Search Count: 20
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Crystal Structure Matriptase (C731S) In Complex With Inhibitor Mm1132-2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.35 Å Release Date: 2024-07-10 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: SO4, CL, GOL, YIL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-07-10
Ligands: SO4, CL, GOL, YIL
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Crystal Structure Matriptase (C731S) In Complex With Inhibitor Vd4162B
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.20 Å Release Date: 2024-02-07 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: CL |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2024-02-07
Ligands: CL
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2.05 A Resolution Structure Of Mers 3Cl Protease In Complex With Inhibitor Gc376
Organism: Middle east respiratory syndrome-related coronavirus
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2018-04-04 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: CA, B1S, K36 |
Organism: Middle east respiratory syndrome-related coronavirus
Method: X-RAY DIFFRACTION
Release Date: 2018-04-04
Ligands: CA, B1S, K36
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1.55 A Resolution Structure Of Mers 3Cl Protease In Complex With Inhibitor Gc813
Organism: Middle east respiratory syndrome-related coronavirus
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2018-04-04 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: PG4, MG, AW4, B3G |
Organism: Middle east respiratory syndrome-related coronavirus
Method: X-RAY DIFFRACTION
Release Date: 2018-04-04
Ligands: PG4, MG, AW4, B3G
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1.85 A Resolution Structure Of Mers 3Cl Protease In Complex With Piperidine-Based Peptidomimetic Inhibitor 17
Organism: Middle east respiratory syndrome-related coronavirus
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2018-04-04 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: AVY, B3J |
Organism: Middle east respiratory syndrome-related coronavirus
Method: X-RAY DIFFRACTION
Release Date: 2018-04-04
Ligands: AVY, B3J
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2.25 A Resolution Structure Of Mers 3Cl Protease In Complex With Piperidine-Based Peptidomimetic Inhibitor 21
Organism: Middle east respiratory syndrome-related coronavirus
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2018-04-04 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: N02, B6Y |
Organism: Middle east respiratory syndrome-related coronavirus
Method: X-RAY DIFFRACTION
Release Date: 2018-04-04
Ligands: N02, B6Y
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1.95 A Resolution Structure Of Norovirus 3Cl Protease In Complex With A Dipeptidyl Oxazolidinone-Based Inhibitor
Organism: Norwalk virus
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2017-12-13 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: V45 |
Organism: Norwalk virus
Method: X-RAY DIFFRACTION
Release Date: 2017-12-13
Ligands: V45
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1.40 A Resolution Structure Of Norovirus 3Cl Protease In Complex With The A M-Chlorophenyl Substituted Macrocyclic Inhibitor (17-Mer)
Organism: Norwalk virus
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2017-01-11 Classification: PROTEASE/PROTEASE INHIBITOR Ligands: CL, V56 |
Organism: Norwalk virus
Method: X-RAY DIFFRACTION
Release Date: 2017-01-11
Ligands: CL, V56
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1.75 A Resolution Structure Of Norovirus 3Cl Protease In Complex With The A N-Pentyl Substituted Macrocyclic Inhibitor (17-Mer)
Organism: Norwalk virus
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2017-01-11 Classification: PROTEASE/PROTEASE INHIBITOR Ligands: V69 |
Organism: Norwalk virus
Method: X-RAY DIFFRACTION
Release Date: 2017-01-11
Ligands: V69
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2.10 A Resolution Structure Of Norovirus 3Cl Protease In Complex With The Dipeptidyl Inhibitor 7L (Hexagonal Form)
Organism: Norwalk virus
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2016-11-23 Classification: PROTEASE/PROTEASE INHIBITOR Ligands: N38 |
Organism: Norwalk virus
Method: X-RAY DIFFRACTION
Release Date: 2016-11-23
Ligands: N38
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1.90 A Resolution Structure Of Norovirus 3Cl Protease In Complex With The Dipeptidyl Inhibitor 7L (Orthorhombic P Form)
Organism: Norwalk virus
