Search Count: 75
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Focal Adhesion Kinase Catalytic Domain In Complex With 6-(1H-Pyrazol-4-Yl)-Nicotinic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.53 Å Release Date: 2025-12-31 Classification: TRANSFERASE Ligands: SO4, A1JNJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-12-31
Ligands: SO4, A1JNJ
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Crystal Structure Of Human Exonuclease 1 (Exo1) With Dna And Compound 20
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2025-12-17 Classification: HYDROLASE Ligands: MG, NA, A1JNC, FMT |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2025-12-17
Ligands: MG, NA, A1JNC, FMT
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Crystal Structure Of Human Exonuclease 1 (Exo1) With Dna And Compound Art5537
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2025-12-17 Classification: HYDROLASE Ligands: MG, A1JO0, NA |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2025-12-17
Ligands: MG, A1JO0, NA
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Crystal Structure Of Flap Endonuclease Fen1 With Compound 28
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2025-09-24 Classification: HYDROLASE Ligands: MG, EDO, A1JD4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-24
Ligands: MG, EDO, A1JD4
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Crystal Structure Of Flap Endonuclease Fen1 With Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2025-09-24 Classification: HYDROLASE Ligands: A1JED, TEW, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-24
Ligands: A1JED, TEW, MG
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Tead1 In Complex With A Reversible Inhibitor N-[(1S)-2-Hydroxy-1-(1-Methyl-1H-Pyrazol-3-Yl)Ethyl]-2-Methyl-8-[4-(Trifluoromethyl)Phenyl]-2H,8H-Pyrazolo[3,4-B]Indole-5-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2025-01-22 Classification: TRANSCRIPTION Ligands: GOL, A1IJL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-22
Ligands: GOL, A1IJL, SO4
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C-Met Y1234E,Y1235E Mutant In Complex With Tepotinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2023-09-06 Classification: TRANSFERASE Ligands: 3E8, PG4, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-09-06
Ligands: 3E8, PG4, PEG
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C-Met F1200I Mutant In Complex With Tepotinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.72 Å Release Date: 2023-09-06 Classification: TRANSFERASE Ligands: 3E8, EDO, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-09-06
Ligands: 3E8, EDO, CL
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C-Met Y1235D Mutant In Complex With Tepotinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2023-09-06 Classification: TRANSFERASE Ligands: 3E8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-09-06
Ligands: 3E8
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Focal Adhesion Kinase Catalytic Domain In Complex With 6-[4-(3-Methanesulfonyl-Benzylamino)-5-Trifluoromethyl-Pyrimidin-2-Ylamino]-3,4-Dihydro-1H-Quinolin-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.36 Å Release Date: 2021-02-10 Classification: TRANSFERASE Ligands: P4N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-02-10
Ligands: P4N
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Focal Adhesion Kinase Catalytic Domain In Complex With N-Methyl-N-(3-{[2-(2-Oxo-1,2,3,4-Tetrahydro-Quinolin-6-Ylamino)-5-Trifluoromethyl-Pyrimidin-4-Ylamino]-Methyl}-Pyridin-2-Yl)-Methanesulfonamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2021-02-10 Classification: TRANSFERASE Ligands: P7N, NA, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-02-10
Ligands: P7N, NA, SO4
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Focal Adhesion Kinase Catalytic Domain In Complex With N-Methyl-N-(2-{[2-(2-Oxo-2,3-Dihydro-1H-Indol-5-Ylamino)-5-Trifluoromethyl-Pyrimidin-4-Ylamino]-Methyl}-Phenyl)-Methanesulfonamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2021-02-10 Classification: TRANSFERASE Ligands: P9K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-02-10
Ligands: P9K
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Focal Adhesion Kinase Catalytic Domain In Complex With N-Methyl-N-(3-{[2-(2-Oxo-2,3-Dihydro-1H-Indol-5-Ylamino)-Pyrimidin-4-Ylamino]-Methyl}-Pyridin-2-Yl)-Methanesulfonamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.54 Å Release Date: 2021-02-10 Classification: TRANSFERASE Ligands: PKE, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-02-10
Ligands: PKE, SO4
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Focal Adhesion Kinase Catalytic Domain In Complex With 5-{4-[(Pyridin-3-Ylmethyl)-Amino]-5-Trifluoromethyl-Pyrimidin-2-Ylamino}-1,3-Dihydro-Indol-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.81 Å Release Date: 2021-02-10 Classification: TRANSFERASE Ligands: PVT, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-02-10
Ligands: PVT, SO4
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Focal Adhesion Kinase Catalytic Domain In Complex With 4-{[4-{[(1R,2R)-2-(Dimethylamino)Cyclopentyl]Amino}-5-(Trifluoromethyl)Pyrimidin-2-Yl]Amino}-N-Methylbenzenesulfonamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2021-02-10 Classification: TRANSFERASE Ligands: P1E, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-02-10
Ligands: P1E, SO4
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Focal Adhesion Kinase Catalytic Domain In Complex With N-Methyl-N-{3-[(2-Phenylamino-5-Trifluoromethyl-Pyrimidin-4-Ylamino)-Methyl]-Pyridin-2-Yl}-Methanesulfonamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2021-02-10 Classification: TRANSFERASE Ligands: Q2H, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-02-10
Ligands: Q2H, SO4
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Crystal Structure Of Human Methionine Aminopeptidase-2 In Complex; With An Inhibitor (S)-3-Hydroxy-2-Oxo-1-(2-Oxo-1,2,3,4-Tetrahydro-Quinolin-6-Yl)-Pyrrolidine-3-Carboxylic Acid 3-Chloro-5-Fluoro-Benzylamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2019-05-01 Classification: HYDROLASE Ligands: EDO, DMS, GOL, HZK, MN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-01
Ligands: EDO, DMS, GOL, HZK, MN
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Crystal Structure Of Human Methionine Aminopeptidase-2 In Complex With An Inhibitor (S)-3-Hydroxy-2-Oxo-1-Phenyl-Pyrrolidine-3-Carboxylic Acid 3-Chloro-5-Fluoro-Benzylamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2019-05-01 Classification: HYDROLASE Ligands: EDO, GOL, HZW, MN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-01
Ligands: EDO, GOL, HZW, MN
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Crystal Structure Of Human Methionine Aminopeptidase-2 In Complex With An Inhibitor 2-Oxo-1-Phenyl-Pyrrolidine-3-Carboxylic Acid (2-Thiophen-2-Yl-Ethyl)-Amide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.08 Å Release Date: 2019-05-01 Classification: HYDROLASE Ligands: GOL, K4K, MN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-01
Ligands: GOL, K4K, MN
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Crystal Structure Of Human Methionine Aminopeptidase-2 In Complex With An Inhibitor 5-Chloro-Quinolin-8-Ol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2019-05-01 Classification: HYDROLASE Ligands: GOL, HZQ, MN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-01
Ligands: GOL, HZQ, MN
