Search Count: 22
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Crystal Structure Of Beta-Trcp Bound By Monophosphorylated Nrf2 Degron Peptide.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2026-04-08 Classification: LIGASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-04-08
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Crystal Structure Of Beta-Trcp Bound By Diphosphorylated Nrf2 Degron Peptide.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2026-04-08 Classification: LIGASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-04-08
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Discovery And Optimisation Of Potent, Efficacious And Selective Inhibitors Targeting Egfr Exon20 Insertion Mutations. Compound 16 Bound To Egfr
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.51 Å Release Date: 2024-06-05 Classification: SIGNALING PROTEIN Ligands: 2I0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-05
Ligands: 2I0
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Discovery And Optimisation Of Potent, Efficacious And Selective Inhibitors Targeting Egfr Exon20 Insertion Mutations. Compound 12 Bound To Egfrinsnpg
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.52 Å Release Date: 2024-06-05 Classification: SIGNALING PROTEIN Ligands: 2I6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-05
Ligands: 2I6
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Discovery And Optimisation Of Potent, Efficacious And Selective Inhibitors Targeting Egfr Exon20 Insertion Mutations. Compound 22 Bound To Egfrinsnpg [V948R]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2024-06-05 Classification: SIGNALING PROTEIN Ligands: 2EI, IOD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-05
Ligands: 2EI, IOD
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Discovery And Optimisation Of Potent, Efficacious And Selective Inhibitors Targeting Egfr Exon20 Insertion Mutations. Compound 33 Bound To Egfrinsnpg [V948R]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.28 Å Release Date: 2024-06-05 Classification: SIGNALING PROTEIN Ligands: 26X |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-05
Ligands: 26X
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Discovery And Optimisation Of Potent, Efficacious And Selective Inhibitors Targeting Egfr Exon20 Insertion Mutations. Compound 18 Bound To Egfr[V948R]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.13 Å Release Date: 2024-06-05 Classification: SIGNALING PROTEIN Ligands: 2II |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-05
Ligands: 2II
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Discovery And Optimisation Of Potent, Efficacious And Selective Inhibitors Targeting Egfr Exon20 Insertion Mutations. Compound 33 Bound To Egfr[V948R]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2024-06-05 Classification: SIGNALING PROTEIN Ligands: 26X, ATP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-05
Ligands: 26X, ATP, MG
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Eed In Complex With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.61 Å Release Date: 2021-12-08 Classification: PROTEIN BINDING Ligands: L9W, 51A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-12-08
Ligands: L9W, 51A
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Eed In Complex With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2021-12-08 Classification: PROTEIN BINDING Ligands: L9W, 52R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-12-08
Ligands: L9W, 52R
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Eed In Complex With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2021-12-08 Classification: PROTEIN BINDING Ligands: MG, L9W, 54N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-12-08
Ligands: MG, L9W, 54N
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Eed In Complex With A Cyano-Benzofuran
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2021-05-12 Classification: PROTEIN BINDING Ligands: CA, L9W, PV5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-12
Ligands: CA, L9W, PV5
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Eed In Complex With A Triazolopyrimidine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2021-05-12 Classification: PROTEIN BINDING Ligands: L9W, GOL, EJR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-12
Ligands: L9W, GOL, EJR
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Crystal Structure Of The Bcl6 Btb Domain In Complex With Anilinopyrimidine Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.39 Å Release Date: 2018-10-24 Classification: TRANSFERASE Ligands: C0H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-24
Ligands: C0H
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Crystal Structure Of The Bcl6 Btb Domain In Complex With Anilinopyrimidine Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2018-10-24 Classification: TRANSFERASE Ligands: CL, C1W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-24
Ligands: CL, C1W
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Crystal Structure Of The Bcl6 Btb Domain In Complex With Anilinopyrimidine Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2018-10-24 Classification: TRANSFERASE Ligands: CL, C0Q |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-24
Ligands: CL, C0Q
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Crystal Structure Of The Protein Kinase Ck2 Catalytic Subunit In Complex With Pyrazolo-Pyrimidine Macrocyclic Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.52 Å Release Date: 2017-05-17 Classification: TRANSFERASE Ligands: SO4, EDO, 8GQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-17
Ligands: SO4, EDO, 8GQ
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Crystal Structure Of The Bcl6 Btb Domain In Complex With Pyrazolo-Pyrimidine Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2017-05-17 Classification: TRANSFERASE Ligands: 8HH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-17
Ligands: 8HH
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Crystal Structure Of The Bcl6 Btb Domain In Complex With Pyrazolo-Pyrimidine Macrocyclic Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.81 Å Release Date: 2017-05-17 Classification: TRANSFERASE Ligands: CL, 8GQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-17
Ligands: CL, 8GQ
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Crystal Structure Of The Bcl6 Btb Domain In Complex With Pyrazolo-Pyrimidine Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.38 Å Release Date: 2017-05-17 Classification: TRANSFERASE Ligands: 8GN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-17
Ligands: 8GN