Search Count: 50
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Complement Factor B In Complex With 5-Bromo-3-Chloro-N-(4,5-Dihydro-1H-Imidazol-2-Yl)-7-Methyl-1H-Indol-4-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.84 Å Release Date: 2020-03-04 Classification: HYDROLASE Ligands: MVZ, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-03-04
Ligands: MVZ, SO4
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Complement Factor B In Complex With (S)-5,7-Dimethyl-4-((2-Phenylpiperidin-1-Yl)Methyl)-1H-Indole
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.29 Å Release Date: 2020-03-04 Classification: HYDROLASE Ligands: SO4, MVK, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-03-04
Ligands: SO4, MVK, ZN
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Complement Factor B In Complex With (-)-4-(1-((5,7-Dimethyl-1H-Indol-4-Yl)Methyl)Piperidin-2-Yl)Benzoic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2020-03-04 Classification: HYDROLASE Ligands: SO4, MVW, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-03-04
Ligands: SO4, MVW, ZN
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Neprilysin In Complex With The Inhibitor (R)-4-(1-Carboxy-3-(3'-Chlorobiphenyl-4-Yl)Propan-2-Ylamino)-4-Oxobutanoic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.54 Å Release Date: 2020-02-12 Classification: HYDROLASE Ligands: NAG, ZN, N9Q |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-02-12
Ligands: NAG, ZN, N9Q
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Complement Factor D In Complex With The Inhibitor (S)-2-(2-((3'-(1-Amino-2-Hydroxyethyl)-[1,1'-Biphenyl]-3-Yl)Methoxy)Phenyl)Acetic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2019-04-24 Classification: HYDROLASE Ligands: J6T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-24
Ligands: J6T
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Complement Factor D In Complex With The Inhibitor 2-(2-(3'-(Aminomethyl)-[1,1'-Biphenyl]-3-Carboxamido)Phenyl)Acetic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2019-04-24 Classification: HYDROLASE Ligands: J7B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-24
Ligands: J7B
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Complement Factor B Protease Domain In Complex With The Reversible Inhibitor 4-((2S,4S)-4-Ethoxy-1-((5-Methoxy-7-Methyl-1H-Indol-4-Yl)Methyl)Piperidin-2-Yl)Benzoic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2019-04-17 Classification: HYDROLASE Ligands: SO4, JGQ, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-17
Ligands: SO4, JGQ, ZN
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Complement Factor B Protease Domain In Complex With The Reversible Inhibitor N-(2-Bromo-4-Methylnaphthalen-1-Yl)-4,5-Dihydro-1H-Imidazol-2-Amine.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2019-03-27 Classification: HYDROLASE Ligands: SO4, JGT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-27
Ligands: SO4, JGT
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Complement Factor B Protease Domain In Complex With The Reversible Inhibitor ((2S,4S)-1-((5,7-Dimethyl-1H-Indol-4-Yl)Methyl)-4-Methoxypiperidin-2-Yl)Methanol.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2019-03-27 Classification: HYDROLASE Ligands: SO4, JGN, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-27
Ligands: SO4, JGN, ZN
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Complement Factor D Complexed With Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2018-06-06 Classification: HYDROLASE Ligands: E7H, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-06-06
Ligands: E7H, GOL
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Complement Factor D Complexed With Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2018-06-06 Classification: HYDROLASE Ligands: E7E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-06-06
Ligands: E7E
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Complement Factor D In Complex With The Inhibitor 3-((3-((3-(Aminomethyl)Phenyl)Amino)-1H-Pyrazolo[3,4-D]Pyrimidin-4-Yl)Amino)Phenol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2018-06-06 Classification: HYDROLASE Ligands: E85 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-06-06
Ligands: E85
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Complement Factor D In Complex With The Inhibitor (4-((3-(Aminomethyl)Phenyl)Amino)Quinazolin-2-Yl)-L-Valine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.37 Å Release Date: 2018-06-06 Classification: HYDROLASE Ligands: E88 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-06-06
Ligands: E88
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Complement Factor D In Complex With The Inhibitor 3-((3-((3-(Aminomethyl)Phenyl)Amino)-1H-Pyrazolo[3,4-D]Pyrimidin-4-Yl)Amino)Phenol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.38 Å Release Date: 2018-06-06 Classification: HYDROLASE Ligands: E7W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-06-06
Ligands: E7W
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Complement Factor D In Complex With The Inhibitor N-(3'-(Aminomethyl)-[1,1'-Biphenyl]-3-Yl)-3-Methylbutanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2018-06-06 Classification: HYDROLASE Ligands: E8B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-06-06
Ligands: E8B
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Complement Factor D In Complex With The Inhibitor (S)-3'-(Aminomethyl)-N-(1,2,3,4-Tetrahydronaphthalen-1-Yl)-[1,1'-Biphenyl]-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2018-06-06 Classification: HYDROLASE Ligands: E82, SIN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-06-06
Ligands: E82, SIN
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Complement Factor D In Complex With The Inhibitor (S)-Pyrrolidine-1,2-Dicarboxylic Acid 1-[(1-Methyl-1H-Indol-3-Yl)-Amide] 2-[(3-Trifluoromethoxy-Phenyl)-Amide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.17 Å Release Date: 2018-03-21 Classification: HYDROLASE Ligands: GOL, 8RT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-21
Ligands: GOL, 8RT
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Complement Factor D In Complex With The Inhibitor (S)-Pyrrolidine-1,2-Dicarboxylic Acid 1-[(1-Carbamoyl-1H-Indol-3-Yl)-Amide] 2-[(3-Trifluoromethoxy-Phenyl)-Amide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2017-06-28 Classification: HYDROLASE Ligands: SO4, 8RW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: SO4, 8RW
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Complement Factor D In Complex With The Inhibitor (1R,3S,5R)-2-Aza-Bicyclo[3.1.0]Hexane-2,3-Dicarboxylic Acid 2-[(1-Carbamoyl-1H-Indol-3-Yl)-Amide] 3-[(3-Trifluoromethoxy-Phenyl)-Amide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.25 Å Release Date: 2017-06-28 Classification: HYDROLASE Ligands: 8RZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: 8RZ
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Complement Factor D In Complex With The Inhibitor (2S,4S)-4-Amino-Pyrrolidine-1,2-Dicarboxylic Acid 1-[(1-Carbamoyl-1H-Indol-3-Yl)-Amide] 2-[(3-Trifluoromethoxy-Phenyl)-Amide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2017-06-28 Classification: HYDROLASE Ligands: 8S2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: 8S2