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2016-11-23 Classification: PROTEASE/PROTEASE INHIBITOR Ligands: N38 |
Organism: Norwalk virus
Method: X-RAY DIFFRACTION
Release Date: 2016-11-23
Ligands: N38
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2.45 A Resolution Structure Of Norovirus 3Cl Protease In Complex With The Dipeptidyl Inhibitor 7M (Hexagonal Form)
Organism: Norwalk virus
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2016-11-23 Classification: PROTEASE/PROTEASE INHIBITOR Ligands: N40 |
Organism: Norwalk virus
Method: X-RAY DIFFRACTION
Release Date: 2016-11-23
Ligands: N40
 |
1.20 A Resolution Structure Of Norovirus 3Cl Protease In Complex With A Triazole-Based Macrocyclic (17-Mer) Inhibitor
Organism: Norwalk virus
Method: X-RAY DIFFRACTION Resolution:1.20 Å Release Date: 2016-05-04 Classification: PROTEASE/PROTEASE INHIBITOR Ligands: CL, 5LG |
Organism: Norwalk virus
Method: X-RAY DIFFRACTION
Release Date: 2016-05-04
Ligands: CL, 5LG
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1.95 A Resolution Structure Of Norovirus 3Cl Protease In Complex With A Triazole-Based Macrocyclic (18-Mer) Inhibitor
Organism: Norwalk virus
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2016-05-04 Classification: PROTEASE/PROTEASE INHIBITOR Ligands: 5LH, GOL |
Organism: Norwalk virus
Method: X-RAY DIFFRACTION
Release Date: 2016-05-04
Ligands: 5LH, GOL
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1.20 A Resolution Structure Of Norovirus 3Cl Protease In Complex With A Triazole-Based Macrocyclic (21-Mer) Inhibitor
Organism: Norwalk virus
Method: X-RAY DIFFRACTION Resolution:1.20 Å Release Date: 2016-05-04 Classification: PROTEASE/PROTEASE INHIBITOR Ligands: CL, 5LJ |
Organism: Norwalk virus
Method: X-RAY DIFFRACTION
Release Date: 2016-05-04
Ligands: CL, 5LJ
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2.35A Resolution Structure Of Norovirus 3Cl Protease In Complex An Oxadiazole-Based, Cell Permeable Macrocyclic (21-Mer) Inhibitor
Organism: Norwalk virus
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2016-02-10 Classification: HYDROLASE/HYDROLASE Inhibitor Ligands: CL, V66 |
Organism: Norwalk virus
Method: X-RAY DIFFRACTION
Release Date: 2016-02-10
Ligands: CL, V66
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1.0A Resolution Structure Of Norovirus 3Cl Protease In Complex An Oxadiazole-Based, Cell Permeable Macrocyclic (20-Mer) Inhibitor
Organism: Norwalk virus
Method: X-RAY DIFFRACTION Resolution:1.00 Å Release Date: 2016-02-10 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: V64 |
Organism: Norwalk virus
Method: X-RAY DIFFRACTION
Release Date: 2016-02-10
Ligands: V64
 |
1.85A Resolution Structure Of Norovirus 3Cl Protease Complex With A Covalently Bound Dipeptidyl Inhibitor Diethyl [(1R,2S)-2-[(N-{[(3-Chlorobenzyl)Oxy]Carbonyl}-3-Cyclohexyl-L-Alanyl)Amino]-1-Hydroxy-3-(2-Oxo-2H-Pyrrol-3-Yl)Propyl]Phosphonate
Organism: Norwalk virus (strain gi/human/united states/norwalk/1968)
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2015-03-25 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 3ZR, SO4 |
Organism: Norwalk virus (strain gi/human/united states/norwalk/1968)
Method: X-RAY DIFFRACTION
Release Date: 2015-03-25
Ligands: 3ZR, SO4
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1.60 A Resolution Structure Of Norovirus 3Cl Protease Complex With A Covalently Bound Dipeptidyl Inhibitor (1R,2S)-2-({N-[(Benzyloxy)Carbonyl]-3-Cyclohexyl-L-Alanyl}Amino)-1-Hydroxy-3-[(3S)-2-Oxopyrrolidin-3-Yl]Propane-1-Sulfonic Acid (Hexagonal Form)
Organism: Norwalk virus (strain gi/human/united states/norwalk/1968)
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2015-03-25 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: M40, PG4 |
Organism: Norwalk virus (strain gi/human/united states/norwalk/1968)
Method: X-RAY DIFFRACTION
Release Date: 2015-03-25
Ligands: M40, PG4
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1.45A Resolution Structure Of Norovirus 3Cl Protease Complex With A Covalently Bound Dipeptidyl Inhibitor (1R,2S)-2-({N-[(Benzyloxy)Carbonyl]-3-Cyclohexyl-L-Alanyl}Amino)-1-Hydroxy-3-[(3S)-2-Oxopyrrolidin-3-Yl]Propane-1-Sulfonic Acid (Orthorhombic P Form)
Organism: Norwalk virus (strain gi/human/united states/norwalk/1968)
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2015-03-25 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: M40 |
Organism: Norwalk virus (strain gi/human/united states/norwalk/1968)
Method: X-RAY DIFFRACTION
Release Date: 2015-03-25
Ligands: M40