Search Count: 41
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Pdgfra-G680R Mutant Kinase Domain In Complex With Avapritinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: 9JI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: 9JI
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Pdgfra-G680R Mutant Kinase Domain In Complex With A 6,7-Dimethoxyquinazoline-Based Compound (43)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JVO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JVO
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Pdgfra-G680R Mutant Kinase Domain In Complex With A 6,7-Bis(2-Methoxyethoxy)Quinazoline-Based Compound (44)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JVS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JVS
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Pdgfra-G680R Mutant Kinase Domain In Complex With A 7-Methoxyquinazolin-6-Ol-Based Compound (45)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JVR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JVR
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Kit Kinase Domain In Complex With A Pyrrolotriazine-Based Compound (11)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JVQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JVQ
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Kit Kinase Domain In Complex With An Aminopyrimidine-Based Compound (15)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JV1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JV1
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Kit Kinase Domain In Complex With A Pyrrolopyrimidine-Based Compound (17)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JVP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JVP
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Kit Kinase Domain In Complex With A 6-,7-Dimethoxyquinoline-Based Compound (19)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JVT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JVT
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Kit Kinase Domain In Complex With A 7-Methylquinazoline-Based Compound (25)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JVW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JVW
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Kit Kinase Domain In Complex With A 6,7-Bis(2-Methoxyethoxy)Quinazoline-Based Compound (33)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JVV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JVV
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Kit Kinase Domain In Complex With A 6,7-Dimethoxyquinazoline-Based Compound (34)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JVZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JVZ
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Kit Kinase Domain In Complex With A Quinoline-3-Carbonitrile-Based Compound (38)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JVY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JVY
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Kit Kinase Domain In Complex With A Methyl Quinazoline-7-Carboxylate-Based Compound (41)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JV0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JV0
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Kit Kinase Domain In Complex With A 7-Methoxyquinazolin-6-Ol-Based Compound (45)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JVR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JVR
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Akt1 Mutant In Complex With Miransertib (Arq 092)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2026-07-01 Classification: TRANSFERASE Ligands: 6S1, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-01
Ligands: 6S1, EDO, GOL
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Pdgfra-T674I In Complex With Covalent Ponatinib Derivative 19
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2025-02-12 Classification: TRANSFERASE Ligands: A1IRC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-12
Ligands: A1IRC
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Enah Evh1 In Complex With Ac-[2-Cl-F]-[Prom-2]-[Prom-1]-Nh2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.36 Å Release Date: 2020-11-25 Classification: CELL INVASION Ligands: NO3, RJQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-25
Ligands: NO3, RJQ
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Enah Evh1 In Complex With Ac-[2-Cl-F]-Pppptedea-Nh2
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.48 Å Release Date: 2020-11-04 Classification: CELL ADHESION Ligands: NO3 |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2020-11-04
Ligands: NO3
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Enah Evh1 In Complex With Ac-[2-Cl-F]-[Prom-2]-[Prom-17]-Ome
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:0.78 Å Release Date: 2020-10-07 Classification: CELL INVASION Ligands: NO3 |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2020-10-07
Ligands: NO3
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Enah Evh1 In Complex With Ac-[2-Cl-F]-[Prom-2]-[Prom-15]-Oh
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.10 Å Release Date: 2020-05-13 Classification: CELL ADHESION Ligands: K0K, NO3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-05-13
Ligands: K0K, NO3
