Search Count: 14
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Crystal Structure Of Human Hdac2 In Complex With Tng260
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2025-09-17 Classification: HYDROLASE Ligands: A1B1V, ZN, CA, NHE, EDO, PEG, PGE, PG4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-17
Ligands: A1B1V, ZN, CA, NHE, EDO, PEG, PGE, PG4
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Crystal Structure Of Alpha-V Beta-1 Integrin Headpiece In Complex With Tr01225179
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2025-01-01 Classification: CELL ADHESION Ligands: CA, NAG, A1AFA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-01
Ligands: CA, NAG, A1AFA
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Structure-Guided Optimization Of A Novel Class Of Ask1 Inhibitors With Increased Sp3 Character And An Exquisite Selectivity Profile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2020-08-12 Classification: METAL BINDING PROTEIN Ligands: V3S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-12
Ligands: V3S
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Structure-Based Design Of Ask1 Inhibitors As Potential First-In-Class Agents For Heart Failure
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2017-06-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 8GV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-07
Ligands: SO4, 8GV
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Structure-Based Design Of Ask1 Inhibitors As Potential First-In-Class Agents For Heart Failure
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2017-06-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 8GY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-07
Ligands: 8GY
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Structure-Based Design Of Ask1 Inhibitors As Potential First-In-Class Agents For Heart Failure
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.95 Å Release Date: 2017-06-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 8GS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-07
Ligands: 8GS
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Discovery Of A Novel, Potent And Selective Inhibitor Of 3-Phosphoinositide Dependent Kinase (Pdk1)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2011-11-16 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GOL, SO4, ABQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-11-16
Ligands: GOL, SO4, ABQ
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Discovery Of A Novel, Potent And Selective Inhibitor Of 3-Phosphoinositide Dependent Kinase (Pdk1)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2011-11-16 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3RW, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-11-16
Ligands: 3RW, GOL, SO4
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Novel Isoquinolone Pdk1 Inhibitors Discovered Through Fragment-Based Lead Discovery
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2011-10-26 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3S1, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-26
Ligands: 3S1, SO4, GOL
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Guinea Pig 11Beta Hydroxysteroid Dehydrogenase With Pf-877423
Organism: Cavia porcellus
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2011-05-04 Classification: Oxidoreductase/Oxidoreductase inhibitor Ligands: NAP, A0D |
Organism: Cavia porcellus
Method: X-RAY DIFFRACTION
Release Date: 2011-05-04
Ligands: NAP, A0D
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Characterization Of The Chk1 Allosteric Inhibitor Binding Site
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2009-10-06 Classification: TRANSFERASE Ligands: AGX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-10-06
Ligands: AGX
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Characterization Of The Chk1 Allosteric Inhibitor Binding Site
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2009-10-06 Classification: TRANSFERASE Ligands: AGY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-10-06
Ligands: AGY
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N-(Pyridin-2-Yl) Arylsulfonamide Inhibitors Of 11B-Hydroxysteroid Dehydrogenase Type 1: Discovery Of Pf-915275
Organism: Cavia porcellus
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2009-08-04 Classification: Oxidoreductase/Oxidoreductase inhibitor Ligands: NAP, 3G4 |
Organism: Cavia porcellus
Method: X-RAY DIFFRACTION
Release Date: 2009-08-04
Ligands: NAP, 3G4
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Active-Site Mobility In Human Immunodeficiency Virus Type 1 Protease As Demonstrated By Crystal Structure Of A28S Mutant
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 1998-04-15 Classification: ASPARTYL PROTEASE Ligands: U0E |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 1998-04-15
Ligands: U0E