Search Count: 21
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Cryoem Structure Of Prmt5 Bound To Covalent Pbm-Site Inhibitor Brd-6988
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2021-03-17 Classification: TRANSFERASE/INHIBITOR Ligands: YJG |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2021-03-17
Ligands: YJG
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Prmt5 Complex Bound To Covalent Pbm Inhibitor Brd6711
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2020-11-25 Classification: SPLICING/TRANSFERASE Ligands: QN4, CL, SFG, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-25
Ligands: QN4, CL, SFG, GOL
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Glycogen Synthase Kinase 3 Beta Complexed With Brd0209
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2018-03-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6VK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-14
Ligands: 6VK
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Glycogen Synthase Kinase 3 Beta Complexed With Brd0705
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2018-03-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6VL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-14
Ligands: 6VL
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Glycogen Synthase Kinase 3 Beta Complexed With Brd3731
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.69 Å Release Date: 2018-03-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6VM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-14
Ligands: 6VM
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Exploiting An Asp-Glu Switch In Glycogen Synthase Kinase 3 To Design Paralog Selective Inhibitors For Use In Acute Myeloid Leukemia
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2018-02-21 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 6VL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-02-21
Ligands: 6VL
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Hdac2 With Ligand Brd4884
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2016-08-31 Classification: HYDROLASE Ligands: ZN, CA, IWX, PG5, PGE, PEG, PG4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-31
Ligands: ZN, CA, IWX, PG5, PGE, PEG, PG4
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Hdac2 With Ligand Brd7232
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2016-08-31 Classification: HYDROLASE Ligands: ZN, CA, 6EZ, PEG, PG4, PG5, PGE, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-31
Ligands: ZN, CA, 6EZ, PEG, PG4, PG5, PGE, EDO
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X-Ray Crystal Structure Of Gsk3B In Complex With Chir99021
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2016-05-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 65C, MG, MES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-25
Ligands: 65C, MG, MES
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X-Ray Crystal Structure Of Gsk3B In Complex With Brd3937
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2016-05-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 65A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-25
Ligands: 65A
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Kinase Domain Mutant Of Human Itk In Complex With An Aminobenzothiazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2014-01-22 Classification: Transferase/Transferase inhibitor Ligands: G7K, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-01-22
Ligands: G7K, SO4
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Crystal Structures Of Caspase-3 In Complex With Aza-Peptide Epoxide Inhibitors.
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2007-05-22 Classification: HYDROLASE/HYDROLASE INHIBITOR |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2007-05-22
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Crystal Structures Of Caspase-3 In Complex With Aza-Peptide Epoxide Inhibitors.
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2007-05-22 Classification: HYDROLASE/HYDROLASE INHIBITOR |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2007-05-22
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Crystal Structures Of Caspase-3 In Complex With Aza-Peptide Epoxide Inhibitors.
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2007-05-22 Classification: HYDROLASE/HYDROLASE INHIBITOR |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2007-05-22
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Crystal Structures Of Caspase-3 In Complex With Aza-Peptide Epoxide Inhibitors.
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2007-05-22 Classification: HYDROLASE/HYDROLASE INHIBITOR |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2007-05-22
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Crystal Structures Of Caspase-3 In Complex With Aza-Peptide Epoxide Inhibitors.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2007-03-20 Classification: HYDROLASE/HYDROLASE INHIBITOR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-03-20
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Crystal Structures Of Caspase-3 In Complex With Aza-Peptide Michael Acceptor Inhibitors.
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2006-09-20 Classification: HYDROLASE/HYDROLASE INHIBITOR |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2006-09-20
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Crystal Structures Of Caspase-3 In Complex With Aza-Peptide Michael Acceptor Inhibitors.
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2006-09-20 Classification: HYDROLASE/HYDROLASE INHIBITOR |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2006-09-20
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Crystal Structures Of Caspase-3 In Complex With Aza-Peptide Michael Acceptor Inhibitors.
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2006-09-20 Classification: HYDROLASE/HYDROLASE INHIBITOR |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2006-09-20
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Crystal Structures Of Caspase-3 In Complex With Aza-Peptide Michael Acceptor Inhibitors.
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2006-09-20 Classification: HYDROLASE/HYDROLASE INHIBITOR |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2006-09-20