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9Y65 image
Plasmodium Falciparum M1 Aminopeptidase (Pfa-M1) Bound To Inhibitor 3K (Mips3415)
Organism: Plasmodium falciparum
Method: X-RAY DIFFRACTION
Resolution:2.20 Å Release Date: 2026-01-28
Classification: HYDROLASE
Ligands: DMS, A1CTH, GOL, ZN, MG, SO4

9YC0 image
Plasmodium Falciparum M17 Aminopeptidase (Pfa-M17) Bound To Inhibitor 3Ab (Mips3413)
Organism: Plasmodium falciparum
Method: X-RAY DIFFRACTION
Resolution:2.37 Å Release Date: 2026-01-28
Classification: HYDROLASE
Ligands: ZN, CO3, PEG, SO4, A1CT4, 1PE, DMS, 2PE, A1CT5

9YC7 image
Plasmodium Falciparum M17 Aminopeptidase (Pfa-M17) Bound To Inhibitor 3K (Mips3415)
Organism: Plasmodium falciparum
Method: X-RAY DIFFRACTION
Resolution:2.37 Å Release Date: 2026-01-28
Classification: HYDROLASE
Ligands: ZN, CO3, PEG, DMS, SO4, GOL, A1CTH, 1PE

9O3E image
Plasmodium Falciparum 20S Proteasome Bound To Inhibitor 159
Organism: Plasmodium falciparum 3d7
Method: ELECTRON MICROSCOPY
Resolution:2.79 Å Release Date: 2025-11-12
Classification: CYTOSOLIC PROTEIN
Ligands: A1B74

9O3F image
Plasmodium Falciparum 20S Proteasome Bound To Inhibitor 296
Organism: Plasmodium falciparum 3d7
Method: ELECTRON MICROSCOPY
Resolution:2.28 Å Release Date: 2025-11-12
Classification: CYTOSOLIC PROTEIN
Ligands: A1B73

9CYB image
Sars-Cov-2 Plpro In Complex With Inhibitor Wehi-P1
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Resolution:1.98 Å Release Date: 2025-04-09
Classification: HYDROLASE/HYDROLASE INHIBITOR
Ligands: A1A0T, SIN

9CYC image
Sars-Cov-2 Plpro In Complex With Inhibitor Wehi-P2
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Resolution:2.01 Å Release Date: 2025-04-09
Classification: HYDROLASE/HYDROLASE INHIBITOR
Ligands: A1A0S, ACY, GOL

9CYD image
Sars-Cov-2 Plpro In Complex With Inhibitor Wehi-P4
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Resolution:2.80 Å Release Date: 2025-04-09
Classification: HYDROLASE/HYDROLASE INHIBITOR
Ligands: A1A0U, ZN, CL

9CYK image
Sars-Cov-2 Plpro In Complex With Inhibitor Wehi-P24
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Resolution:1.88 Å Release Date: 2025-04-09
Classification: HYDROLASE/HYDROLASE INHIBITOR
Ligands: A1A0V, ACY, GOL

9DKO image
Crystal Structure Of Plasmodium Falciparum Dihydroorotate Dehydrogenase Bound With Inhibitor Dsm1010 (6-Cyclopropyl-2,4-Dimethyl-3-(4-(Trifluoromethyl)Benzyl)-2,6-Dihydro-7H-Pyrazolo[3,4-C]Pyridin-7-One)
Organism: Plasmodium falciparum 3d7
Method: X-RAY DIFFRACTION
Resolution:3.00 Å Release Date: 2025-01-29
Classification: OXIDOREDUCTASE
Ligands: A1A5P, FMN, OG6

9DI6 image
Crystal Structure Of Plasmodium Falciparum Dihydroorotate Dehydrogenase Bound With Inhibitor Dsm679 (Ethyl 1,4-Dimethyl-5-((6-(Trifluoromethyl)Pyridin-3-Yl)Methyl)-1H-Pyrazole-3-Carboxylate)
Organism: Plasmodium falciparum 3d7
Method: X-RAY DIFFRACTION
Resolution:2.41 Å Release Date: 2025-01-01
Classification: OXIDOREDUCTASE/INHIBITOR
Ligands: A1A51, FMN, OG6, CIT, LDA

