Search Count: 15
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Inhibitor Bound Vim1
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION Resolution:1.15 Å Release Date: 2024-10-16 Classification: HYDROLASE Ligands: MG, ZN, A1AUQ |
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION
Release Date: 2024-10-16
Ligands: MG, ZN, A1AUQ
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Inhibitor Bound Vim1
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION Resolution:1.01 Å Release Date: 2023-05-24 Classification: HYDROLASE Ligands: ZN, OKC |
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION
Release Date: 2023-05-24
Ligands: ZN, OKC
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Inhibitor Bound Vim1
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION Resolution:1.11 Å Release Date: 2023-05-24 Classification: HYDROLASE Ligands: ZN, OK0 |
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION
Release Date: 2023-05-24
Ligands: ZN, OK0
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Inhibitor Bound Vim1
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION Resolution:1.02 Å Release Date: 2023-05-24 Classification: HYDROLASE Ligands: MG, ZN, OJR |
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION
Release Date: 2023-05-24
Ligands: MG, ZN, OJR
 |
Inhibitor Bound Vim1
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION Resolution:1.00 Å Release Date: 2023-05-24 Classification: HYDROLASE Ligands: EDO, ACT, ZN |
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION
Release Date: 2023-05-24
Ligands: EDO, ACT, ZN
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Ndm1-Inhibitor Co-Structure
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION Resolution:0.99 Å Release Date: 2023-03-08 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ACT, CA, ZN, CD, O0L |
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION
Release Date: 2023-03-08
Ligands: ACT, CA, ZN, CD, O0L
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Ndm1-Inhibitor Co-Structure
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION Resolution:1.47 Å Release Date: 2023-03-08 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, CD, O0F |
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION
Release Date: 2023-03-08
Ligands: ZN, CD, O0F
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Ndm1-Inhibitor Co-Structure
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION Resolution:1.11 Å Release Date: 2023-03-08 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, CD, NZR |
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION
Release Date: 2023-03-08
Ligands: ZN, CD, NZR
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Ndm1-Inhibitor Co-Structure
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION Resolution:1.13 Å Release Date: 2023-03-08 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, NZR |
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION
Release Date: 2023-03-08
Ligands: ZN, NZR
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Ndm1-Inhibitor Co-Structure
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2023-03-08 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: CD, ZN, NZ0, EPE |
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION
Release Date: 2023-03-08
Ligands: CD, ZN, NZ0, EPE
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Discovery Of Mk-8353: An Orally Bioavailable Dual Mechanism Erk Inhibitor For Oncology
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2018-08-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, G67 |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2018-08-08
Ligands: SO4, G67
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Discovery Of 3(S)-Thiomethyl Pyrrolidine Erk Inhibitors For Oncology
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2018-05-23 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: SO4, F8V |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2018-05-23
Ligands: SO4, F8V
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Dissecting Therapeutic Resistance To Erk Inhibition Rat Wild Type Sch772984 In Complex With (3R)-1-(2-Oxo-2-{4-[4-(Pyrimidin-2-Yl)Phenyl]Piperazin-1-Yl}Ethyl)-N-[3-(Pyridin-4-Yl)-2H-Indazol-5-Yl]Pyrrolidine-3-Carboxamide
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2016-02-24 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 38Z, SO4, PG4, DMS |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2016-02-24
Ligands: 38Z, SO4, PG4, DMS
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Dissecting Therapeutic Resistance To Erk Inhibition Rat Mutant Sch772984 In Complex With (3R)-1-(2-Oxo-2-{4-[4-(Pyrimidin-2-Yl)Phenyl]Piperazin-1-Yl}Ethyl)-N-[3-(Pyridin-4-Yl)-2H-Indazol-5-Yl]Pyrrolidine-3-Carboxamide
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2016-02-24 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 38Z, SO4 |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2016-02-24
Ligands: 38Z, SO4
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Discovery Of Novel, Dual Mechanism Erk Inhibitors By Affinity Selection Screening Of An Inactive Kinase State
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2014-11-12 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3G7, SO4 |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2014-11-12
Ligands: 3G7, SO4