Search Count: 42
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Structure Of Chk1 10-Pt. Mutant Complex With Macrocyclic Lrrk2 Inhibitor Compound 1 ((11R)-8-Chloro-3,11-Dimethyl-2-(Oxan-4-Yl)-2,4,10,11,12,13-Hexahydro-9,5-(Azeno)Pyrazolo[3,4-B][1,4,6,10]Oxatriazacyclotridecine)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2026-04-08 Classification: TRANSFERASE/INHIBITOR Ligands: A1C5F |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-04-08
Ligands: A1C5F
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Structure Of Chk1 10-Pt. Mutant Complex With Macrocyclic Lrrk2 Inhibitor Compound 7 ((10As,13As)-3-Cyclobutyl-1-Methyl-8-(Trifluoromethyl)-3,4,10A,11,13A,14-Hexahydro-10H,13H-9,5-(Azeno)Furo[3,4-K]Pyrazolo[4,3-B][1,4,6,10]Oxatriazacyclotridecine)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2026-04-08 Classification: TRANSFERASE/INHIBITOR Ligands: A1C5G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-04-08
Ligands: A1C5G
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Structure Of Chk1 10-Pt. Mutant Complex With Macrocyclic Lrrk2 Inhibitor Compound 12 ((10As,13As)-3-Cyclopropyl-1-Methyl-8-(Trifluoromethyl)-3,4,10A,11,13A,14-Hexahydro-10H,13H-9,5-(Azeno)Furo[3,4-K]Pyrazolo[4,3-B][1,4,6,10]Oxatriazacyclotridecine)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.74 Å Release Date: 2026-04-08 Classification: TRANSFERASE/INHIBITOR Ligands: A1C5H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-04-08
Ligands: A1C5H
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Mpp8 Chromodomain In Complex With Nanobody 3A02
Organism: Lama glama, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.01 Å Release Date: 2025-11-05 Classification: GENE REGULATION |
Organism: Lama glama, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-11-05
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Structure Of The C-Terminal Domain Of Ckap5/Chtog
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Organism: Homo sapiens
Method: SOLUTION NMR
Release Date: 2025-03-19
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Fascin-1 In Complex With Nb 3E11
Organism: Homo sapiens, Lama glama
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2023-09-27 Classification: STRUCTURAL PROTEIN Ligands: EDO, PEG |
Organism: Homo sapiens, Lama glama
Method: X-RAY DIFFRACTION
Release Date: 2023-09-27
Ligands: EDO, PEG
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Aurora-A Kinase Domain In Complex With Coenzyme A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2019-10-02 Classification: TRANSFERASE Ligands: COA, MG, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-10-02
Ligands: COA, MG, PEG
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Aurora-A In Complex With Tacc3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2018-03-14 Classification: TRANSFERASE Ligands: ADP, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-14
Ligands: ADP, GOL, SO4
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Crystal Structure Of Aurora-A Kinase In Complex With An Allosterically Binding Fragment
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2017-11-01 Classification: TRANSFERASE Ligands: ADP, MG, CL, A4W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-01
Ligands: ADP, MG, CL, A4W
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Crystal Structure Of Aurora-A Kinase In Complex With An Allosterically Binding Fragment
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.19 Å Release Date: 2017-11-01 Classification: TRANSFERASE Ligands: ADP, MG, A5E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-01
Ligands: ADP, MG, A5E
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Crystal Structure Of Aurora-A Kinase In Complex With An Allosterically Binding Fragment
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.12 Å Release Date: 2017-11-01 Classification: TRANSFERASE Ligands: ADP, MG, A5H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-01
Ligands: ADP, MG, A5H
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Crystal Structure Of Aurora-A Kinase In Complex With An Allosterically Binding Fragment
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.19 Å Release Date: 2017-11-01 Classification: TRANSFERASE Ligands: ADP, MG, A5K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-01
Ligands: ADP, MG, A5K
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Crystal Structure Of Aurora-A Kinase In Complex With An Allosterically Binding Fragment
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2017-11-01 Classification: TRANSFERASE Ligands: ADP, MG, A5Q, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-01
Ligands: ADP, MG, A5Q, CL
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Crystal Structure Of Aurora-A Kinase In Complex With An Allosterically Binding Fragment
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2017-11-01 Classification: TRANSFERASE Ligands: ADP, MG, A5W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-01
Ligands: ADP, MG, A5W
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Crystal Structure Of Aurora-A Kinase In Complex With An Allosterically Binding Fragment
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.56 Å Release Date: 2017-11-01 Classification: TRANSFERASE Ligands: ADP, MG, CL, A5Z |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-01
Ligands: ADP, MG, CL, A5Z
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Crystal Structure Of Aurora-A Kinase In Complex With An Allosterically Binding Fragment
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2017-11-01 Classification: TRANSFERASE Ligands: ADP, MG, CL, A65 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-01
Ligands: ADP, MG, CL, A65
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Crystal Structure Of Aurora-A Kinase In Complex With An Allosterically Binding Fragment
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2017-11-01 Classification: TRANSFERASE Ligands: ADP, MG, A6E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-01
Ligands: ADP, MG, A6E
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Crystal Structure Of Aurora-A Kinase In Complex With An Allosterically Binding Fragment
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2017-11-01 Classification: TRANSFERASE Ligands: ADP, MG, A6H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-01
Ligands: ADP, MG, A6H
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Crystal Structure Of Aurora-A Kinase In Complex With An Allosterically Binding Fragment
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2017-11-01 Classification: TRANSFERASE Ligands: ADP, MG, CL, AY4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-01
Ligands: ADP, MG, CL, AY4
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Crystal Structure Of Aurora-A Kinase In Complex With An Allosterically Binding Fragment
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2017-11-01 Classification: TRANSFERASE Ligands: ADP, MG, CL, A6W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-01
Ligands: ADP, MG, CL, A6W
