Search Count: 31
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Crystal Structure Of Selective Inhibitor 16 Bound At The Active Site Of Cdk1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2026-07-08 Classification: SIGNALING PROTEIN Ligands: A1DEQ, A1DJL, GOL, SO4, DMS, EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-08
Ligands: A1DEQ, A1DJL, GOL, SO4, DMS, EPE
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Structure Of Tead2 Bound To G8025
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2026-07-08 Classification: TRANSCRIPTION/INHIBITOR Ligands: A1CA7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-08
Ligands: A1CA7
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Structure Of Tead2 Bound To G2181
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2026-07-08 Classification: TRANSCRIPTION/INHIBITOR Ligands: A1CA6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-08
Ligands: A1CA6
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Crystal Structure Of Htead2 Bound To A Methoxypyridine Lipid Pocket Binder
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2023-08-16 Classification: TRANSCRIPTION/INHIBITOR Ligands: TRS, Y2S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-08-16
Ligands: TRS, Y2S
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Tead2 Bound To Gne-7883
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2023-05-03 Classification: TRANSCRIPTION Ligands: TRS, KUR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-05-03
Ligands: TRS, KUR
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Tead2 Bound To Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2023-05-03 Classification: TRANSCRIPTION Ligands: KUI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-05-03
Ligands: KUI
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Tead2 Bound To Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2023-05-03 Classification: TRANSCRIPTION Ligands: KTF, TRS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-05-03
Ligands: KTF, TRS
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Rock1 In Complex With Ligand G4998
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.34 Å Release Date: 2022-10-05 Classification: TRANSFERASE Ligands: CL, 86G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-10-05
Ligands: CL, 86G
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Rock1 In Complex With Ligand G5018
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.74 Å Release Date: 2022-10-05 Classification: TRANSFERASE Ligands: EPE, 86K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-10-05
Ligands: EPE, 86K
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Crystal Structure Of Tead2 Bound To Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.54 Å Release Date: 2020-06-24 Classification: Transcription/Transcription Inhibitor Ligands: GOL, QSJ, TRS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-06-24
Ligands: GOL, QSJ, TRS
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Crystal Structure Of Tead2 Bound To Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2020-06-24 Classification: TRANSCRIPTION/INHIBITOR Ligands: QLV, TRS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-06-24
Ligands: QLV, TRS
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Selective & Brain-Permeable Polo-Like Kinase-2 (Plk-2) Inhibitors That Reduce -Synuclein Phosphorylation In Rat Brain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2013-12-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: R78 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-12-25
Ligands: R78
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Selective & Brain-Permeable Polo-Like Kinase-2 (Plk-2) Inhibitors That Reduce -Synuclein Phosphorylation In Rat Brain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.74 Å Release Date: 2013-12-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1D1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-12-25
Ligands: 1D1
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Spr And Structural Analysis Yield Insight Towards Mechanism Of Inhibition Of Bace Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2013-11-20 Classification: hydrolase/hydrolase inhibitor Ligands: 957 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-11-20
Ligands: 957
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Selective & Brain-Permeable Polo-Like Kinase-2 (Plk-2) Inhibitors That Reduce -Synuclein Phosphorylation In Rat Brain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2013-11-20 Classification: transferase/transferase inhibitor Ligands: 11G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-11-20
Ligands: 11G
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Selective & Brain-Permeable Polo-Like Kinase-2 (Plk-2) Inhibitors That Reduce -Synuclein Phosphorylation In Rat Brain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2013-11-20 Classification: transferase/transferase inhibitor Ligands: 1C7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-11-20
Ligands: 1C7
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Design And Synthesis Of Thiophene Dihydroisoquinolins As Novel Bace-1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2013-10-09 Classification: hydrolase/hydrolase inhibitor Ligands: ZN, 1B7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-10-09
Ligands: ZN, 1B7
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Selective & Brain-Permeable Polo-Like Kinase-2 (Plk-2) Inhibitors That Reduce Alpha-Synuclein Phosphorylation In Rat Brain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2013-08-14 Classification: transferase/transferase inhibitor Ligands: 1C8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-08-14
Ligands: 1C8
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Structure-Based Design Of Novel Dihydroisoquinoline Bace-1 Inhibitors That Do Not Engage The Catalytic Aspartates
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2013-03-06 Classification: hydrolase/hydrolase inhibitor Ligands: ZN, 0ZA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-06
Ligands: ZN, 0ZA
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Design And Synthesis Of Thiophene Dihydroisoquinolins As Novel Bace-1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2013-03-06 Classification: hydrolase/hydrolase inhibitor Ligands: ZN, 1B8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-06
Ligands: ZN, 1B8