Search Count: 19
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Computational Design Of Highly Signaling Active Membrane Receptors Through De Novo Solvent-Mediated Allosteric Networks
Organism: Tequatrovirus t4, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.90 Å Release Date: 2024-12-18 Classification: MEMBRANE PROTEIN Ligands: NGI |
Organism: Tequatrovirus t4, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: NGI
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Crystal Structures Of Flap Bound To Dg-031
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.37 Å Release Date: 2020-12-02 Classification: MEMBRANE PROTEIN Ligands: QY1, CA, BOG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-02
Ligands: QY1, CA, BOG
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Crystal Structures Of Flap Bound To Mk-866
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.61 Å Release Date: 2020-12-02 Classification: MEMBRANE PROTEIN Ligands: QY7, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-02
Ligands: QY7, SO4
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Crystal Structure Of Mpges-1 Bound To Dg-031
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2020-12-02 Classification: ISOMERASE, MEMBRANE PROTEIN Ligands: QY1, BOG, PG4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-02
Ligands: QY1, BOG, PG4
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Crystal Structure Of Akt1 In Complex With A Selective Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2018-05-02 Classification: TRANSFERASE/INHIBITOR Ligands: EX4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-02
Ligands: EX4
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Metabotropic Glutamate Receptor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2016-12-28 Classification: SIGNALING PROTEIN Ligands: NAG, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-12-28
Ligands: NAG, MG
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Metabotropic Glutamate Receptor In Complex With Antagonist (1~{S},2~{R},3~{S},4~{S},5~{R},6~{R})-2-Azanyl-3-[[3,4-Bis(Fluoranyl)Phenyl]Sulfanylmethyl]-4-Oxidanyl-Bicyclo[3.1.0]Hexane-2,6-Dicarboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2016-12-28 Classification: SIGNALING PROTEIN Ligands: 6YS, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-12-28
Ligands: 6YS, NAG
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Crystal Structure Of Mpges-1 Bound To An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.44 Å Release Date: 2016-04-13 Classification: Isomerase/Isomerase inhibitor Ligands: 4UJ, GSH, JZR, BOG, PGE, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-13
Ligands: 4UJ, GSH, JZR, BOG, PGE, PEG
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Discovery Of A Potent And Selective Mpges-1 Inhibitor For The Treatment Of Pain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2016-04-13 Classification: Isomerase/isomerase inhibitor Ligands: 4UK, GSH, BOG, PG4, 1KA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-13
Ligands: 4UK, GSH, BOG, PG4, 1KA
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Discovery Of A Potent And Selective Mpges-1 Inhibitor For The Treatment Of Pain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2016-04-13 Classification: Isomerase/isomerase inhibitor Ligands: 4UL, GSH, BOG, PG4, 1KA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-13
Ligands: 4UL, GSH, BOG, PG4, 1KA
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Crystal Structures Of Mpges-1 Inhibitor Complexes
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.42 Å Release Date: 2015-07-15 Classification: ISOMERASE/ISOMERASE INHIBITOR Ligands: 4DV, PG0, GSH, JZR, BOG, PG4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-15
Ligands: 4DV, PG0, GSH, JZR, BOG, PG4
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Crystal Structures Of Mpges-1 Inhibitor Complexes
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.41 Å Release Date: 2015-07-08 Classification: ISOMERASE/ISOMERASE INHIBITOR Ligands: 4U9, GSH, BOG, PG4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-08
Ligands: 4U9, GSH, BOG, PG4
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Crystal Structures Of Mpges-1 Inhibitor Complexes
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2015-06-10 Classification: ISOMERASE/ISOMERASE INHIBITOR Ligands: 4DZ, GSH, BOG, PG4, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-10
Ligands: 4DZ, GSH, BOG, PG4, PEG
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Crystal Structures Of Mpges-1 Inhibitor Complexes
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.41 Å Release Date: 2015-06-10 Classification: ISOMERASE/ISOMERASE INHIBITOR Ligands: 4U8, PEG, GSH, BOG, PG4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-10
Ligands: 4U8, PEG, GSH, BOG, PG4
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Crystal Structure Of The Glucocorticoid Receptor Ligand Binding Domain Bound To A Dibenzoxapine Sulfonamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2014-01-29 Classification: TRANSCRIPTION Ligands: LSJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-01-29
Ligands: LSJ
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Crystal Structure Of The Ezh2 Set Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2014-01-08 Classification: TRANSFERASE Ligands: SO4, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-01-08
Ligands: SO4, ZN
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Crystal Structure Of The Sirt1 Catalytic Domain Bound To Nad And An Ex527 Analog
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2013-01-23 Classification: HYDROLASE Ligands: 4I5, NAD, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-01-23
Ligands: 4I5, NAD, ZN
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Crystal Structure Of Human F508A Nbd1 Domain With Atp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2004-11-09 Classification: MEMBRANE PROTEIN, HYDROLASE Ligands: MG, ATP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-11-09
Ligands: MG, ATP
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Crystal Structure Of Human Deltaf508 Human Nbd1 Domain With Atp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2004-11-09 Classification: MEMBRANE PROTEIN, HYDROLASE Ligands: MG, ATP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-11-09
Ligands: MG, ATP
