Search Count: 16
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Type-Iii C-Met Inhibitor Enabled By Free-Energy Perturbation Calculations
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2026-05-27 Classification: TRANSFERASE Ligands: A1C9B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-05-27
Ligands: A1C9B
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Crystal Structure Of Human Cyclic Gmp-Amp Synthase (Cgas) In Complex With Compound 5; 3-((2-((3-Chloro-4-Fluorophenyl)Amino)-2-Oxoethyl)Carbamoyl)Picolinic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.53 Å Release Date: 2025-01-01 Classification: TRANSFERASE Ligands: ANP, A1BJH, ZN, MN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-01
Ligands: ANP, A1BJH, ZN, MN
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Crystal Structure Of Human Cyclic Gmp-Amp Synthase (Cgas) In Complex With Compound 36; (S)-(6,7-Dichloro-1-Methyl-1,3,4,5-Tetrahydro-2H-Pyrido[4,3-B]Indol-2-Yl)(5-(2-Hydroxyethoxy)Pyrimidin-2-Yl)Methanone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.25 Å Release Date: 2025-01-01 Classification: TRANSFERASE Ligands: ZN, A1BJA, ANP, MN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-01
Ligands: ZN, A1BJA, ANP, MN
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Crystal Structure Of Human Cyclic Gmp-Amp Synthase (Cgas) In Complex With Compound 23; (S)-1-(6,7-Dichloro-1-Methyl-1,3,4,5-Tetrahydro-2H-Pyrido[4,3-B]Indol-2-Yl)-2-Methoxyethan-1-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2025-01-01 Classification: TRANSFERASE Ligands: ZN, A1BJD, ANP, MN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-01
Ligands: ZN, A1BJD, ANP, MN
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The Allosteric Binding Mode Of Alphad-Conotoxin Vxxxb
Organism: Lymnaea stagnalis, Conus vexillum
Method: X-RAY DIFFRACTION Resolution:2.47 Å Release Date: 2023-04-12 Classification: PEPTIDE BINDING PROTEIN |
Organism: Lymnaea stagnalis, Conus vexillum
Method: X-RAY DIFFRACTION
Release Date: 2023-04-12
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Structure-Function Characterization Of An Aldo-Keto Reductase Involved In Detoxification Of The Mycotoxin, Deoxynivalenol
Organism: Rhizobium leguminosarum
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2022-09-07 Classification: OXIDOREDUCTASE Ligands: SO4, FLC |
Organism: Rhizobium leguminosarum
Method: X-RAY DIFFRACTION
Release Date: 2022-09-07
Ligands: SO4, FLC
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Alpha-Conotoxin Omia With Unusual Pharmacological Properties At Alpha7 Nicotinic Receptors
Organism: Lymnaea stagnalis, Conus omaria
Method: X-RAY DIFFRACTION Resolution:2.47 Å Release Date: 2021-12-01 Classification: CHOLINE-BINDING PROTEIN |
Organism: Lymnaea stagnalis, Conus omaria
Method: X-RAY DIFFRACTION
Release Date: 2021-12-01
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Rigidity Of Loop 1 Contributes To Equipotency Of Globular And Ribbon Isomers Of Alpha-Conotoxin Ausia
Organism: Lymnaea stagnalis, Conus australis
Method: X-RAY DIFFRACTION Resolution:2.46 Å Release Date: 2021-11-17 Classification: CHOLINE-BINDING PROTEIN/ANTAGONIST |
Organism: Lymnaea stagnalis, Conus australis
Method: X-RAY DIFFRACTION
Release Date: 2021-11-17
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Rigidity Of Loop 1 Contributes To Equipotency Of Globular And Ribbon Isomers Of Alpha-Conotoxin Ausia
Organism: Lymnaea stagnalis, Conus australis
Method: X-RAY DIFFRACTION Resolution:2.58 Å Release Date: 2021-11-17 Classification: CHOLINE-BINDING PROTEIN/ANTAGONIST |
Organism: Lymnaea stagnalis, Conus australis
Method: X-RAY DIFFRACTION
Release Date: 2021-11-17
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Nmr Structure Of Truncated Alpha Conotoxin Sii: Ile-Sii(3-14)
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Organism: Conus striatus
Method: SOLUTION NMR
Release Date: 2020-05-06
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Structure Of Single Disulfide Peptide Czon1107-P5A
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Organism: Conus zonatus
Method: SOLUTION NMR
Release Date: 2020-04-08
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Structure Of Single Disulfide Peptide Czon1107-Wt (Major Conformer)
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Organism: Conus zonatus
Method: SOLUTION NMR
Release Date: 2020-04-08
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Structure Of Single Disulfide Peptide Czon1107-Wt (Minor Conformer)
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Organism: Conus zonatus
Method: SOLUTION NMR
Release Date: 2020-04-08
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Structure Of Single Disulfide Peptide Czon1107-P7A (Minor Conformer)
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Organism: Conus zonatus
Method: SOLUTION NMR
Release Date: 2020-04-08
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Structure Of Single Disulfide Peptide Czon1107-P7A(Major Conformer)
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Organism: Conus zonatus
Method: SOLUTION NMR
Release Date: 2020-04-08
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Structural Mechanisms For Alpha-Conotoxin Selectivity At The Human Alpha3Beta4 Nicotinic Acetylcholine Receptor
Organism: Lymnaea stagnalis, Conus
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2017-04-12 Classification: PROTEIN BINDING |
Organism: Lymnaea stagnalis, Conus
Method: X-RAY DIFFRACTION
Release Date: 2017-04-12
