Search Count: 17
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Hiv Reverse Transcriptase With Compound Pyr01
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2022-11-23 Classification: VIRAL PROTEIN Ligands: 9QI |
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION
Release Date: 2022-11-23
Ligands: 9QI
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Hiv Reverse Transcriptase With Compound Pyr02
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION Resolution:2.08 Å Release Date: 2022-11-23 Classification: VIRAL PROTEIN Ligands: 9PJ |
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION
Release Date: 2022-11-23
Ligands: 9PJ
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Dpp9 In Complex With Ligand Iced-2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.46 Å Release Date: 2022-10-05 Classification: HYDROLASE Ligands: D06 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-10-05
Ligands: D06
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Dpp8 In Complex With Ligand Iced-2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.69 Å Release Date: 2022-10-05 Classification: HYDROLASE Ligands: D06, TMO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-10-05
Ligands: D06, TMO
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Dpp9 In Complex With Ligand Iced-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.78 Å Release Date: 2022-10-05 Classification: HYDROLASE Ligands: CW8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-10-05
Ligands: CW8
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Dpp8 In Complex With Ligand Iced-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.58 Å Release Date: 2022-10-05 Classification: HYDROLASE Ligands: CW8, TMO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-10-05
Ligands: CW8, TMO
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Selective Small Molecule Inhibition Of The Fmn Riboswitch
Organism: Fusobacterium nucleatum
Method: X-RAY DIFFRACTION Resolution:2.93 Å Release Date: 2015-10-07 Classification: RNA/INHIBITOR Ligands: K, MG, 51B |
Organism: Fusobacterium nucleatum
Method: X-RAY DIFFRACTION
Release Date: 2015-10-07
Ligands: K, MG, 51B
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Structure And Function Of The Hypertension Variant A486V Of G Protein-Coupled Receptor Kinase 4 (Grk4)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2015-07-08 Classification: TRANSFERASE Ligands: AN2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-08
Ligands: AN2
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The Structure Of Trka Kinase Bound To The Inhibitor N-(3-Cyclopropyl-1-Phenyl-1H-Pyrazol-5-Yl)-2-{4-[3-Methoxy-4-(4-Methyl-1H-Imidazol-1-Yl)Phenyl]-1H-1,2,3-Triazol-1-Yl}Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2014-06-18 Classification: Transferase/Transferase inhibitor Ligands: 31V, GOL, CL, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-06-18
Ligands: 31V, GOL, CL, ACT
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The Structure Of Trka Kinase Bound To The Inhibitor 1-Cyclopropyl-1-[3-(1,3-Thiazol-2-Yl)Benzyl]-3-[4-(Trifluoromethoxy)Phenyl]Urea
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2014-06-18 Classification: Transferase/Transferase inhibitor Ligands: 31W, CL, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-06-18
Ligands: 31W, CL, ACT
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The Structure Of Trka Kinase Bound To The Inhibitor 4-Naphthalen-1-Yl-1-[(5-Phenyl-1,2,4-Oxadiazol-3-Yl)Methyl]-1H-Pyrrolo[3,2-C]Pyridine-2-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2014-06-18 Classification: Transferase/Transferase inhibitor Ligands: 31X, CL, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-06-18
Ligands: 31X, CL, ACT
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The Structure Of Trka Kinase Bound To The Inhibitor N~4~-(4-Morpholin-4-Ylphenyl)-N~6~-(Pyridin-3-Ylmethyl)Pyrido[3,2-D]Pyrimidine-4,6-Diamine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2014-06-18 Classification: Transferase/Transferase inhibitor Ligands: 31Y, CL, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-06-18
Ligands: 31Y, CL, ACT
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Discovery Of Pyrrolidine-Based B-Secretase Inhibitors: Lead Advancement Through Conformational Design For Maintenance Of Ligand Binding Efficiency
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2012-01-18 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 508, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-01-18
Ligands: 508, SO4, GOL
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Discovery Of Aminoheterocycles As A Novel Beta-Secretase Inhibitor Class
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2009-07-07 Classification: HYDROLASE Ligands: B35 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-07-07
Ligands: B35
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Crystal Structure Of Bace1 Bound To Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2009-02-03 Classification: HYDROLASE Ligands: SO4, GOL, 5MS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-02-03
Ligands: SO4, GOL, 5MS
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Crystal Structure Of Chk1 Kinase In Complex With Inhibitor 38
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2009-01-20 Classification: TRANSFERASE Ligands: 38M, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-01-20
Ligands: 38M, SO4
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Crystal Structure Of Human Beta Secretase Complexed With Spiropiperdine Iminohydantoin Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2009-01-20 Classification: HYDROLASE Ligands: SII |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-01-20
Ligands: SII
