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Erap1 In Complex With 1-[2-(5-Bromo-7-Fluoro-2-Oxo-2,3-Dihydro-1,3-Benzothiazol-3-Yl)Acetamido]-4,4-Difluorocyclohexane-1-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2026-05-06 Classification: PEPTIDE BINDING PROTEIN Ligands: ZN, SIN, PO4, EDO, A1JVE |
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Erap1 In Complex With 1-[2-(6-Bromo-2,2-Difluoro-3-Oxo-3,4-Dihydro-2H-1,4-Benzoxazin-4-Yl)Acetamido]Cyclohexane-1-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.57 Å Release Date: 2026-04-22 Classification: PEPTIDE BINDING PROTEIN Ligands: ZN, PO4, EDO, A1JVD |
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Erap1 In Complex With 1-[2-(2-Oxo-5-Phenyl-2,3-Dihydro-1,3-Benzoxazol-3-Yl)Acetamido]Cyclohexane-1-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2026-04-22 Classification: PEPTIDE BINDING PROTEIN Ligands: ZN, MLT, EDO, A1JVG |
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Erap1 In Complex With 1-[2-(5-Chloro-2-Oxo-2,3-Dihydro-1,3-Benzothiazol-3-Yl)Acetamido]Cyclohexane-1-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2026-04-22 Classification: PEPTIDE BINDING PROTEIN Ligands: ZN, PO4, EDO, A1JVH |
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Erap1 In Complex With 1-[2-(3-Oxo-6-Phenyl-3,4-Dihydro-2H-1,4-Benzoxazin-4-Yl)Acetamido]Cyclohexane-1-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.37 Å Release Date: 2026-04-22 Classification: PEPTIDE BINDING PROTEIN Ligands: ZN, PO4, EDO, A1JVF |
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Organism: Methanocaldococcus jannaschii
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2023-07-12 Classification: DNA BINDING PROTEIN |
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Human Jak3 Kinase Domain With 1-(4-((2-((1-Methyl-1H-Pyrazol-4-Yl)Amino)Quinazolin-8-Yl)Amino)Piperidin-1-Yl)Ethan-1-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2022-02-02 Classification: SIGNALING PROTEIN Ligands: 934, SO4, PHU |
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Jak2 In Complex With 4-{8-Methoxy-2-[(1-Methyl-1H-Pyrazol-4-Yl)Amino]Quinazolin-6-Yl}Phenol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2022-02-02 Classification: SIGNALING PROTEIN Ligands: 9I8 |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.61 Å Release Date: 2022-02-02 Classification: SIGNALING PROTEIN Ligands: 9I5 |
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Jak2 In Complex With 4-(2-Amino-8-{[(2S)-1-Hydroxypropan-2-Yl]Amino}Quinazolin-6-Yl)-5-Ethyl-2-Fluorophenol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2022-02-02 Classification: SIGNALING PROTEIN Ligands: 9I2, GOL |
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Jak2 In Complex With 4-(2-{[5-(Dimethylamino)Pentyl]Amino}-8-{[(2S)-1-Hydroxypropan-2-Yl]Amino}Quinazolin-6-Yl)-5-Ethyl-2-Fluorophenol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2022-02-02 Classification: SIGNALING PROTEIN Ligands: 9HR |
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Organism: Escherichia coli
Method: SOLUTION NMR Release Date: 2018-06-06 Classification: RNA BINDING PROTEIN |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2016-05-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 65C, MG, MES |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2016-05-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 65A |