9DIK image
Crystal Structure Of Plasmodium Falciparum Dihydroorotate Dehydrogenase Bound With Inhibitor Dsm681 (N-Cyclopropyl-1,4-Dimethyl-5-((6-(Trifluoromethyl)Pyridin-3-Yl)Methyl)-1H-Pyrazole-3-Carboxamide)
Organism: Plasmodium falciparum 3d7
Method: X-RAY DIFFRACTION
Resolution:2.10 Å Release Date: 2025-01-01
Classification: OXIDOREDUCTASE/INHIBITOR
Ligands: A1A52, FMN, OG6, NA

9DIZ image
Crystal Structure Of Plasmodium Falciparum Dihydroorotate Dehydrogenase Bound With Inhibitor Dsm959 (6-Cyclopropyl-2,4-Dimethyl-3-((6-(Trifluoromethyl)Pyridin-3-Yl)Methyl)-2,6-Dihydro-7H-Pyrazolo[3,4-C]Pyridin-7-One)
Organism: Plasmodium falciparum 3d7
Method: X-RAY DIFFRACTION
Resolution:3.10 Å Release Date: 2025-01-01
Classification: OXIDOREDUCTASE/INHIBITOR
Ligands: A1A53, FMN, OG6

9DKQ image
Crystal Structure Of Plasmodium Falciparum Dihydroorotate Dehydrogenase Bound With Inhibitor Dsm1153 (4,6-Dicyclopropyl-3-(3-Fluoro-4-(Trifluoromethyl)Benzyl)-2-Methyl-2,6-Dihydro-7H-Pyrazolo[3,4-D]Pyridazin-7-One)
Organism: Plasmodium falciparum 3d7
Method: X-RAY DIFFRACTION
Resolution:3.15 Å Release Date: 2025-01-01
Classification: OXIDOREDUCTASE
Ligands: A1A5Q, FMN, OG6

9DKY image
Crystal Structure Of Plasmodium Falciparum Dihydroorotate Dehydrogenase Bound With Inhibitor Dsm1174 (3-((7-Azaspiro[3.5]Nonan-7-Yl)Methyl)-4-Cyclopropyl-6-Ethyl-2-Methyl-2,6-Dihydro-7H-Pyrazolo[3,4-C]Pyridin-7-One)
Organism: Plasmodium falciparum 3d7
Method: X-RAY DIFFRACTION
Resolution:3.30 Å Release Date: 2025-01-01
Classification: OXIDOREDUCTASE
Ligands: A1A59, FMN, OG6

9DLK image
Crystal Structure Of Plasmodium Falciparum Dihydroorotate Dehydrogenase Bound With Inhibitor Dsm1398 ((S)-3-(Amino(3-Chloro-4-(Trifluoromethyl)Phenyl)(Cyclopropyl)Methyl)-6-Cyclopropyl-2-Methyl-2,6-Dihydro-7H-Pyrazolo[3,4-D]Pyridazin-7-One)
Organism: Plasmodium falciparum 3d7
Method: X-RAY DIFFRACTION
Resolution:2.90 Å Release Date: 2025-01-01
Classification: OXIDOREDUCTASE
Ligands: A1A6D, FMN, OG6, ACY

9DLY image
Crystal Structure Of Plasmodium Falciparum Dihydroorotate Dehydrogenase Bound With Inhibitor Dsm1211 ((R)-3-(Amino(6-(Trifluoromethyl)Pyridin-3-Yl)Methyl)-4-Cyclopropyl-6-Ethyl-2-Methyl-2,6-Dihydro-7H-Pyrazolo[3,4-C]Pyridin-7-One)
Organism: Plasmodium falciparum 3d7
Method: X-RAY DIFFRACTION
Resolution:3.10 Å Release Date: 2025-01-01
Classification: OXIDOREDUCTASE
Ligands: A1A6E, FMN, OG6

8W2F image
Plasmodium Falciparum 20S Proteasome Bound To An Inhibitor
Organism: Plasmodium falciparum 3d7
Method: ELECTRON MICROSCOPY
Release Date: 2024-07-31
Classification: CYTOSOLIC PROTEIN/INHIBITOR
Ligands: A1AE6

8DD5 image
Crystal Structure Of Kat6A In Complex With Inhibitor Ctx-648 (Pf-9363)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.58 Å Release Date: 2023-07-05
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: R7L, ZN

7UT5 image
Acinetobacter Baumannii Dihydroorotate Dehydrogenase Bound With Inhibitor Dsm186
Organism: Acinetobacter baumannii
Method: X-RAY DIFFRACTION
Resolution:1.40 Å Release Date: 2022-12-28
Classification: OXIDOREDUCTASE/INHIBITOR
Ligands: OBR, FMN, ORO, GOL
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