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9PSJ image
Crystal Structure Of Baf60A (Smarcd1) Apo Containing Partial Coiled Coil And The Yeats-Like Domain With Topologically-Linked Swib

9PSL image
Co-Crystal Structure Of Baf60A (Smarcd1) In Complex With Pu.1 Peptide

9PSQ image
Co-Crystal Structure Of Baf60A (Smarcd1) Bound To Ppsc-001

9PSR image
Co-Crystal Structure Of Baf60A (Smarcd1) Bound To Ppsc-002

7TAB image
G-925 Bound To The Smarca4 (Brg1) Bromodomain

7TD9 image
G-059 Bound To The Smarca4 (Brg1) Bromodomain

6DF7 image
Taf1-Bd2 In Complex With Cpd27 (6-(But-3-En-1-Yl)-4-(1-Methyl-6-(Morpholine-4-Carbonyl)-1H-Benzo[D]Imidazol-4-Yl)-1,6-Dihydro-7H-Pyrrolo[2,3-C]Pyridin-7-One)

6DF4 image
Taf1-Bd2 In Complex With Cpd8 (6-(But-3-En-1-Yl)-4-(3-(Morpholine-4-Carbonyl)Phenyl)-1,6-Dihydro-7H-Pyrrolo[2,3-C]Pyridin-7-One)

5V84 image
Cecr2 In Complex With Cpd6 (6-Allyl-N,2-Dimethyl-7-Oxo-N-(1-(1-Phenylethyl)Piperidin-4-Yl)-6,7-Dihydro-1H-Pyrrolo[2,3-C]Pyridine-4-Carboxamide)

5LS6 image
Structure Of Human Polycomb Repressive Complex 2 (Prc2) With Inhibitor

5KTU image
Crystal Structure Of The Bromodomain Of Human Crebbp Bound To Pyrazolopiperidine Scaffold
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.38 Å Release Date: 2016-11-02
Classification: TRANSFERASE
Ligands: 6XB, DMS

5KTW image
Crebbp Bromodomain In Complex With Cpd 44 (3-((5-Acetyl-1-(Cyclopropylmethyl)-4,5,6,7-Tetrahydro-1H-Pyrazolo[4,3-C]Pyridin-3-Yl)Amino)-N-Isopropylbenzamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.09 Å Release Date: 2016-11-02
Classification: TRANSFERASE
Ligands: 6XG, EDO

5KTX image
Crebbp Bromodomain In Complex With Cpd59 ((S)-1-(3-((2-Fluoro-4-(1-Methyl-1H-Pyrazol-4-Yl)Phenyl)Amino)-1-(Tetrahydrofuran-3-Yl)-6,7-Dihydro-1H-Pyrazolo[4,3-C]Pyridin-5(4H)-Yl)Ethanone)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.27 Å Release Date: 2016-11-02
Classification: TRANSFERASE
Ligands: 6XH, EDO, DMS

5KU3 image
Brd4 Bromodomain In Complex With Cpd59 ((S)-1-(3-((2-Fluoro-4-(1-Methyl-1H-Pyrazol-4-Yl)Phenyl)Amino)-1-(Tetrahydrofuran-3-Yl)-6,7-Dihydro-1H-Pyrazolo[4,3-C]Pyridin-5(4H)-Yl)Ethanone)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.14 Å Release Date: 2016-11-02
Classification: TRANSFERASE
Ligands: EDO, DMS, GOL, PEG, 6XH

5I40 image
Brd9 In Complex With Cpd1 (6-Methyl-1,6-Dihydro-7H-Pyrrolo[2,3-C]Pyridin-7-One)

5I7X image
Brd9 In Complex With Cpd2 (N,N-Dimethyl-3-(6-Methyl-7-Oxo-6,7-Dihydro-1H-Pyrrolo[2,3-C]Pyridin-4-Yl)Benzamide)

5I7Y image
Brd9 In Complex With Cpd4 ((E)-3-(6-(But-2-En-1-Yl)-7-Oxo-6,7-Dihydro-1H-Pyrrolo[2,3-C]Pyridin-4-Yl)-N,N-Dimethylbenzamide)

5I80 image
Brd4 In Complex With Cpd2 (N,N-Dimethyl-3-(6-Methyl-7-Oxo-6,7-Dihydro-1H-Pyrrolo[2,3-C]Pyridin-4-Yl)Benzamide)

5I88 image
Brd4 In Complex With Cpd4 ((E)-3-(6-(But-2-En-1-Yl)-7-Oxo-6,7-Dihydro-1H-Pyrrolo[2,3-C]Pyridin-4-Yl)-N,N-Dimethylbenzamide)

5JIY image
Structure Of G9A Set-Domain With Histone H3K9Norleucine Mutant Peptide And Bound S-Adenosylmethionine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.48 Å Release Date: 2016-09-14
Classification: TRANSFERASE
Ligands: ZN, SAM
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