Search Count: 37
 |
Crystal Structure Of Compound 19 Bound To Irak4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.74 Å Release Date: 2019-11-20 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: QL7, SO4 Modified Residue(s): TPO, SEP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-20
Ligands: QL7, SO4
 |
Crystal Structure Of Irak4 In Complex With Compound 23
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2019-05-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: LS7, SO4, GOL Modified Residue(s): TPO, SEP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-22
Ligands: LS7, SO4, GOL
 |
Structure Of The Irak4 Kinase Domain With Compound 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2019-05-22 Classification: IMMUNE SYSTEM Ligands: CA, LRS Modified Residue(s): TPO, SEP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-22
Ligands: CA, LRS
 |
Structure Of The Irak4 Kinase Domain With Compound 41
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2019-05-22 Classification: IMMUNE SYSTEM Ligands: SO4, LSV Modified Residue(s): TPO, SEP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-22
Ligands: SO4, LSV
 |
Structure Of The Irak4 Kinase Domain With Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.51 Å Release Date: 2019-05-22 Classification: IMMUNE SYSTEM Ligands: LTY Modified Residue(s): TPO, SEP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-22
Ligands: LTY
 |
Egfr Kinase Domain Mutant "Tmlr" With Azabenzimidazole Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2016-09-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 60B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-07
Ligands: SO4, 60B
 |
Egfr Kinase Domain Mutant "Tmlr" With 3-Carboxamide Azaindole Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.46 Å Release Date: 2016-09-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 60D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-07
Ligands: SO4, 60D
 |
Egfr Kinase Domain Mutant "Tmlr" With 3-Azetidinyl Azaindazole Compound 21
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.62 Å Release Date: 2016-09-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 60E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-07
Ligands: SO4, 60E
 |
Egfr Kinase Domain Mutant "Tmlr" With Pyridone Compound 2: 4-[2-(4-Chlorophenyl)Ethylamino]-~{N}-[4-(4-Methylpiperazin-1-Yl)Phenyl]-2-Oxidanylidene-1~{H}-Pyridine-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2015-12-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 5Q2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-30
Ligands: 5Q2
 |
Egfr Kinase Domain Mutant "Tmlr" With Pyridone Compound 19: 4-[(2-Azanylpyrimidin-4-Yl)Amino]-~{N}-[4-(4-Methylpiperazin-1-Yl)Phenyl]-2-Oxidanylidene-1~{H}-Pyridine-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.78 Å Release Date: 2015-12-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 5Q3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-30
Ligands: SO4, 5Q3
 |
Egfr Kinase Domain Mutant "Tmlr" With Pyridone Compound 13: 4-[(2-Methoxyphenyl)Amino]-~{N}-[4-(4-Methylpiperazin-1-Yl)Phenyl]-2-Oxidanylidene-1~{H}-Pyridine-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.81 Å Release Date: 2015-12-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 5Q4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-30
Ligands: SO4, 5Q4
 |
Egfr Kinase Domain With Pyridone Compound 13: 4-[(2-Methoxyphenyl)Amino]-~{N}-[4-(4-Methylpiperazin-1-Yl)Phenyl]-2-Oxidanylidene-1~{H}-Pyridine-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2015-12-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 5Q4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-30
Ligands: 5Q4
 |
Egfr Kinase (T790M/L858R) Apo
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2015-12-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-02
 |
Egfr Kinase (T790M/L858R) With Inhibitor Compound 15: ~{N}-(7-Chloranyl-1~{H}-Indazol-3-Yl)-7,7-Dimethyl-2-(1~{H}-Pyrazol-4-Yl)-5~{H}-Furo[3,4-D]Pyrimidin-4-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2015-12-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 5N3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-02
Ligands: 5N3
 |
Egfr Kinase (T790M/L858R) With Inhibitor Compound 27: ~{N}-(1~{H}-Indazol-3-Yl)-7,7-Dimethyl-2-(2-Methylpyrazol-3-Yl)-5~{H}-Furo[3,4-D]Pyrimidin-4-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2015-12-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 5N4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-02
Ligands: 5N4
 |
Egfr Kinase Domain Mutant "Tmlr" With Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2015-10-28 Classification: Transferase/transferase inhibitor Ligands: 4YV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: 4YV
 |
Egfr Kinase Domain Mutant "Tmlr" With Compound 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2015-10-28 Classification: Transferase/transferase inhibitor Ligands: 4YW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: 4YW
 |
Egfr Kinase Domain Mutant "Tmlr" With Compound 23
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2015-10-28 Classification: Transferase/transferase inhibitor Ligands: SO4, 4YX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: SO4, 4YX
 |
Egfr Kinase Domain Mutant "Tmlr" With Compound 24
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2015-10-28 Classification: Transferase/transferase inhibitor Ligands: 4Z8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: 4Z8
 |
Egfr Kinase Domain Mutant "Tmlr" With Compound 27
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2015-10-28 Classification: Transferase/transferase inhibitor Ligands: SO4, 4ZB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: SO4, 4ZB