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7T97 image
Crystal Structure Of Engineered Cys-Cys Fab Dimer Ch1-207 (Hc4)

7T98 image
Crystal Structure Of Engineered Cys-Cys Fab Dimer Vl-108 (Lc33)

7T99 image
Crystal Structure Of Engineered Cys-Cys Fab Dimer Cl-205 (Lc25)

6OKM image
Human Ox40R (Tnfrsf4) Bound To Fab 3C8

6OGX image
Ternary Complex Of Ox40R (Tnfrsf4) Bound To Fab1 And Fab2

6OKN image
Ox40R (Tnfrsf4) Bound To Fab 1A7

6E25 image
Nmr Solution Structure Of The Card9 Card Bound To Zinc

6E26 image
Nmr Solution Structure Of The Card9 Card

6E27 image
The Card9 Card Domain-Swapped Dimer With A Zinc Ion Bound To One Of The Two Zinc Binding Sites

6E28 image
The Card9 Card Domain-Swapped Dimer

6ALC image
Crebbp Bromodomain In Complex With Cpd 4 (1-(1-(Cyclopropylmethyl)-3-(1H-Indol-4-Yl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridin-5-Yl)Ethan-1-One)

5W0F image
Crebbp Bromodomain In Complex With Cpd3 ((S)-1-(3-(6-(1-Methyl-1H-Pyrazol-4-Yl)-3,4-Dihydroquinolin-1(2H)-Yl)-1-(Tetrahydrofuran-3-Yl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridin-5-Yl)Ethan-1-One)

5W0I image
Crebbp Bromodomain In Complex With Cpd8 (1-(3-(7-(Difluoromethyl)-6-(1-Methyl-1H-Pyrazol-4-Yl)-3,4-Dihydroquinolin-1(2H)-Yl)-1-(Tetrahydrofuran-3-Yl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridin-5-Yl)Ethan-1-One)

5W0L image
Crebbp Bromodomain In Complex With Cpd10 (1-(3-(7-(Difluoromethyl)-6-(1-Methyl-1H-Pyrazol-4-Yl)-3,4-Dihydroquinolin-1(2H)-Yl)-1-(Tetrahydro-2H-Pyran-4-Yl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridin-5-Yl)Ethan-1-One)

5W0Q image
Crebbp Bromodomain In Complex With Cpd17 (N,2,7-Trimethyl-2,3-Dihydro-4H-Benzo[B][1,4]Oxazine-4-Carboxamide)

5W0E image
Crebbp Bromodomain In Complex With Cpd19 (3-(7-(Difluoromethyl)-6-(1-Methyl-1H-Pyrazol-4-Yl)-3,4-Dihydroquinolin-1(2H)-Yl)-N-Methyl-1-(Tetrahydro-2H-Pyran-4-Yl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridine-5-Carboxamide)

6AXQ image
Crebbp Bromodomain In Complex With Cpd6 (Methyl 1H-Indole-3-Carboxylate)

6AY3 image
Crebbp Bromodomain In Complex With Cpd16 (5-(7-(Difluoromethyl)-6-(1-Methyl-1H-Pyrazol-4-Yl)-3,4-Dihydroquinolin-1(2H)-Yl)-N-Methyl-1H-Indole-3-Carboxamide)

6AY5 image
Crebbp Bromodomain In Complex With Cpd17 (5-(7-(Difluoromethyl)-6-(1-Methyl-1H-Pyrazol-4-Yl)-3,4-Dihydroquinolin-1(2H)-Yl)-3-Methylbenzo[D]Thiazol-2(3H)-One)

5KTU image
Crystal Structure Of The Bromodomain Of Human Crebbp Bound To Pyrazolopiperidine Scaffold
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.38 Å Release Date: 2016-11-02
Classification: TRANSFERASE
Ligands: 6XB, DMS
Protein Functional Filters:
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