Search Count: 144
![]() |
Mycobacterium Tuberculosis Pks13 Acyltransferase Serine Converted To Beta-Lactam Form By Cec215 Via Sufex Reaction
Organism: Mycobacterium tuberculosis h37rv
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2025-05-21 Classification: ANTIBIOTIC Ligands: SO4, CL, PG4, EDO, DMS, GOL, PEG |
Organism: Mycobacterium tuberculosis h37rv
Method: X-RAY DIFFRACTION
Release Date: 2025-05-21
Ligands: SO4, CL, PG4, EDO, DMS, GOL, PEG
![]() |
Mycobaterium Tuberculosis Pks13 Acyltransferase Incubated With Dmso
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv)
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2025-05-21 Classification: ANTIBIOTIC Ligands: DMS, SO4, PE5, EDO, PEG, GOL, CL, NA, P33 |
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv)
Method: X-RAY DIFFRACTION
Release Date: 2025-05-21
Ligands: DMS, SO4, PE5, EDO, PEG, GOL, CL, NA, P33
![]() |
M. Tuberculosis Pks13 Acyltransferase (At) Domain In Complex With Sufex Inhibitor Cec215
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2025-05-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1PE, SO4, A1ATV |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2025-05-07
Ligands: 1PE, SO4, A1ATV
![]() |
M. Tuberculosis Pks13 Acyltransferase (At) Domain In Complex With Sufex Inhibitor Cmx410
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv)
Method: X-RAY DIFFRACTION Resolution:2.57 Å Release Date: 2025-05-07 Classification: TRANSFERASE/TRANSFERSE INHIBITOR Ligands: 1PE, SO4, A1ATW |
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv)
Method: X-RAY DIFFRACTION
Release Date: 2025-05-07
Ligands: 1PE, SO4, A1ATW
![]() |
M. Tuberculosis Pks13 Acyltransferase (At) Domain Sulfate Free Apo Form
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2025-05-07 Classification: TRANSFERASE Ligands: 1PE, SO4 |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2025-05-07
Ligands: 1PE, SO4
![]() |
M. Tuberculosis Pks13 Acyltransferase (At) Domain In Complex With Sufex Inhibitor Cmx410 - Reaction Product
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv)
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2025-05-07 Classification: TRANSFERASE Ligands: SO4, 1PE, A1AVL |
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv)
Method: X-RAY DIFFRACTION
Release Date: 2025-05-07
Ligands: SO4, 1PE, A1AVL
![]() |
Crystal Structure Of Mycobacterium Tuberculosis Cytochrome P450 Cyp125 In Complex With An Inhibitor
Organism: Mycobacterium tuberculosis h37rv
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2025-01-29 Classification: OXIDOREDUCTASE Ligands: HEM, SO4, A1H47 |
Organism: Mycobacterium tuberculosis h37rv
Method: X-RAY DIFFRACTION
Release Date: 2025-01-29
Ligands: HEM, SO4, A1H47
![]() |
X-Ray Crystal Structure Of Cyp142 From Mycobacterium Tuberculosis In Complex With A Fragment Bound In Two Poses
Organism: Mycobacterium tuberculosis h37rv
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2025-01-29 Classification: OXIDOREDUCTASE Ligands: 3QO, HEM |
Organism: Mycobacterium tuberculosis h37rv
Method: X-RAY DIFFRACTION
Release Date: 2025-01-29
Ligands: 3QO, HEM
![]() |
Crystal Structure Of Mycobacterium Smegmatis Coab In Complex With Ctp And 5-Methoxy-1H-Indole-2-Carboxylic Acid
Organism: Mycolicibacterium smegmatis mc2 155
Method: X-RAY DIFFRACTION Resolution:2.84 Å Release Date: 2024-05-08 Classification: LIGASE Ligands: CTP, CA, VEO |
Organism: Mycolicibacterium smegmatis mc2 155
Method: X-RAY DIFFRACTION
Release Date: 2024-05-08
Ligands: CTP, CA, VEO
![]() |
Crystal Structure Of Mycobacterium Smegmatis Coab In Complex With Ctp And 2-(5-Bromo-1-(4-Hydroxyphenyl)-1H-Indol-3-Yl)-2-Oxoacetic Acid
Organism: Mycolicibacterium smegmatis mc2 155
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2024-05-08 Classification: LIGASE Ligands: CTP, CA, VE6 |
Organism: Mycolicibacterium smegmatis mc2 155
Method: X-RAY DIFFRACTION
Release Date: 2024-05-08
