Search Count: 31
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Crystal Structure Of Human Wrn Helicase With Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.42 Å Release Date: 2026-05-13 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, A1C4J, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-05-13
Ligands: ZN, A1C4J, EDO
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Crystal Structure Of Human Wrn Helicase With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.37 Å Release Date: 2026-05-13 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, A1C4L, CL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-05-13
Ligands: ZN, A1C4L, CL, EDO
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Crystal Structure Of Human Wrn Helicase With Compound 26
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.58 Å Release Date: 2026-05-13 Classification: HYDROLASE Ligands: A1C4O, ATP, ZN, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-05-13
Ligands: A1C4O, ATP, ZN, EDO
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Crystal Structure Of Cdk2 Bound By Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.16 Å Release Date: 2025-09-10 Classification: TRANSFERASE Ligands: A1INI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-10
Ligands: A1INI
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Crystal Structure Of Cdk2-Cyclin E1 Bound By Compound 30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.16 Å Release Date: 2025-09-10 Classification: TRANSFERASE Ligands: A1IOI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-10
Ligands: A1IOI
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Crystal Structure Of Cdk2-Cyclin E1 Bound By Compound 11 (Azd8421)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2025-09-10 Classification: TRANSFERASE Ligands: A1IOP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-10
Ligands: A1IOP
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Crystal Structure Of Human 15-Pgdh In Complex With Small Molecule Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2025-09-10 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: A1CH2, NAD, IOD, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-10
Ligands: A1CH2, NAD, IOD, EDO, GOL
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Crystal Structure Of Human 15-Pgdh In Complex With Small Molecule Compound 8B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2025-09-03 Classification: OXIDOREDUCTASE Ligands: NAD, SWL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-03
Ligands: NAD, SWL, EDO
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Crystal Structure Of Parp1 Catalytic Domain Bound To Azd5305 (Saruparib)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2024-12-04 Classification: TRANSFERASE Ligands: A1H63, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-04
Ligands: A1H63, SO4
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Crystal Structure Of Parp1 Catalytic Domain Bound To Azd9574
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2024-12-04 Classification: TRANSFERASE Ligands: A1H64, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-04
Ligands: A1H64, SO4
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Crystal Structure Of The Tyk2 Pseudokinase Domain In Complex With Compound 8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2023-07-26 Classification: TRANSFERASE Ligands: ZRU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-26
Ligands: ZRU
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Crystal Structure Of The Tyk2 Pseudokinase Domain In Complex With Compound 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.71 Å Release Date: 2023-07-26 Classification: TRANSFERASE Ligands: ZS3, EDO, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-26
Ligands: ZS3, EDO, ACT
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Crystal Structure Of The Tyk2 Pseudokinase Domain In Complex With Tak-279
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2023-07-26 Classification: TRANSFERASE Ligands: ZSB, ACT, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-26
Ligands: ZSB, ACT, EDO
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Syk Kinase Domain In Complex With Macrocyclic Inhibitor 20A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.51 Å Release Date: 2023-06-14 Classification: TRANSFERASE Ligands: QR7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-14
Ligands: QR7
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Crystal Structure Of Tyk2 Kinase Domain In Complex With Compound 12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2022-08-24 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: OVI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-24
Ligands: OVI
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Crystal Structure Of Tyk2 Kinase Domain In Complex With Compound 16
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2022-08-24 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: OVC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-24
Ligands: OVC
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Crystal Structure Of Tyk2 Kinase Domain In Complex With Compound 25
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2022-08-24 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: OV5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-24
Ligands: OV5
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Crystal Structure Of Tyk2 Kinase Domain In Complex With Compound 30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2022-08-24 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: OV0, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-24
Ligands: OV0, SO4
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Crystal Structure Of Jak3 Kinase Domain In Complex With Compound 25
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2022-08-24 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: OV5, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-24
Ligands: OV5, CL
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Crystal Structure Of Jak2 Kinase Domain In Complex With Compound 30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.51 Å Release Date: 2022-08-24 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: OV0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-24
Ligands: OV0
