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Crystal Structure Of Fgfr1 (C488A, C584S) In Complex With Azd4547 (N-{3-[2-(3,5-Dimethoxyphenyl)Ethyl]-1H-Pyrazol-5-Yl}-4-[(3R,5S)-3,5-Dimethylpiperazin-1-Yl]Benzamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2015-04-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 66T |
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Crystal Structure Of V561M Fgfr1 Gatekeeper Mutation (C488A, C584S, V561M) In Complex With N-{3-[2-(3,5-Dimethoxyphenyl)Ethyl]-1H-Pyrazol-5-Yl}-4-[(3R,5S)-3,5-Dimethylpiperazin-1-Yl]Benzamide (Azd4547)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.98 Å Release Date: 2015-04-15 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 66T, MG |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.57 Å Release Date: 2014-12-10 Classification: TRANSFERASE Ligands: EDO, 66T, SO4 |
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Structure Of Fgfr1 In Complex With Azd4547 (N-{3-[2-(3,5-Dimethoxyphenyl)Ethyl]-1H-Pyrazol-5-Yl}-4-[(3R,5S)-3,5-Dimethylpiperazin-1-Yl]Benzamide) At 1.65 Angstrom
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2014-11-19 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 66T |




