Search Count: 40
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Structure Of Human Vaccinia-Related Kinase 1 (Vrk1) Bound To Ldsm311
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2020-03-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, RYA, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-03-11
Ligands: SO4, RYA, EDO
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Human Prpf4B Bound To Benzothiophene Inhibitor 224
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2019-08-28 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: OCJ, EDO, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-28
Ligands: OCJ, EDO, PO4
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Human Prpf4B Bound To Benzothiophene Inhibitor 329
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2019-08-28 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: SO4, OND |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-28
Ligands: SO4, OND
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Human Pim1 Bound To Benzothiophene Inhibitor 213
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2019-07-24 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: O97, GOL |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2019-07-24
Ligands: O97, GOL
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Human Pim1 Bound To Benzothiophene Inhibitor 224
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2019-07-24 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: OCJ, GOL, EDO |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2019-07-24
Ligands: OCJ, GOL, EDO
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Human Pim1 Bound To Benzothiophene Inhibitor 292
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2019-07-24 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: OD4, GOL |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2019-07-24
Ligands: OD4, GOL
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Human Pim1 Bound To Benzothiophene Inhibitor 354
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2019-07-24 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: OD1 |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2019-07-24
Ligands: OD1
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Human Pim1 Bound To Benzothiophene Inhibitor 379
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2019-07-24 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: SO4, OBY |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2019-07-24
Ligands: SO4, OBY
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Crystal Structure Of The Human Vaccinia-Related Kinase Bound To A N,N-Dipropynyl-Dihydropteridine-3-Hydroxyindazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2019-02-20 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: KWJ, SO4, EDO, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-20
Ligands: KWJ, SO4, EDO, PEG
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Crystal Structure Of Human Vaccinia-Related Kinase 2 (Vrk-2) Bound To Pyridin-Benzenesulfonamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2019-01-16 Classification: TRANSFERASE Ligands: KJD, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-01-16
Ligands: KJD, SO4
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Co-Crystal Of Pseudokinase Drik1 (Drought Responsive Inactive Kinase 1) Bound To Enmd-2076
Organism: Zea mays
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2018-08-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: J3A, GOL |
Organism: Zea mays
Method: X-RAY DIFFRACTION
Release Date: 2018-08-22
Ligands: J3A, GOL
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Crystal Structure Of Sugarcane Sapk10 (Serine/Threonine-Protein Kinase 10)
Organism: Saccharum officinarum complex
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2018-08-15 Classification: SIGNALING PROTEIN Ligands: GOL |
Organism: Saccharum officinarum complex
Method: X-RAY DIFFRACTION
Release Date: 2018-08-15
Ligands: GOL
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Crystal Structure Of The Human Vaccinia-Related Kinase Bound To A N,N-Dipropyl-Dihydropteridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2018-05-23 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: CL, ACT, G6J, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-23
Ligands: CL, ACT, G6J, SO4, GOL
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Crystal Structure Of The Human Vaccinia-Related Kinase 1 (Vrk1) Bound To An N-Propynyl-N-Isopentyl-Dihydropteridin Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2018-04-04 Classification: Transferase/Transferase Inhibitor Ligands: F87, SO4, ACT, GOL, FCS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-04-04
Ligands: F87, SO4, ACT, GOL, FCS
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Structure Of Apo Grmzm2G135359 Pseudokinase
Organism: Zea mays
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2018-04-04 Classification: TRANSFERASE |
Organism: Zea mays
Method: X-RAY DIFFRACTION
Release Date: 2018-04-04
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Crystal Structure Of The Human Vaccinia-Related Kinase Bound To A N-Methyl-N-Propyl-Dihydropteridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2018-04-04 Classification: Transferase/Transferase Inhibitor Ligands: SO4, ACT, PG4, FBY, GOL, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-04-04
Ligands: SO4, ACT, PG4, FBY, GOL, CL
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Human Prpf4B In Complex With Rebastinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2018-03-28 Classification: TRANSFERASE Ligands: 919, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-28
Ligands: 919, SO4
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Crystal Structure Of The Human Vaccinia-Related Kinase Bound To A N-Propynyl-N-Ethyl-Dihydropteridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2018-03-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: F8Y, SO4, ACT, GOL, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-28
Ligands: F8Y, SO4, ACT, GOL, CL
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Crystal Structure Of The Human Vaccinia-Related Kinase Bound To A N,N-Dipropynyl-Dihydropteridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2018-03-21 Classification: Transferase/Transferase Inhibitor Ligands: ACT, F7D, SO4, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-21
Ligands: ACT, F7D, SO4, PEG
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Crystal Structure Of The Human Camkk1A In Complex With Hesperadin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2018-03-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: H1N, SCN, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-07
Ligands: H1N, SCN, EDO
