Search Count: 30
![]() |
Cdk2/Cycline Bound To Compound 11 With P-Loop In The Ee And Cc Conformations
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.12 Å Release Date: 2025-04-30 Classification: CELL CYCLE Ligands: A1CAE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-04-30
Ligands: A1CAE
![]() |
Cdk2/Cycline Bound To Compound 16 With P-Loop In The Ee Conformation
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2025-04-30 Classification: CELL CYCLE Ligands: A1CAH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-04-30
Ligands: A1CAH
![]() |
Cdk2/Cycline Bound To Compound 19 With P-Loop In The Ee And Ec Conformations
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2025-04-30 Classification: CELL CYCLE Ligands: A1CAF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-04-30
Ligands: A1CAF
![]() |
Cdk2/Cycline Bound To Compound 20 With P-Loop In The Ee And Cc Conformations
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2025-04-30 Classification: CELL CYCLE Ligands: A1CAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-04-30
Ligands: A1CAG
![]() |
Cdk2/Cycline Bound To Compound 21 With P-Loop In The Ee And Cc Conformations
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2025-04-30 Classification: CELL CYCLE Ligands: A1CAI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-04-30
Ligands: A1CAI
![]() |
Fgfr2 Kinase Domain Bound To Reversible Inhibitor Cmpd 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2024-02-14 Classification: ONCOPROTEIN Ligands: GOL, GSH, WXQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-14
Ligands: GOL, GSH, WXQ
![]() |
Fgfr2 Kinase Domain Bound To Irreversible Inhibitor Cmpd 10
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.33 Å Release Date: 2024-02-14 Classification: Transferase/Inhibitor Ligands: GOL, UIM, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-14
Ligands: GOL, UIM, SO4
![]() |
Human Pi3K P85Alpha/P110Alpha
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.71 Å Release Date: 2023-11-22 Classification: SIGNALING PROTEIN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-22
![]() |
P85Alpha/P110Alpha Heterodimer H1047R Mutant
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.72 Å Release Date: 2023-11-22 Classification: SIGNALING PROTEIN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-22
![]() |
Human Pi3K P85Alpha/P110Alpha H1047R Bound To Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.83 Å Release Date: 2023-11-22 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: UE9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-22
Ligands: UE9
![]() |
Human Pi3K P85Alpha/P110Alpha H1047R Bound To Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.51 Å Release Date: 2023-11-22 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: UIW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-22
Ligands: UIW
![]() |
Human Pi3K P85Alpha/P110Alpha Bound To Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.53 Å Release Date: 2023-11-22 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: UIW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-22
Ligands: UIW
![]() |
Human Pi3K P85Alpha/P110Alpha H1047R Bound To Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.62 Å Release Date: 2023-11-22 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: UJC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-22
Ligands: UJC
![]() |
Human Pi3K P85Alpha/P110Alpha Bound To Rly-2608
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2023-11-22 Classification: SIGNALING PROTEIN,TRANSFERASE/INHIBITOR Ligands: XUZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-22
Ligands: XUZ
![]() |
Cryoem Structure Of Pi3Kalpha
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2023-11-15 Classification: CYTOSOLIC PROTEIN |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2023-11-15
![]() |
Crystal Structure Of The C-Met Kinase Domain In Complex With A Pyrazolone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2016-09-21 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 75H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-21
Ligands: 75H
![]() |
Crystal Structure Of C-Met In Complex With Naphthyridinone Inhibitor 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2016-02-10 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 5SZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-10
Ligands: 5SZ
![]() |
Crystal Structure Of C-Met In Complex With Amg 337
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2016-02-10 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 5T1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-10
Ligands: 5T1
![]() |
Crystal Structure Of C-Met In Complex With (R)-5-(8-Fluoro-3-(1-Fluoro-1-(3-Methoxyquinolin-6-Yl)Ethyl)-[1,2,4]Triazolo[4,3-A]Pyridin-6-Yl)-3-Methylisoxazole
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2015-03-11 Classification: Transferase/transferase inhibitor Ligands: 46G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-03-11
Ligands: 46G
![]() |
Crystal Structure Of C-Met In Complex With (S)-5-(8-Fluoro-3-(1-(3-(2-Methoxyethoxy)Quinolin-6-Yl)Ethyl)-[1,2,4]Triazolo[4,3-A]Pyridin-6-Yl)-3-Methylisoxazole
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2015-03-11 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: 44X |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-03-11
Ligands: 44X
