9BRN image
Deposition Date 2024-05-11
Release Date 2025-11-12
Last Version Date 2025-11-12
Entry Detail
PDB ID:
9BRN
Keywords:
SIGNALING PROTEIN/INHIBITOR
Title:
Crystal Structure of Human G Protein-Coupled Receptor Kinase 5 in Complex with GRL050-22
Biological Source:
Source Organism(s):
Homo sapiens (Taxon ID: 9606)
Expression System(s):
Escherichia coli bl21(de3)
Method Details:
Experimental Method:
X-RAY DIFFRACTION
Resolution:
2.90 Å
R-Value Free:
0.25
R-Value Work:
0.20
R-Value Observed:
0.20
Space Group:
P 41 21 2
9BRN validation report missing
Macromolecular Entities
Structures with similar UniProt ID
Structural Superimposition Protein Blast
Polymer Type:polypeptide(L)
Molecule:G protein-coupled receptor ki
Gene (Uniprot):GRK5
Chain IDs:A
Chain Length:598
Number of Molecules:1
Biological Source:Homo sapiens
UniProt ID:P34947 Pfam ID:PF00615, PF00069 EC:2.7.11.16
Ligand Molecules
A1ARD
Primary Citation
Structures of GRK5 bound to novel inhibitors
To be published ? ? ? (?)
Primary Citation of related structures
9BRN
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