Search Count: 25
![]() |
Trim21 Pryspry Domain Bound To An Enhanced Prlx-93936 Analog
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2025-08-27 Classification: IMMUNE SYSTEM Ligands: A1BLD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-08-27
Ligands: A1BLD
![]() |
Smooth Muscle Myosin Ii In Complex With Mt-228
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.58 Å Release Date: 2025-07-09 Classification: MOTOR PROTEIN Ligands: ADP, VO4, MG, DMS, EDO, A1IGE, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-07-09
Ligands: ADP, VO4, MG, DMS, EDO, A1IGE, CL
![]() |
Biased Agonist Bound Cb1-Gi Structure
Organism: Homo sapiens, Mus musculus
Method: ELECTRON MICROSCOPY Release Date: 2025-03-05 Classification: SIGNALING PROTEIN Ligands: A1AIW |
Organism: Homo sapiens, Mus musculus
Method: ELECTRON MICROSCOPY
Release Date: 2025-03-05
Ligands: A1AIW
![]() |
Biased Agonist Bound Cb1-Gi Structure
Organism: Homo sapiens, Mus musculus
Method: ELECTRON MICROSCOPY Release Date: 2025-03-05 Classification: SIGNALING PROTEIN Ligands: KCA |
Organism: Homo sapiens, Mus musculus
Method: ELECTRON MICROSCOPY
Release Date: 2025-03-05
Ligands: KCA
![]() |
C6-Guano Bound Mu Opioid Receptor-Gi Protein Complex
Organism: Homo sapiens, Mus musculus
Method: ELECTRON MICROSCOPY Release Date: 2022-12-07 Classification: MEMBRANE PROTEIN Ligands: KZR |
Organism: Homo sapiens, Mus musculus
Method: ELECTRON MICROSCOPY
Release Date: 2022-12-07
Ligands: KZR
![]() |
C5Guano-Uor-Gi-Scfv16
Organism: Homo sapiens, Mus musculus
Method: ELECTRON MICROSCOPY Release Date: 2022-05-04 Classification: MEMBRANE PROTEIN Ligands: L0X |
Organism: Homo sapiens, Mus musculus
Method: ELECTRON MICROSCOPY
Release Date: 2022-05-04
Ligands: L0X
![]() |
Her2 In Complex With Jbj-08-178-01
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.27 Å Release Date: 2021-09-08 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: VOY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-08
Ligands: VOY
![]() |
Egfr Kinase (T790M/V948R) In Complex With Allosteric Inhibitor Jbj-09-063
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2021-09-08 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: MG, ANP, VNS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-08
Ligands: MG, ANP, VNS
![]() |
Crystal Structure Of H38C2 K99R Mutation
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2019-07-10 Classification: IMMUNE SYSTEM Ligands: FLC, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-10
Ligands: FLC, SO4
![]() |
Egfr With An Allosteric Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2019-06-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: MG, ANP, JBJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-05
Ligands: MG, ANP, JBJ
![]() |
Crystal Structure Analysis Of Cruzain Bound To The No-Covalent Analog Of Wrr-483 (Wrr-669)
Organism: Trypanosoma cruzi
Method: X-RAY DIFFRACTION Resolution:2.51 Å Release Date: 2015-03-11 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 2VC, EDO |
Organism: Trypanosoma cruzi
Method: X-RAY DIFFRACTION
Release Date: 2015-03-11
Ligands: 2VC, EDO
![]() |
Binding Mode, Selectivity And Potency Of N-Indolyl-Oxopyridinyl-4- Amino-Propanyl-Based Inhibitors Targeting Trypanosoma Cruzi Cyp51
Organism: Trypanosoma cruzi
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2014-11-26 Classification: OXIDOREDUCTASE Ligands: HEM, J5Y, SO4 |
Organism: Trypanosoma cruzi
Method: X-RAY DIFFRACTION
Release Date: 2014-11-26
Ligands: HEM, J5Y, SO4
![]() |
Crystal Structure Analysis Of Cruzain Bound To Vinyl Sulfone Analog Of Wrr-483 (Wrr-666)
Organism: Trypanosoma cruzi
Method: X-RAY DIFFRACTION Resolution:1.27 Å Release Date: 2014-11-12 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 2V5 |
Organism: Trypanosoma cruzi
Method: X-RAY DIFFRACTION
Release Date: 2014-11-12
Ligands: 2V5
![]() |
Crystal Structure Of Trypanosoma Cruzi Cyp51 Bound To The Inhibitor (R)-N-(3-(1H-Indol-3-Yl)-1-Oxo-1-(Pyridin-4-Ylamino)Propan-2-Yl)-2-Fluoro-4-(4-(4-(Trifluoromethyl)Phenyl)Piperazin-1-Yl)Benzamide
Organism: Trypanosoma cruzi
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2014-09-03 Classification: OXIDOREDUCTASE Ligands: HEM, 26N, EDO, CL |
Organism: Trypanosoma cruzi
Method: X-RAY DIFFRACTION
Release Date: 2014-09-03
Ligands: HEM, 26N, EDO, CL
![]() |
Crystal Structure Of Trypanosoma Cruzi Cyp51 Bound To The Inhibitor (R)-N-(3-(1H-Indol-3-Yl)-1-Oxo-1-(Pyridin-4-Ylamino)Propan-2-Yl)-4-(4-(4-Chlorophenyl)Piperazin-1-Yl)-2-Fluorobenzamide.
