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Crystal Structure Of The Nuak1-Mark3 Kinase Domain Chimera Bound With Small Molecule Inhibitor 2-Amino-N-(5-((5-Chloro-4-(((3R,3Ar,6R,6Ar)-6-Methoxyhexahydrofuro[3,2-B]Furan-3-Yl)Oxy)Pyrimidin-2-Yl)Amino)-2-((2-(Dimethylamino)Ethyl)(Methyl)Amino)Phenyl)Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2026-04-22 Classification: TRANSFERASE Ligands: A1ER0 |
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Crystal Structure Of The Nuak1-Mark3 Kinase Domain Chimera Bound With Small Molecule Inhibitor 4-((5-((5-Chloro-4-(((3R,3Ar,6R,6Ar)-6-Methoxyhexahydrofuro[3,2-B]Furan-3-Yl)Oxy)Pyrimidin-2-Yl)Amino)-2-((2-(Dimethylamino)Ethyl)(Methyl)Amino)Phenyl)Carbamoyl)-1-Methyl-3H-Pyrazol-1-Ium-3-Ide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2026-04-22 Classification: CYTOSOLIC PROTEIN Ligands: A1ER9 |
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Crystal Structure Of The Nuak1-Mark3 Kinase Domain Chimera Bound With Small Molecule Inhibitor N-(5-((5-Chloro-4-(((3As,6R,6Ar)-6-Methoxy-3A,5,6,6A-Tetrahydrofuro[3,2-B]Furan-3-Yl)Oxy)Pyrimidin-2-Yl)Amino)-2-(((2R,7Ar)-2-Fluorotetrahydro-1H-Pyrrolizin-7A(5H)-Yl)Methoxy)Phenyl)-1-Methyl-1H-Pyrazole-4-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2026-04-22 Classification: CYTOSOLIC PROTEIN Ligands: A1ESF |
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Organism: Equus caballus
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2025-12-24 Classification: METAL BINDING PROTEIN Ligands: CU, SO4, NA |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2025-12-03 Classification: UNKNOWN FUNCTION |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2025-12-03 Classification: UNKNOWN FUNCTION |
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Crystal Structure Of Cdk12/Cyclin K In Complex With Covalent Inhibitor Yjz5118
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.72 Å Release Date: 2025-05-07 Classification: TRANSFERASE Ligands: EDO, A1EB3, MG, PEG |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.95 Å Release Date: 2025-02-12 Classification: LIGASE Ligands: CL, A1LY0 |
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Crystal Structure Of Hpk1 Kinase Domain T165E,S171E Phosphomimetic Mutant In Complex With Compound 9F
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2024-04-10 Classification: TRANSFERASE Ligands: A1LVT |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2024-01-31 Classification: HYDROLASE Ligands: GDP, MG, DWI |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2024-01-31 Classification: HYDROLASE Ligands: GDP, MG, DNU |
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Organism: Escherichia coli (strain k12)
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2023-10-18 Classification: DNA BINDING PROTEIN Ligands: ZN, ADP, MG |
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Organism: Escherichia coli k-12
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2023-10-18 Classification: DNA BINDING PROTEIN Ligands: AGS, ZN |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2023-09-27 Classification: HYDROLASE Ligands: ZLL, MG |
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The Crystal Structure Of Trka(F589L) Kinase In Complex With N-(3-Cyclopropyl-5-((4-Methylpiperazin-1-Yl)Methyl)Phenyl)-4^6-Methyl-14-Oxo-5-Oxa-13-Aza-1(3,6)-Imidazo[1,2-B]Pyridazina-4(1,3)-Benzenacyclotetradecaphan-2-Yne-4^5-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.28 Å Release Date: 2023-09-20 Classification: TRANSFERASE Ligands: A4U |
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The Crystal Structure Of Trka(G595R) Kinase In Complex With N-(3-Cyclopropyl-5-((4-Methylpiperazin-1-Yl)Methyl)Phenyl)-4^6-Methyl-14-Oxo-5-Oxa-13-Aza-1(3,6)-Imidazo[1,2-B]Pyridazina-4(1,3)-Benzenacyclotetradecaphan-2-Yne-4^5-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2023-09-20 Classification: TRANSFERASE Ligands: A4U |
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The Crystal Structure Of Trka Kinase In Complex With 4^6-Methyl-N-(3-(4-Methyl-1H-Imidazol-1-Yl)-5-(Trifluoromethyl)Phenyl)-14-Oxo-5-Oxa-13-Aza-1(3,6)-Imidazo[1,2-B]Pyridazina-4(1,3)-Benzenacyclotetradecaphan-2-Yne-4^5-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.05 Å Release Date: 2023-09-20 Classification: TRANSFERASE Ligands: A0X |
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The Crystal Structure Of Trka Kinase In Complex With 4^6-Methyl-N-(3-(4-Methyl-1H-Imidazol-1-Yl)-5-(Trifluoromethyl)Phenyl)-11-Oxo-5-Oxa-10,14-Diaza-1(3,6)-Imidazo[1,2-B]Pyridazina-4(1,3)-Benzenacyclotetradecaphan-2-Yne-4^5-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2023-09-20 Classification: TRANSFERASE Ligands: A6X |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2023-08-09 Classification: STRUCTURAL PROTEIN/INHIBITOR Ligands: IGS |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.54 Å Release Date: 2023-08-09 Classification: STRUCTURAL PROTEIN/INHIBITOR Ligands: IGV |