Search Count: 55
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Crystal Structure Of Human Kras G12C Covalently Bound To Thiazol-2-Yl Piperidine Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2026-08-12 Classification: SIGNALING PROTEIN Ligands: MG, GDP, A1DI3, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-08-12
Ligands: MG, GDP, A1DI3, EDO
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Crystal Structure Of Human Kras G12C Covalently Bound To 4-Methyl-Thiazol-5-Yl Piperidine Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.10 Å Release Date: 2026-08-12 Classification: SIGNALING PROTEIN Ligands: MG, GDP, A1DI5, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-08-12
Ligands: MG, GDP, A1DI5, EDO
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Crystal Structure Of Human Kras G12C Covalently Bound To 1,4-Dimethyl-Pyrazol-5-Yl Piperidine Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.26 Å Release Date: 2026-08-12 Classification: SIGNALING PROTEIN Ligands: MG, GDP, A1DI6, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-08-12
Ligands: MG, GDP, A1DI6, EDO
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Crystal Structure Of Human Kras G12C Covalently Bound To Am-8719
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2026-08-12 Classification: SIGNALING PROTEIN Ligands: MG, GDP, A1DI7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-08-12
Ligands: MG, GDP, A1DI7
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Crystal Structure Of Human Kras G12D In Complex With Gdp And Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.25 Å Release Date: 2026-07-22 Classification: SIGNALING PROTEIN,ONCOPROTEIN/INHIBITOR Ligands: MG, GDP, A1CZE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-22
Ligands: MG, GDP, A1CZE
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Crystal Structure Of Human Kras G12D In Complex With Gdp And Am-2383
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.25 Å Release Date: 2026-07-22 Classification: SIGNALING PROTEIN,ONCOPROTEIN/INHIBITOR Ligands: MG, GDP, A1AG3, EDO, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-22
Ligands: MG, GDP, A1AG3, EDO, SO4
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Crystal Structure Of Human Kras G12D In Complex With Gmppcp And Am-2383
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.12 Å Release Date: 2026-07-22 Classification: SIGNALING PROTEIN,ONCOPROTEIN/INHIBITOR Ligands: MG, GCP, A1AG3, EDO, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-22
Ligands: MG, GCP, A1AG3, EDO, SO4
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Crystal Structure Of Human Kras G12V In Complex With Gdp And Am-2383
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.20 Å Release Date: 2026-07-22 Classification: SIGNALING PROTEIN,ONCOPROTEIN/INHIBITOR Ligands: MG, GDP, A1AG3, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-22
Ligands: MG, GDP, A1AG3, EDO
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Crystal Structure Of Human Kras G12V In Complex With Gmppcp And Am-2383
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.20 Å Release Date: 2026-07-22 Classification: SIGNALING PROTEIN,ONCOPROTEIN/INHIBITOR Ligands: MG, GCP, A1AG3, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-22
Ligands: MG, GCP, A1AG3, EDO
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Structure Determination Of Pedobacter Sp. Kp-2 Pahz1
Organism: Pedobacter sp. kp-2
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2026-03-11 Classification: HYDROLASE |
Organism: Pedobacter sp. kp-2
Method: X-RAY DIFFRACTION
Release Date: 2026-03-11
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From Dna-Encoded Library Screening To Am-9747 - An Mta-Cooperative Prmt5 Inhibitor With Potent Oral In Vivo Efficacy
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2025-03-26 Classification: TRANSFERASE/INHIBITOR Ligands: A1BQW, MTA, GOL, PEG, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-03-26
Ligands: A1BQW, MTA, GOL, PEG, DMS
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Crystal Structure Of Human Kras G12C Covalently Bound To Del Triazine Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2025-02-26 Classification: SIGNALING PROTEIN,ONCOPROTEIN/INHIBITOR Ligands: CA, GDP, A1BH6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-26
Ligands: CA, GDP, A1BH6
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Crystal Structure Of Human Kras G12C Covalently Bound To Nopinone-Derived Naphthol Compound 21
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.18 Å Release Date: 2025-02-26 Classification: SIGNALING PROTEIN,ONCOPROTEIN/INHIBITOR Ligands: MG, GDP, A1BH5, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-26
Ligands: MG, GDP, A1BH5, EDO
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Amg 193, A Clinical Stage Mta-Cooperative Prmt5 Inhibitor, Drives Anti-Tumor Activity Preclinically And In Patients With Mtap-Deleted Cancers
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2024-10-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GOL, DMS, A1ATH, MTA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-02
Ligands: GOL, DMS, A1ATH, MTA
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Crystal Structure Of A Mycobacteriophage Cluster A2 Immunity Repressor:Dna Complex
Organism: Mycobacterium phage tipsythetrex
Method: X-RAY DIFFRACTION Resolution:3.13 Å Release Date: 2022-07-20 Classification: GENE REGULATION/DNA |
Organism: Mycobacterium phage tipsythetrex
Method: X-RAY DIFFRACTION
Release Date: 2022-07-20
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Crystal Structure Of A Mycobacteriophage Cluster A2 Immunity Repressor:Dna Complex
Organism: Mycobacterium phage tipsythetrex
Method: X-RAY DIFFRACTION Resolution:2.79 Å Release Date: 2022-07-20 Classification: GENE REGULATION/DNA |
Organism: Mycobacterium phage tipsythetrex
Method: X-RAY DIFFRACTION
Release Date: 2022-07-20
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Structure Of Poly(Aspartic Acid) Hydrolase Pahz2 With Zn+2 Bound
Organism: Sphingomonas sp. kt-1
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2021-12-08 Classification: HYDROLASE Ligands: ZN |
Organism: Sphingomonas sp. kt-1
Method: X-RAY DIFFRACTION
Release Date: 2021-12-08
Ligands: ZN
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Structure Of Poly(Aspartic Acid) Hydrolase Pahz2 With Gd+3 Bound
Organism: Sphingomonas sp. kt-1
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2021-12-08 Classification: HYDROLASE Ligands: GD3 |
Organism: Sphingomonas sp. kt-1
Method: X-RAY DIFFRACTION
Release Date: 2021-12-08
Ligands: GD3
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A Structural Characterization Of Poly(Aspartic Acid) Hydrolase-1 From Sphingomonas Sp. Kt-1.
Organism: Sphingomonas sp. kt-1
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2020-12-09 Classification: HYDROLASE |
Organism: Sphingomonas sp. kt-1
Method: X-RAY DIFFRACTION
Release Date: 2020-12-09
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Crystal Structure Of Bace1 In Complex With (Z)-Fluoro-Olefin Containing Compound 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2020-06-03 Classification: HYDROLASE/HYDROLASE Inhibitor Ligands: U64, IOD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-06-03
Ligands: U64, IOD
