Search Count: 23
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Protein Kinase Mkk7 In Complex With Phenethyltriazole-Substituted Pyrazolopyrimidine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2022-07-20 Classification: TRANSFERASE Ligands: 2GI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-07-20
Ligands: 2GI
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Protein Kinase Mkk7 In Complex With Difluoro-Phenethyltriazole-Substituted Pyrazolopyrimidine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2022-07-20 Classification: TRANSFERASE Ligands: 24N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-07-20
Ligands: 24N
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Protein Kinase Mkk7 In Complex With 5-Bromo-2-Hydroxyphenyl-Substituted Pyrazolopyrimidine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2022-07-20 Classification: TRANSFERASE Ligands: GOL, 2I5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-07-20
Ligands: GOL, 2I5
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Protein Kinase Mkk7 In Complex With Methoxycyclohexyl-Substituted Indazole
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2022-07-20 Classification: TRANSFERASE Ligands: 1XZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-07-20
Ligands: 1XZ
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Protein Kinase Mkk7 In Complex With Cyclobutyl-Substituted Indazole
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2022-07-20 Classification: TRANSFERASE Ligands: 21I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-07-20
Ligands: 21I
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Protein Kinase Mkk7 In Complex With Tolyl-Substituted Indazole
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2022-07-20 Classification: TRANSFERASE Ligands: 2I8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-07-20
Ligands: 2I8
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Crystal Structure Analysis Of Human Pin1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.42 Å Release Date: 2020-12-30 Classification: ISOMERASE/ISOMERASE INHIBITOR Ligands: QT7, SO4, PG4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-30
Ligands: QT7, SO4, PG4
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Ligand-Induced Aziridine-Formation At The Yeast Proteasomal Subunit Beta5 By Sulfonate Esters
Organism: Saccharomyces cerevisiae (strain atcc 204508 / s288c)
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2017-04-26 Classification: HYDROLASE Ligands: MG, 3K4 |
Organism: Saccharomyces cerevisiae (strain atcc 204508 / s288c)
Method: X-RAY DIFFRACTION
Release Date: 2017-04-26
Ligands: MG, 3K4
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Ligand-Induced Lys33-Thr1 Crosslinking At The Yeast Proteasomal Subunit Beta5 By Sulfonate Esters
Organism: Saccharomyces cerevisiae (strain atcc 204508 / s288c)
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2017-04-26 Classification: HYDROLASE Ligands: MG |
Organism: Saccharomyces cerevisiae (strain atcc 204508 / s288c)
Method: X-RAY DIFFRACTION
Release Date: 2017-04-26
Ligands: MG
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Yeast 20S Proteasome With Human Beta5I (1-138) And Human Beta6 (97-111; 118-133) In Complex With Thiazole Based Inhibitor Ro19
Organism: Homo sapiens, Saccharomyces cerevisiae s288c, Saccharomyces cerevisiae (strain atcc 204508 / s288c)
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2017-01-25 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: MG, CL, 7DX |
Organism: Homo sapiens, Saccharomyces cerevisiae s288c, Saccharomyces cerevisiae (strain atcc 204508 / s288c)
Method: X-RAY DIFFRACTION
Release Date: 2017-01-25
Ligands: MG, CL, 7DX
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Yeast 20S Proteasome Beta5-G48C Mutant In Complex With Alpha-Chloroacetamide 5
Organism: Synthetic construct, Saccharomyces cerevisiae s288c
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2015-12-02 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: MG, CL, MES, 54L |
Organism: Synthetic construct, Saccharomyces cerevisiae s288c
Method: X-RAY DIFFRACTION
Release Date: 2015-12-02
Ligands: MG, CL, MES, 54L
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Yeast 20S Proteasome Beta5-G48C Mutant
Organism: Saccharomyces cerevisiae (strain atcc 204508 / s288c), Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2015-11-25 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: MG, CL |
Organism: Saccharomyces cerevisiae (strain atcc 204508 / s288c), Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2015-11-25
Ligands: MG, CL
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Yeast 20S Proteasome Beta5-G48C Mutant In Complex With Alpha-Chloroacetamide 1
Organism: Saccharomyces cerevisiae (strain atcc 204508 / s288c), Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2015-11-25 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: MG, CL, MES |
Organism: Saccharomyces cerevisiae (strain atcc 204508 / s288c), Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2015-11-25
Ligands: MG, CL, MES
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Yeast 20S Proteasome Beta5-G48C Mutant In Complex With Onx 0914
Organism: Synthetic construct, Saccharomyces cerevisiae (strain atcc 204508 / s288c)
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2015-11-25 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: MG, CL, MES, 04C, NA |
Organism: Synthetic construct, Saccharomyces cerevisiae (strain atcc 204508 / s288c)
Method: X-RAY DIFFRACTION
Release Date: 2015-11-25
Ligands: MG, CL, MES, 04C, NA
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Yeast 20S Proteasome In Complex With Macyranone A
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2015-02-18 Classification: HYDROLASE Ligands: MG, CL, 7IM, MES |
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION
Release Date: 2015-02-18
Ligands: MG, CL, 7IM, MES
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Ligand-Induced Aziridine-Formation At Subunit Beta5 Of The Yeast 20S Proteasome
Organism: Saccharomyces cerevisiae s288c
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2014-10-15 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: MG, 3K4 |
Organism: Saccharomyces cerevisiae s288c
Method: X-RAY DIFFRACTION
Release Date: 2014-10-15
Ligands: MG, 3K4
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Ligand-Induced Lys33-Thr1 Crosslinking At Subunit Beta5 Of The Yeast 20S Proteasome
Organism: Saccharomyces cerevisiae s288c
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2014-10-15 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: MG, ABA |
Organism: Saccharomyces cerevisiae s288c
Method: X-RAY DIFFRACTION
Release Date: 2014-10-15
Ligands: MG, ABA
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Ycp In Complex With Mg132
Organism: Saccharomyces cerevisiae s288c
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2014-02-12 Classification: HYDROLASE/HYDROLASE Inhibitor Ligands: MG, ALD |
Organism: Saccharomyces cerevisiae s288c
Method: X-RAY DIFFRACTION
Release Date: 2014-02-12
Ligands: MG, ALD
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Ycp In Complex With Z-Leu-Leu-Leu-Ketoaldehyde
Organism: Saccharomyces cerevisiae s288c
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2014-02-12 Classification: HYDROLASE/HYDROLASE Inhibitor Ligands: MG, 2MK |
Organism: Saccharomyces cerevisiae s288c
Method: X-RAY DIFFRACTION
Release Date: 2014-02-12
Ligands: MG, 2MK
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Ycp In Complex With Z-Leu-Leu-Leu-B(Oh)2
Organism: Saccharomyces cerevisiae s288c
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2014-02-12 Classification: HYDROLASE/HYDROLASE Inhibitor Ligands: MG, CIX |
Organism: Saccharomyces cerevisiae s288c
Method: X-RAY DIFFRACTION
Release Date: 2014-02-12
Ligands: MG, CIX
