidase (Cd73) In Complex With A2396 (Compound 74 In Publication) In The Closed Form In Crystal Form Iv
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2020-04-22 Classification: HYDROLASE Ligands: ZN, CA, PO4, O1H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-22
Ligands: ZN, CA, PO4, O1H
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Human Ecto-5'-Nucleotidase (Cd73) In Complex With A2410 (Compound 53 In Publication) In The Closed Form In Crystal Form Iv
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2020-04-22 Classification: HYDROLASE Ligands: ZN, CA, PO4, O1Q |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-22
Ligands: ZN, CA, PO4, O1Q
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Human Ecto-5'-Nucleotidase (Cd73) In Complex With A1618 (Compound 1B In Publication) In The Closed State In Crystal Form Iii
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2020-04-22 Classification: HYDROLASE Ligands: ZN, CA, O1T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-22
Ligands: ZN, CA, O1T
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Crystal Structure Of Cathepsin K With N-Desmethyl Thalassospiramide C
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2019-06-26 Classification: HYDROLASE Ligands: G4B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-26
Ligands: G4B
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Crystal Structure Of Human Hdac2 In Complex With (R)-6-[3,4-Dioxo-2-(4-Trifluoromethoxy-Phenylamino)-Cyclobut-1-Enylamino]-Heptanoic Acid Hydroxyamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2018-06-27 Classification: HYDROLASE Ligands: ZN, CA, NA, EL8, 1PE, SO4, PG4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-06-27
Ligands: ZN, CA, NA, EL8, 1PE, SO4, PG4
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Crystal Structure Of Human Caspase-1 With N-{3-[1-((S)-2-Hydroxy-5-Oxo-Tetrahydro-Furan-3-Ylcarbamoyl)-Ethyl]-1-Methyl-2,4-Dioxo-1,2,3,4-Tetrahydro-Pyrimidin-5-Yl}-4-(Quinoxalin-2-Ylamino)-Benzamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2018-05-02 Classification: HYDROLASE Ligands: CVE, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-02
Ligands: CVE, SO4
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Crystal Structure Of Human Caspase-1 With (3S,6S,10As)-N-((2S,3S)-2-Hydroxy-5-Oxotetrahydrofuran-3-Yl)-6-(Isoquinoline-1-Carboxamido)-5-Oxodecahydropyrrolo[1,2-A]Azocine-3-Carboxamide (Pge-3935199)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.53 Å Release Date: 2018-02-28 Classification: HYDROLASE Ligands: N7N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-02-28
Ligands: N7N
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Crystal Structure Of Human Caspase-1 With 2-((2-Naphthoyl)-L-Valyl)-4-Hydroxy-N-((3S)-2-Hydroxy-5-Oxotetrahydrofuran-3-Yl)-2-Azabicyclo[2.2.2]Octane-3-Carboxamide (Compound 1)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2017-12-20 Classification: HYDROLASE Ligands: WE0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-20
Ligands: WE0
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Crystal Structure Of The First Bacterial Vanadium Dependant Iodoperoxidase
Organism: Zobellia galactanivorans
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2014-10-08 Classification: TRANSFERASE Ligands: VO4, NA |
Organism: Zobellia galactanivorans
Method: X-RAY DIFFRACTION
Release Date: 2014-10-08
Ligands: VO4, NA
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Crystal Structure Of The First Bacterial Vanadium Dependant Iodoperoxidase
Organism: Zobellia galactanivorans
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2014-10-08 Classification: OXIDOREDUCTASE Ligands: VO4, NA |
Organism: Zobellia galactanivorans
Method: X-RAY DIFFRACTION
Release Date: 2014-10-08
Ligands: VO4, NA
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Crystal Structure Of A Monoclonal Antibody Directed Against An Antigenic Determinant Common To Ogawa And Inaba Serotypes Of Vibrio Cholerae O1
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2008-05-13 Classification: IMMUNE SYSTEM |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2008-05-13
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Crystal Structure Of An Anti-Carbohydrate Antibody Directed Against Vibrio Cholerae O1 In Complex With Antigen
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2000-08-02 Classification: IMMUNE SYSTEM |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2000-08-02
