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Search Count: 4

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4RWJ image
Crystal Structure Of Fgfr1 (C488A, C584S) In Complex With Azd4547 (N-{3-[2-(3,5-Dimethoxyphenyl)Ethyl]-1H-Pyrazol-5-Yl}-4-[(3R,5S)-3,5-Dimethylpiperazin-1-Yl]Benzamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.49 Å Release Date: 2015-04-22
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: 66T

4RWK image
Crystal Structure Of V561M Fgfr1 Gatekeeper Mutation (C488A, C584S, V561M) In Complex With N-{3-[2-(3,5-Dimethoxyphenyl)Ethyl]-1H-Pyrazol-5-Yl}-4-[(3R,5S)-3,5-Dimethylpiperazin-1-Yl]Benzamide (Azd4547)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.98 Å Release Date: 2015-04-15
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: 66T, MG

4V05 image
Fgfr1 In Complex With Azd4547.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.57 Å Release Date: 2014-12-10
Classification: TRANSFERASE
Ligands: EDO, 66T, SO4

4WUN image
Structure Of Fgfr1 In Complex With Azd4547 (N-{3-[2-(3,5-Dimethoxyphenyl)Ethyl]-1H-Pyrazol-5-Yl}-4-[(3R,5S)-3,5-Dimethylpiperazin-1-Yl]Benzamide) At 1.65 Angstrom
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.65 Å Release Date: 2014-11-19
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: 66T
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