Search Count: 6
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Dissecting Therapeutic Resistance To Erk Inhibition Rat Wild Type Sch772984 In Complex With (3R)-1-(2-Oxo-2-{4-[4-(Pyrimidin-2-Yl)Phenyl]Piperazin-1-Yl}Ethyl)-N-[3-(Pyridin-4-Yl)-2H-Indazol-5-Yl]Pyrrolidine-3-Carboxamide
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2016-02-24 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 38Z, SO4, PG4, DMS |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2016-02-24
Ligands: 38Z, SO4, PG4, DMS
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Dissecting Therapeutic Resistance To Erk Inhibition Rat Mutant Sch772984 In Complex With (3R)-1-(2-Oxo-2-{4-[4-(Pyrimidin-2-Yl)Phenyl]Piperazin-1-Yl}Ethyl)-N-[3-(Pyridin-4-Yl)-2H-Indazol-5-Yl]Pyrrolidine-3-Carboxamide
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2016-02-24 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 38Z, SO4 |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2016-02-24
Ligands: 38Z, SO4
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Structure Of Human Erk2 In Complex With Sch772984 Revealing A Novel Inhibitor-Induced Binding Pocket
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2014-07-23 Classification: Transferase/transferase inhibitor Ligands: EDO, SO4, 38Z |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-23
Ligands: EDO, SO4, 38Z
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Structure Of Human Erk1 In Complex With Sch772984 Revealing A Novel Inhibitor-Induced Binding Pocket
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2014-07-23 Classification: Transferase/transferase inhibitor Ligands: EDO, DMS, CL, SO4, 38Z |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-23
Ligands: EDO, DMS, CL, SO4, 38Z
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Structure Of Human Haspin (Gsg2) In Complex With Sch772984 Revealing The First Type-I Binding Mode
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2014-07-23 Classification: Transferase/transferase inhibitor Ligands: MPD, GOL, 38Z |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-23
Ligands: MPD, GOL, 38Z
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Structure Of Human Jnk1 In Complex With Sch772984 And The Amppnp-Hydrolysed Triphosphate Revealing The Second Type-I Binding Mode
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2014-07-23 Classification: Transferase/transferase inhibitor Ligands: EDO, EPE, 38Z, ANP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-23
Ligands: EDO, EPE, 38Z, ANP, MG