Search Count: 27
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Structure Of Cbl-B Bound To Compound 33
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2026-07-01 Classification: LIGASE Ligands: GOL, IOD, EDO, MG, ZN, A1DCD, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-01
Ligands: GOL, IOD, EDO, MG, ZN, A1DCD, DMS
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Structure Of C-Cbl Bound To Compound 33
Organism: Schistosoma japonicum, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2026-07-01 Classification: LIGASE Ligands: A1DCD, ZN, MG |
Organism: Schistosoma japonicum, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-01
Ligands: A1DCD, ZN, MG
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Structure Of Cbl-B Bound To Compound 8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2026-07-01 Classification: LIGASE/INHIBITOR Ligands: GOL, ZN, EDO, MG, A1DCC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-01
Ligands: GOL, ZN, EDO, MG, A1DCC
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Human Ebp Complexed With Compound 1
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2024-06-19 Classification: ISOMERASE/INHIBITOR Ligands: A1AEU |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2024-06-19
Ligands: A1AEU
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Human Ebp Complexed With Compound 3A
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2024-06-19 Classification: ISOMERASE/INHIBITOR Ligands: A1AEV |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2024-06-19
Ligands: A1AEV
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Crystal Structure Of Selective Ire1A Inhibitor 29 At The Enzyme Active Site
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.43 Å Release Date: 2024-05-29 Classification: TRANSFERASE/INHIBITOR Ligands: EDO, XOE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-05-29
Ligands: EDO, XOE
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Nik Bound To Inhibitor G02792917
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2023-06-07 Classification: SIGNALING PROTEIN Ligands: SO4, DYQ |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2023-06-07
Ligands: SO4, DYQ
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Crystal Structure Of Htdo2 Bound To Inhibitor Gne1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.18 Å Release Date: 2020-05-06 Classification: OXIDOREDUCTASE/Inhibitor Ligands: HEM, QVY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-05-06
Ligands: HEM, QVY
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Crystal Structure Of Murine Nf-Kappab Inducing Kinase (Nik) Bound To Inhibitor R7
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.74 Å Release Date: 2019-08-07 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: SO4, K6Y |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2019-08-07
Ligands: SO4, K6Y
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Crystal Structure Of Murine Nf-Kappab Inducing Kinase (Nik) In Complex With Compound 1A
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2018-07-04 Classification: TRANSFERASE Ligands: SO4, ELZ |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2018-07-04
Ligands: SO4, ELZ
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Crystal Structure Of Murine Nf-Kappab Inducing Kinase (Nik) In Complex With Compound 2F
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.84 Å Release Date: 2018-07-04 Classification: TRANSFERASE Ligands: ELW |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2018-07-04
Ligands: ELW
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Map4K4 In Complex With Inhibitor Compound 12 (N3-Methyl-10-(3-Methyl-3-(5-Methyloxazol-2-Yl)But-1-Yn-1-Yl)-6,7-Dihydro-5H-5,7-Methanobenzo[C]Imidazo[1,2-A]Azepine-2,3-Dicarboxamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.33 Å Release Date: 2018-06-20 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 9X4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-06-20
Ligands: 9X4
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Bruton'S Tyrosine Kinase (Btk) With Gdc-0853
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2018-02-28 Classification: Transferase/Transferase Inhibitor Ligands: 9AJ, EDO, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-02-28
Ligands: 9AJ, EDO, SO4
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P110Delta/P85Alpha With Taselisib (Gdc-0032)
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.91 Å Release Date: 2017-01-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 799 |
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2017-01-11
Ligands: 799
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Crystal Structure Of Murine Nf-Kappab Inducing Kinase (Nik) Bound To Imidazobenzoxepin Compound 3
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2017-01-11 Classification: TRANSFERASE Ligands: SO4, 76Z |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2017-01-11
Ligands: SO4, 76Z
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Crystal Structure Of Murine Nf-Kappab Inducing Kinase (Nik) Bound To Benzoxepin Compound 2
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.32 Å Release Date: 2017-01-11 Classification: TRANSFERASE Ligands: 774, SO4 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2017-01-11
Ligands: 774, SO4
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Crystal Structure Of Murine Nf-Kappab Inducing Kinase (Nik) Bound To Aryl Pyrrole Fragment 17
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.63 Å Release Date: 2017-01-11 Classification: TRANSFERASE Ligands: SO4, 76Y |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2017-01-11
Ligands: SO4, 76Y
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Potent And Selective Inhibitors Of Pi3K-Delta: Obtaining Isoform Selectivity From The Affinity Pocket And Tryptophan Shelf
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.67 Å Release Date: 2013-04-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0SC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-17
Ligands: 0SC
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Potent And Selective Inhibitors Of Pi3K-Delta: Obtaining Isoform Selectivity From The Affinity Pocket And Tryptophan Shelf
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2013-04-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0SD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-17
Ligands: 0SD
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Potent And Selective Inhibitors Of Pi3K-Delta: Obtaining Isoform Selectivity From The Affinity Pocket And Tryptophan Shelf
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.94 Å Release Date: 2013-04-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0SE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-17
Ligands: 0SE