Ligands: CTP, CA, VE6
![]() |
Crystal Structure Of Mycobacterium Smegmatis Coab In Complex With Ctp And 2-(1-(4-Hydroxyphenyl)-5-Phenyl-1H-Indol-3-Yl)-2-Oxoacetic Acid
Organism: Mycolicibacterium smegmatis mc2 155
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2024-05-08 Classification: LIGASE Ligands: CTP, CA, W52, ACT |
Organism: Mycolicibacterium smegmatis mc2 155
Method: X-RAY DIFFRACTION
Release Date: 2024-05-08
Ligands: CTP, CA, W52, ACT
![]() |
Crystal Structure Of Mycobacterium Smegmatis Coab In Complex With Ctp And 2-(1-(3,4-Dihydroxyphenyl)-5-Phenyl-1H-Indol-3-Yl)-2-Oxoacetic Acid
Organism: Mycolicibacterium smegmatis mc2 155
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2024-05-08 Classification: LIGASE Ligands: CTP, CA, W4X |
Organism: Mycolicibacterium smegmatis mc2 155
Method: X-RAY DIFFRACTION
Release Date: 2024-05-08
Ligands: CTP, CA, W4X
![]() |
Crystal Structure Of Mycobacterium Smegmatis Coab In Complex With Ctp And 2-(1-(3,4-Dihydroxyphenyl)-5-(3-Hydroxyphenyl)-1H-Indol-3-Yl)-2-Oxoacetic Acid
Organism: Mycolicibacterium smegmatis mc2 155
Method: X-RAY DIFFRACTION Resolution:2.44 Å Release Date: 2024-05-08 Classification: LIGASE Ligands: CTP, CA, W5E, ACT |
Organism: Mycolicibacterium smegmatis mc2 155
Method: X-RAY DIFFRACTION
Release Date: 2024-05-08
Ligands: CTP, CA, W5E, ACT
![]() |
Identification And Optimisation Of Novel Inhibitors Of The Polyketide Synthetase 13 Thioesterase Domain With Antitubercular Activity
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2023-11-22 Classification: TRANSFERASE Ligands: IJJ |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2023-11-22
Ligands: IJJ
![]() |
Identification And Optimisation Of Novel Inhibitors Of The Polyketide Synthetase 13 Thioesterase Domain With Antitubercular Activity
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2023-11-22 Classification: TRANSFERASE Ligands: SO4, IKG |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2023-11-22
Ligands: SO4, IKG
![]() |
Identification And Optimisation Of Novel Inhibitors Of The Polyketide Synthetase 13 Thioesterase Domain With Antitubercular Activity
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:1.71 Å Release Date: 2023-11-22 Classification: TRANSFERASE Ligands: SO4, IL8, GOL, 2Q5 |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2023-11-22
Ligands: SO4, IL8, GOL, 2Q5
![]() |
Crystal Structure Of Cyp125 From Mycobacterium Tuberculosis In Complex With An Inhibitor
Organism: Mycobacterium tuberculosis h37rv
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2023-04-19 Classification: OXIDOREDUCTASE Ligands: EIQ, HEM, CL, DMS |
Organism: Mycobacterium tuberculosis h37rv
Method: X-RAY DIFFRACTION
Release Date: 2023-04-19
Ligands: EIQ, HEM, CL, DMS
![]() |
Crystal Structure Of Cyp125 From Mycobacterium Tuberculosis In Complex With An Inhibitor
Organism: Mycobacterium tuberculosis h37rv
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2023-04-19 Classification: OXIDOREDUCTASE Ligands: GOL, 5YG, HEM, SO4, CL |
Organism: Mycobacterium tuberculosis h37rv
Method: X-RAY DIFFRACTION
Release Date: 2023-04-19
Ligands: GOL, 5YG, HEM, SO4, CL
![]() |
Crystal Structure Of Cyp125 From Mycobacterium Tuberculosis In Complex With An Inhibitor
Organism: Mycobacterium tuberculosis h37rv
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2023-04-05 Classification: OXIDOREDUCTASE Ligands: JFC, HEM, SO4 |
Organism: Mycobacterium tuberculosis h37rv
Method: X-RAY DIFFRACTION
Release Date: 2023-04-05
Ligands: JFC, HEM, SO4
![]() |
Crystal Structure Of Cyp125 From Mycobacterium Tuberculosis In Complex With An Inhibitor
Organism: Mycobacterium tuberculosis h37rv
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2023-04-05 Classification: OXIDOREDUCTASE Ligands: GOL, HEM, JK9, SO4, CL |
Organism: Mycobacterium tuberculosis h37rv
Method: X-RAY DIFFRACTION
Release Date: 2023-04-05
Ligands: GOL, HEM, JK9, SO4, CL