Organism: Trypanosoma cruzi
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2014-09-03 Classification: OXIDOREDUCTASE Ligands: HEM, TW5, EDO, CL |
Organism: Trypanosoma cruzi
Method: X-RAY DIFFRACTION
Release Date: 2014-09-03
Ligands: HEM, TW5, EDO, CL
![]() |
Crystal Structure Of Trypanosoma Cruzi Cyp51 Bound To The Inhibitor (R)-N-(3-(1H-Indol-3-Yl)-1-Oxo-1-(Pyridin-4-Ylamino)Propan-2-Yl)-4-(4-(2,4-Difluorophenyl)Piperazin-1-Yl)-2-Fluorobenzamide.
Organism: Trypanosoma cruzi
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2014-08-20 Classification: OXIDOREDUCTASE Ligands: HEM, WVH, SO4, GOL |
Organism: Trypanosoma cruzi
Method: X-RAY DIFFRACTION
Release Date: 2014-08-20
Ligands: HEM, WVH, SO4, GOL
![]() |
Crystal Structure Of Trypanosoma Cruzi Cyp51 Bound To The Inhibitor (R)-N-(3-(1H-Indol-3-Yl)-1-Oxo-1-(Pyridin-4-Ylamino)Propan-2-Yl)-4-(4-(3,4-Difluorophenyl)Piperazin-1-Yl)-2-Fluorobenzamide.
Organism: Trypanosoma cruzi
Method: X-RAY DIFFRACTION Resolution:2.43 Å Release Date: 2014-08-20 Classification: OXIDOREDUCTASE Ligands: HEM, SO4, 25S |
Organism: Trypanosoma cruzi
Method: X-RAY DIFFRACTION
Release Date: 2014-08-20
Ligands: HEM, SO4, 25S
![]() |
Crystal Structure Of Trypanosoma Cruzi Cyp51 Bound To The Inhibitor (R)-N-(3-(1H-Indol-3-Yl)-1-Oxo-1-(Pyridin-4-Ylamino)Propan-2-Yl)-2',3, 5'-Trifluoro-(1,1'-Biphenyl)-4-Carboxamide
Organism: Trypanosoma cruzi
Method: X-RAY DIFFRACTION Resolution:2.84 Å Release Date: 2014-06-11 Classification: OXIDOREDUCTASE Ligands: HEM, TU1 |
Organism: Trypanosoma cruzi
Method: X-RAY DIFFRACTION
Release Date: 2014-06-11
Ligands: HEM, TU1
![]() |
Crystal Structure Of Trypanosoma Cruzi Cyp51 Bound To The Inhibitor (R)-N-(3-(1H-Indol-3-Yl)-1-Oxo-1-(Pyridin-4-Ylamino)Propan-2-Yl)-3,3'- Difluoro-(1,1'-Biphenyl)-4-Carboxamide
Organism: Trypanosoma cruzi
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2014-01-22 Classification: OXIDOREDUCTASE Ligands: HEM, 5PS |
Organism: Trypanosoma cruzi
Method: X-RAY DIFFRACTION
Release Date: 2014-01-22
Ligands: HEM, 5PS
![]() |
Cyp51 Of Trypanosoma Brucei Bound To (S)-N-(3-(1H-Indol-3-Yl)-1-Oxo-1- (Pyridin-4-Ylamino)Propan-2-Yl)-3,3'-Difluoro-(1,1'-Biphenyl)-4- Carboxamide
Organism: Trypanosoma brucei
Method: X-RAY DIFFRACTION Resolution:2.67 Å Release Date: 2013-09-04 Classification: OXIDOREDUCTASE Ligands: HEM, 18I |
Organism: Trypanosoma brucei
Method: X-RAY DIFFRACTION
Release Date: 2013-09-04
Ligands: HEM, 18I
