Search Count: 33
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Factor Xia In Complex With Compound 2A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2022-08-03 Classification: Blood Clotting, Hydrolase Ligands: OQ6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-03
Ligands: OQ6
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Factor Xia In Complex With Compound 2D
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2022-08-03 Classification: BLOOD CLOTTING, Hydrolase Ligands: OQI, CIT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-03
Ligands: OQI, CIT
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Factor Xia In Complex With Compound 2E
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.47 Å Release Date: 2022-08-03 Classification: BLOOD CLOTTING, hydrolase Ligands: OQO, CIT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-03
Ligands: OQO, CIT
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Factor Xia In Complex With Compound 2F
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2022-08-03 Classification: BLOOD CLOTTING, Hydrolase Ligands: OR0, CIT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-03
Ligands: OR0, CIT
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Factor Xia In Complex With Compound 2G
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2022-08-03 Classification: BLOOD CLOTTING, Hydrolase Ligands: CIT, ORF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-03
Ligands: CIT, ORF
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Factor Xia In Complex With Compound 2H
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2022-08-03 Classification: BLOOD CLOTTING, Hydrolase Ligands: CIT, ORU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-03
Ligands: CIT, ORU
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Factor Xia In Complex With Compound 2I
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2022-08-03 Classification: BLOOD CLOTTING, Hydrolase Ligands: CIT, OSX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-03
Ligands: CIT, OSX
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Factor Xia In Complex With Compound 2J
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.51 Å Release Date: 2022-08-03 Classification: BLOOD CLOTTING, Hydrolase Ligands: CIT, OT7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-03
Ligands: CIT, OT7
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Factor Xia In Complex With Compound 2K
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2022-08-03 Classification: BLOOD CLOTTING, Hydrolase Ligands: CIT, OTL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-03
Ligands: CIT, OTL
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Factor Xia In Complex With Compound 3F
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2022-08-03 Classification: BLOOD CLOTTING, Hydrolase Ligands: CIT, OTX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-03
Ligands: CIT, OTX
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Molecular Mechanism And Structural Basis Of Small-Molecule Modulation Of Acid-Sensing Ion Channel 1 (Asic1)
Organism: Gallus gallus
Method: X-RAY DIFFRACTION Resolution:3.01 Å Release Date: 2020-12-30 Classification: TRANSPORT PROTEIN Ligands: NAG, UZG, NA |
Organism: Gallus gallus
Method: X-RAY DIFFRACTION
Release Date: 2020-12-30
Ligands: NAG, UZG, NA
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Structure Of A Hit For G Protein Coupled Receptor Kinase 2 (Grk2) Inhibitor For The Potential Treatment Of Heart Failure
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.54 Å Release Date: 2020-10-28 Classification: SIGNALING PROTEIN,TRANSFERASE/INHIBITOR Ligands: MG, W4D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-10-28
Ligands: MG, W4D
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Structure Of A Hit For G Protein Coupled Receptor Kinase 2 (Grk2) Inhibitor For The Potential Treatment Of Heart Failure
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.61 Å Release Date: 2020-10-28 Classification: SIGNALING PROTEIN,TRANSFERASE/INHIBITOR Ligands: W4G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-10-28
Ligands: W4G
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Crystal Structure Of A Soluble Form Of Human Mgll In Complex With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.35 Å Release Date: 2011-03-02 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZYH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-02
Ligands: ZYH
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Cfms Tyrosine Kinase In Complex With 4-Cyano-1H-Imidazole-2-Carboxylic Acid (2-Cyclohex-1-Enyl-4-Piperidin-4-Yl-Phenyl)-Amide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2010-12-01 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ACT, KRJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-12-01
Ligands: ACT, KRJ
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Cfms Tyrosine Kinase In Complex With 5-Cyano-Furan-2-Carboxylic Acid [4-(4-Methyl-Piperazin-1-Yl)-2-Piperidin-1-Yl-Phenyl]-Amide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2010-12-01 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: KRL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-12-01
Ligands: KRL, SO4
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Cfms Tyrosine Kinase In Complex With A Pyridopyrimidinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2009-02-17 Classification: TRANSFERASE Ligands: SO4, 8C5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-02-17
Ligands: SO4, 8C5
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Cfms Tyrosine Kinase (Tie2 Kid) In Complex With A Pyrimidinopyridone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2008-07-15 Classification: TRANSFERASE Ligands: SO4, IXH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-07-15
Ligands: SO4, IXH
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X-Ray Structure Of Novel Biaryl-Based Dipeptidyl Peptidase Iv Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2005-11-08 Classification: HYDROLASE Ligands: NAG, JNH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-11-08
Ligands: NAG, JNH
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Use Of Papain As A Model For The Structure-Based Design Of Cathepsin K Inhibitors. Crystal Structures Of Two Papain Inhibitor Complexes Demonstrate Binding To S'-Subsites.
Organism: Carica papaya
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 1999-08-16 Classification: HYDROLASE Ligands: SBA |
Organism: Carica papaya
Method: X-RAY DIFFRACTION
Release Date: 1999-08-16
Ligands: SBA
