Search Count: 15
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Crystal Structure Of The First Bromodomain Of Human Brdt In Complex With The Inhibitor Ccd-956
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2022-06-08 Classification: TRANSCRIPTION/INHIBITOR Ligands: MJN, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-06-08
Ligands: MJN, DMS
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Oxa-48 Bound By Compound 2.2
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2021-12-15 Classification: HYDROLASE/INHIBITOR Ligands: VBV, CL |
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION
Release Date: 2021-12-15
Ligands: VBV, CL
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Oxa-48 Bound By Compound 2.3
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2021-12-01 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: VAJ, NA, EDO, PEG, CL |
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION
Release Date: 2021-12-01
Ligands: VAJ, NA, EDO, PEG, CL
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Oxa-48 Bound By Compound 3.1
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2021-12-01 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: BIH, CL, NA, EDO |
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION
Release Date: 2021-12-01
Ligands: BIH, CL, NA, EDO
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Oxa-48 Bound By Compound 4.3
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2021-12-01 Classification: HYDROLASE/INHIBITOR Ligands: EDO, XV7, NA, CL |
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION
Release Date: 2021-12-01
Ligands: EDO, XV7, NA, CL
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Oxa-48 Bound By Compound 3.3
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2021-12-01 Classification: HYDROLASE/INHIBITOR Ligands: 3I0, EDO, DMS, CL |
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION
Release Date: 2021-12-01
Ligands: 3I0, EDO, DMS, CL
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Crystal Structure Of Brdt Bromodomain 2 In Complex With Cdd-1302
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2021-06-30 Classification: TRANSCRIPTION Ligands: XWJ, JEF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-06-30
Ligands: XWJ, JEF
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Crystal Structure Of Brdt Bromodomain 2 In Complex With Cdd-1102
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2021-06-30 Classification: TRANSCRIPTION/INHIBITOR Ligands: XWP, BME |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-06-30
Ligands: XWP, BME
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Oxa-48 Bound By Inhibitor Cdd-97
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2020-05-06 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: QHY, EDO, GOL, CL |
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION
Release Date: 2020-05-06
Ligands: QHY, EDO, GOL, CL
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Crystal Structure Of T110A Mutant Human Glutamate Oxaloacetate Transaminase 1 (Got1)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2018-11-14 Classification: TRANSFERASE Ligands: PG4, PLP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-14
Ligands: PG4, PLP
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Crystal Structure Of T110A:S256A Mutant Human Glutamate Oxaloacetate Transaminase 1 (Got1)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2018-11-14 Classification: TRANSFERASE Ligands: PG4, GOL, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-14
Ligands: PG4, GOL, PO4
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Crystal Structure Of Wild-Type (Wt) Human Glutamate Oxaloacetate Transaminase 1 (Got1)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2018-11-14 Classification: TRANSFERASE Ligands: PG4, PLP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-14
Ligands: PG4, PLP
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Crystal Structure Of A Metabolic Reductase With 1-Hydroxy-6-(4-Hydroxybenzyl)-4-Methylpyridin-2(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.31 Å Release Date: 2013-05-22 Classification: oxidoreductase/oxidoreductase inhibitor Ligands: NDP, SO4, 1BX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-22
Ligands: NDP, SO4, 1BX
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Crystal Structure Of A Metabolic Reductase With 6-Benzyl-1-Hydroxy-4-Methylpyridin-2(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.29 Å Release Date: 2013-05-22 Classification: oxidoreductase/oxidoreductase inhibitor Ligands: NDP, SO4, 1BZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-22
Ligands: NDP, SO4, 1BZ
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Crystal Structure Of Human Dot1L In Complex With A Selective Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2011-10-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: TT8, GOL, ACT, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-05
Ligands: TT8, GOL, ACT, SO4
