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9TFV image
Cryo-Em Structure Of The Inward Rectifying Potassium Channel 7.1 (Kir7.1)

9TG3 image
Cryo-Em Structure Of The R162W Mutant Inward Rectifying Potassium Channel 7.1 (Kir7.1)

9TG6 image
Cryo-Em Structure Of The Inward Rectifying Potassium Channel 7.1 (Kir7.1) In Complex With Pip2

7NZY image
Crystal Structure Of Human Casein Kinase I Delta In Complex With Cgs-15943
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.85 Å Release Date: 2022-10-05
Classification: TRANSFERASE
Ligands: UX2, MLI, PO4

7ZBN image
Cryo-Em Structure Of The Human Gs-Gn Complex In The Inhibited State

5AEP image
Novel Pyrrole Carboxamide Inhibitors Of Jak2 As Potential Treatment Of Myeloproliferative Disorders
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.95 Å Release Date: 2015-04-29
Classification: TRANSFERASE
Ligands: QUP

4D0W image
Pyrrole-3-Carboxamides As Potent And Selective Jak2 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.77 Å Release Date: 2014-07-23
Classification: TRANSFERASE
Ligands: GOL, VVQ

4D0X image
Pyrrole-3-Carboxamides As Potent And Selective Jak2 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.82 Å Release Date: 2014-07-23
Classification: TRANSFERASE
Ligands: 953, GOL

4D1S image
Pyrrole-3-Carboxamides As Potent And Selective Jak2 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.66 Å Release Date: 2014-07-23
Classification: TRANSFERASE
Ligands: BJG

4O3M image
Ternary Complex Of Bloom'S Syndrome Helicase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.30 Å Release Date: 2014-03-12
Classification: Hydrolase/DNA
Ligands: CA, ZN, ADP, EDO

4BKY image
Crystal Structure Of Unphosphorylated Maternal Embryonic Leucine Zipper Kinase (Melk) In Complex With Pyrrolopyrazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.83 Å Release Date: 2013-08-21
Classification: TRANSFERASE
Ligands: 82B, UNX

4BKZ image
Crystal Structure Of Unphosphorylated Maternal Embryonic Leucine Zipper Kinase (Melk) In Complex With A Benzodipyrazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.20 Å Release Date: 2013-08-21
Classification: TRANSFERASE
Ligands: 1WS

4BL1 image
Crystal Structure Of Unphosphorylated Maternal Embryonic Leucine Zipper Kinase (Melk) In Complex With Amp-Pnp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.60 Å Release Date: 2013-05-08
Classification: TRANSFERASE
Ligands: ANP

4AQ3 image
Human Bcl-2 With Phenylacylsulfonamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.40 Å Release Date: 2012-06-06
Classification: APOPTOSIS
Ligands: 398

4A4L image
Crystal Structure Of Polo-Like Kinase 1 In Complex With A 5-(2-Amino- Pyrimidin-4-Yl)-1H-Pyrrole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.35 Å Release Date: 2012-01-11
Classification: TRANSFERASE
Ligands: ZN, TLA, 939

4A4O image
Crystal Structure Of Polo-Like Kinase 1 In Complex With A 2-(2-Amino- Pyrimidin-4-Yl)-1,5,6,7-Tetrahydro-Pyrrolopyridin-4-One Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.70 Å Release Date: 2012-01-11
Classification: TRANSFERASE
Ligands: ZN, TLA, 664

3U0Z image
Tetramerization Dynamics Of The C-Terminus Underlies Isoform-Specific Camp-Gating In Hcn Channels

3U10 image
Tetramerization Dynamics Of The C-Terminus Underlies Isoform-Specific Camp-Gating In Hcn Channels

3U11 image
Tetramerization Dynamics Of The C-Terminus Underlies Isoform-Specific Camp-Gating In Hcn Channels

2XCL image
Nucleotide-Bound Structures Of Bacillus Subtilis Glycinamide Ribonucleotide Synthetase
Organism: Bacillus subtilis
Method: X-RAY DIFFRACTION
Resolution:2.10 Å Release Date: 2011-03-23
Classification: LIGASE
Ligands: ANP, MG
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